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Beta-1 adrenergic receptor Inhibitors (IC50, Ki)

Structure
▲
▼
Compound Name
▲
▼
Standard Type
▲
▼
Standard Values (in nM)
▲
▼
AtenololIC501.77 [1], 1640.0 [2], 1740.0 [3]
AtenololKi170.0 [1], 430.0 [2], 758.0 [3], 1513.56 [4]
SalmeterolIC50501.19 [1]
SalmeterolKi784.0 [1], 801.0 [2], 2300.0 [3], 2511.89 [4]
PropranololIC5018.0 [1], 251.19 [2]
PropranololKi1.47 [1], 2.3 [2], 11.75 [3]
FormoterolIC50630.96 [1]
FormoterolKi315.0 [1], 319.0 [2], 1995.26 [3]
SotalolIC508900.0 [1], 9000.0 [2]
SotalolKi833.5 [1]
IndacaterolIC50316.23 [1]
IndacaterolKi91.0 [1], 91.4 [2]
2-(4-((2R)-2-(((2R)-2-(3-Chlorophenyl)-2-hydroxyethyl)amino)propyl)phenoxy)acetic acidIC505000.0 [1]
2-(4-((2R)-2-(((2R)-2-(3-Chlorophenyl)-2-hydroxyethyl)amino)propyl)phenoxy)acetic acidKi1130.0 [1], 11300.0 [2]
1-[(3,4,5-Trimethoxyphenyl)methyl]-1,2,3,4-tetrahydroisoquinoline-6,7-diolIC506.1 [1]
1-[(3,4,5-Trimethoxyphenyl)methyl]-1,2,3,4-tetrahydroisoquinoline-6,7-diolKi323.59 [1]
SibenadetIC5010000.0 [1]
SibenadetKi3922.0 [1]
L-796568 Free baseIC501000.0 [1], 2300.0 [2]
2-(2-Amino-1,3-thiazol-4-yl)-N-[4-[[(2S,5R)-5-[(R)-hydroxy(phenyl)methyl]pyrrolidin-2-yl]methyl]phenyl]acetamideIC5020000.0 [1]
(6Ar,7R)-1,2-dimethoxy-5,6,6a,7-tetrahydro-4H-dibenzo[de,g]quinolin-7-olIC501.7 [1], 17.0 [2]
(6Ar,7R)-1,2-dimethoxy-5,6,6a,7-tetrahydro-4H-dibenzo[de,g]quinolin-7-olKi19.0 [1]
IsoprenalineKi193.0 [1], 1584.89 [2]
PindololKi0.52 [1], 0.53 [2]
TimololKi1.5 [1], 5.37 [2]
DarifenacinIC50316.23 [1]
DarifenacinKi180.0 [1]
1-(Isopropylamino)-3-(1-naphthyloxy)-2-propanolIC502.5 [1]
1-(Isopropylamino)-3-(1-naphthyloxy)-2-propanolKi1.1 [1]
1-PhenylpiperazineIC5019000.0 [1]
1-PhenylpiperazineKi1348.96 [1]
CID 9829836IC50200.0 [1]
CID 9829836Ki570.0 [1]
4-Methyl-2-piperazin-1-yl-quinolineKi220.0 [1], 223.87 [2]
4-(3-Hexyl-2-oxoimidazol-1-yl)-N-[4-[2-[[(2R)-2-hydroxy-2-pyridin-3-ylethyl]amino]ethyl]phenyl]benzenesulfonamideIC5018000.0 [1]
4-(1-Piperazinyl)-1H-indoleKi67.61 [1], 68.0 [2]
1-Hexyl-3-[4-[[4-[2-[[(2R)-2-hydroxy-2-pyridin-3-ylethyl]amino]ethyl]phenyl]sulfamoyl]phenyl]ureaIC508000.0 [1]
4-(3-Hexyl-2-oxoimidazolidin-1-yl)-N-[4-[2-[[(2R)-2-hydroxy-2-pyridin-3-ylethyl]amino]ethyl]phenyl]benzenesulfonamideIC505000.0 [1]
1-(3,5-Diiodo-4-methoxybenzyl)-1,2,3,4-tetrahydroisoquinoline-6,7-diolKi2.04 [1], 79.43 [2]
[3-[(2R)-2-[[(2R)-2-Hydroxy-2-[3-(thiophen-2-ylsulfonylamino)phenyl]ethyl]amino]propyl]-1H-indol-7-yl] methanesulfonateKi66.0 [1]
N-[4-[2-[[(2R)-2-Hydroxy-2-pyridin-3-ylethyl]amino]ethyl]phenyl]-4-(3-octyl-2-oxoimidazolidin-1-yl)benzenesulfonamideIC50580.0 [1]
CID 16118894IC50170.0 [1]
N-[4-[2-[[(2R)-2-Hydroxy-2-pyridin-3-ylethyl]amino]ethyl]phenyl]-4-(3-octyl-2-oxoimidazol-1-yl)benzenesulfonamideIC505500.0 [1]
7-((R)-2-((1S,2S)-2-(Benzyloxy)cyclopentylamino)-1-hydroxyethyl)-4-hydroxybenzo[d]thiazol-2(3H)-oneKi70.0 [1], 107.0 [2]
4-[4-(3,4-Difluorophenyl)-1,3-thiazol-2-yl]-N-[4-[2-[[(2R)-2-hydroxy-2-pyridin-3-ylethyl]amino]ethyl]phenyl]benzenesulfonamideIC501700.0 [1]
7-[(1R)-2-[[(1R,2R)-2-Cyclopentylcyclopentyl]amino]-1-hydroxyethyl]-4-hydroxy-3H-1,3-benzothiazol-2-oneKi17.0 [1], 17.8 [2]
(6S)-N-[4-[[(2S,5R)-5-[(R)-Hydroxy(pyridin-3-yl)methyl]pyrrolidin-2-yl]methyl]phenyl]-5,6-dihydro-4H-pyrrolo[1,2-b]pyrazole-6-carboxamideIC5020000.0 [1]
(4R)-N-[4-[[(2S,5R)-5-[(R)-Hydroxy(pyridin-3-yl)methyl]pyrrolidin-2-yl]methyl]phenyl]-5,6-dihydro-4H-cyclopenta[d][1,3]thiazole-4-carboxamideIC5020000.0 [1]
4-(3,5-Diiodo-4-methoxybenzyl)-4,5,6,7-tetrahydrothiazolo[5,4-c]pyridine-2-amineIC50780.0 [1]
4-(3,5-Diiodo-4-methoxybenzyl)-4,5,6,7-tetrahydrothiazolo[5,4-c]pyridine-2-amineKi724.44 [1]
Ethyl (1S,5R)-3-[4-[[(2S,5R)-5-[(R)-hydroxy(phenyl)methyl]pyrrolidin-2-yl]methyl]benzoyl]-3-azabicyclo[3.1.0]hexane-6-carboxylateIC5020000.0 [1]
2-[[1-[2-Hydroxy-3-(5-methyl-2-propan-2-ylphenoxy)propyl]piperidin-4-yl]methyl]benzo[de]isoquinoline-1,3-dioneIC50377.0 [1]
2-[[1-[2-Hydroxy-3-(5-methyl-2-propan-2-ylphenoxy)propyl]piperidin-4-yl]methyl]benzo[de]isoquinoline-1,3-dioneKi1000.0 [1]
DexpropranololKi214.0 [1]
TamoxifenKi9984.0 [1]
AmiodaroneKi25202.0 [1]
DiethylstilbestrolKi12755.0 [1]
BromocriptineKi1386.0 [1]
MetoprololKi102.0 [1]
DobutamineKi1123.0 [1]
LysergideKi140.0 [1]
CarvedilolKi0.1 [1]
MiconazoleKi7296.0 [1]
ClotrimazoleKi6513.0 [1]
LabetalolKi5.84 [1]
ErgotamineKi2392.0 [1]
CisaprideIC5010000.0 [1]
PropafenoneKi205.0 [1]
ClenbuterolKi69.0 [1]
AlprenololIC504.88 [1]
HarmineKi10000.0 [1]
1-(3-Chlorophenyl)piperazineIC502000.0 [1]
AcebutololKi422.0 [1]
EsmololKi113.7 [1]
LisurideKi323.0 [1]
AstemizoleKi10037.0 [1]
EconazoleKi7404.0 [1]
QuipazineKi6309.57 [1]
BetaxololIC5037.1 [1]
4-[(2S)-3-(Tert-butylamino)-2-hydroxypropoxy]-1,3-dihydrobenzimidazol-2-oneKi0.25 [1]
CarteololKi1.9 [1]
LevobunololKi3.98 [1]
Cl-316243 Free diacidKi100000.0 [1]
BopindololKi27.0 [1]
1-(2-Methoxyphenyl)piperazineIC502000.0 [1]
(+)-DihydrexidineKi1500.0 [1]
SB 224289Ki1000.0 [1]
alpha-MethyltryptamineKi3801.89 [1]
SB 204070 hydrochlorideKi1000.0 [1]
CipargaminIC5010000.0 [1]
(4-{(R)-2-[(R)-2-(3-Chloro-phenyl)-2-hydroxy-ethylamino]-propyl}-phenoxy)-acetic acid methyl esterKi170.0 [1]
(S)-(-)-PindololKi0.43 [1]
ClorprenalineKi1497.0 [1]
4-(4-Butylpiperidin-1-yl)-1-o-tolylbutan-1-oneKi1000.0 [1]
4-Amino-5-chloro-N-((hexahydro-1H-pyrrolizin-1-yl)methyl)-2-methoxybenzamide hydrochlorideIC5010000.0 [1]
1-[3-(4-Butylpiperidino)propyl]-3,4-dihydroquinoline-2(1H)-oneKi47863.01 [1]
1-(4-Methoxyphenyl)piperazineIC5038000.0 [1]
SolabegronKi398.11 [1]
Benzonitrile, 3-fluoro-5-(2-(2-(fluoromethyl)-4-thiazolyl)ethynyl)-Ki10000.0 [1]
VibegronIC5020000.0 [1]
Items per page: 1 - 10 of 100
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References

This online tool may be cited as follows

MLA

"Quest Database™ Beta-1 adrenergic receptor Inhibitors (IC50, Ki)." AAT Bioquest, Inc., 21 Feb. 2025, https://www.aatbio.com/data-sets/beta-1-adrenergic-receptor-inhibitors-ic50-ki.

APA

AAT Bioquest, Inc. (2025, February 21). Quest Database™ Beta-1 adrenergic receptor Inhibitors (IC50, Ki). AAT Bioquest. https://www.aatbio.com/data-sets/beta-1-adrenergic-receptor-inhibitors-ic50-ki.
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