![](https://images.aatbio.com/dataset/ic50/beta-1-adrenergic-receptor_faac9f61879fd14d1ee20cc8818ffd60.svg) | Atenolol | IC50 | 1.77 [1], 1640.0 [2], 1740.0 [3] |
![](https://images.aatbio.com/dataset/ic50/beta-1-adrenergic-receptor_faac9f61879fd14d1ee20cc8818ffd60.svg) | Atenolol | Ki | 170.0 [1], 430.0 [2], 758.0 [3], 1513.56 [4] |
![](https://images.aatbio.com/dataset/ic50/beta-1-adrenergic-receptor_0b1e406a221d2c8c7961dd461e08e86f.svg) | Salmeterol | IC50 | 501.19 [1] |
![](https://images.aatbio.com/dataset/ic50/beta-1-adrenergic-receptor_0b1e406a221d2c8c7961dd461e08e86f.svg) | Salmeterol | Ki | 784.0 [1], 801.0 [2], 2300.0 [3], 2511.89 [4] |
![](https://images.aatbio.com/dataset/ic50/beta-1-adrenergic-receptor_c70f5b79af37726016ec15cea0b55e94.svg) | Propranolol | IC50 | 18.0 [1], 251.19 [2] |
![](https://images.aatbio.com/dataset/ic50/beta-1-adrenergic-receptor_c70f5b79af37726016ec15cea0b55e94.svg) | Propranolol | Ki | 1.47 [1], 2.3 [2], 11.75 [3] |
![](https://images.aatbio.com/dataset/ic50/beta-1-adrenergic-receptor_79ff1a8f4ced1806080b29930fcdd199.svg) | Formoterol | IC50 | 630.96 [1] |
![](https://images.aatbio.com/dataset/ic50/beta-1-adrenergic-receptor_79ff1a8f4ced1806080b29930fcdd199.svg) | Formoterol | Ki | 315.0 [1], 319.0 [2], 1995.26 [3] |
![](https://images.aatbio.com/dataset/ic50/beta-1-adrenergic-receptor_9c9b6aadd4f8caa0bf86f9d7bbd70a7c.svg) | Sotalol | IC50 | 8900.0 [1], 9000.0 [2] |
![](https://images.aatbio.com/dataset/ic50/beta-1-adrenergic-receptor_9c9b6aadd4f8caa0bf86f9d7bbd70a7c.svg) | Sotalol | Ki | 833.5 [1] |
![](https://images.aatbio.com/dataset/ic50/beta-1-adrenergic-receptor_401e7d8739619d44f5d212db396141d1.svg) | Indacaterol | IC50 | 316.23 [1] |
![](https://images.aatbio.com/dataset/ic50/beta-1-adrenergic-receptor_401e7d8739619d44f5d212db396141d1.svg) | Indacaterol | Ki | 91.0 [1], 91.4 [2] |
![](https://images.aatbio.com/dataset/ic50/beta-1-adrenergic-receptor_72456aaaa543e799097de36c30caec7a.svg) | 2-(4-((2R)-2-(((2R)-2-(3-Chlorophenyl)-2-hydroxyethyl)amino)propyl)phenoxy)acetic acid | IC50 | 5000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/beta-1-adrenergic-receptor_72456aaaa543e799097de36c30caec7a.svg) | 2-(4-((2R)-2-(((2R)-2-(3-Chlorophenyl)-2-hydroxyethyl)amino)propyl)phenoxy)acetic acid | Ki | 1130.0 [1], 11300.0 [2] |
![](https://images.aatbio.com/dataset/ic50/beta-1-adrenergic-receptor_5ecfabed9d7ba5abe95feae80d831bd0.svg) | 1-[(3,4,5-Trimethoxyphenyl)methyl]-1,2,3,4-tetrahydroisoquinoline-6,7-diol | IC50 | 6.1 [1] |
![](https://images.aatbio.com/dataset/ic50/beta-1-adrenergic-receptor_5ecfabed9d7ba5abe95feae80d831bd0.svg) | 1-[(3,4,5-Trimethoxyphenyl)methyl]-1,2,3,4-tetrahydroisoquinoline-6,7-diol | Ki | 323.59 [1] |
![](https://images.aatbio.com/dataset/ic50/beta-1-adrenergic-receptor_7509c93b47093292622400bf49e18d93.svg) | Sibenadet | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/beta-1-adrenergic-receptor_7509c93b47093292622400bf49e18d93.svg) | Sibenadet | Ki | 3922.0 [1] |
![](https://images.aatbio.com/dataset/ic50/beta-1-adrenergic-receptor_9182e75261c4c9a90083bb44381e7fec.svg) | L-796568 Free base | IC50 | 1000.0 [1], 2300.0 [2] |
![](https://images.aatbio.com/dataset/ic50/beta-1-adrenergic-receptor_99f04051f3a3c2e2d86079a90b1965c9.svg) | 2-(2-Amino-1,3-thiazol-4-yl)-N-[4-[[(2S,5R)-5-[(R)-hydroxy(phenyl)methyl]pyrrolidin-2-yl]methyl]phenyl]acetamide | IC50 | 20000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/beta-1-adrenergic-receptor_9744b3d5a6c31103aec2468ffba68afd.svg) | (6Ar,7R)-1,2-dimethoxy-5,6,6a,7-tetrahydro-4H-dibenzo[de,g]quinolin-7-ol | IC50 | 1.7 [1], 17.0 [2] |
![](https://images.aatbio.com/dataset/ic50/beta-1-adrenergic-receptor_9744b3d5a6c31103aec2468ffba68afd.svg) | (6Ar,7R)-1,2-dimethoxy-5,6,6a,7-tetrahydro-4H-dibenzo[de,g]quinolin-7-ol | Ki | 19.0 [1] |
![](https://images.aatbio.com/dataset/ic50/beta-1-adrenergic-receptor_0f316e08160d2999e6ea804928aa42e0.svg) | Isoprenaline | Ki | 193.0 [1], 1584.89 [2] |
![](https://images.aatbio.com/dataset/ic50/beta-1-adrenergic-receptor_7ba45ba2f8b56f9250d9067912b4ab0b.svg) | Pindolol | Ki | 0.52 [1], 0.53 [2] |
![](https://images.aatbio.com/dataset/ic50/beta-1-adrenergic-receptor_90fc937ca80a4f307c8f0c3397d5e0f0.svg) | Timolol | Ki | 1.5 [1], 5.37 [2] |
![](https://images.aatbio.com/dataset/ic50/beta-1-adrenergic-receptor_2caadd3ec7b2c08ae34435ae889a6a0b.svg) | Darifenacin | IC50 | 316.23 [1] |
![](https://images.aatbio.com/dataset/ic50/beta-1-adrenergic-receptor_2caadd3ec7b2c08ae34435ae889a6a0b.svg) | Darifenacin | Ki | 180.0 [1] |
![](https://images.aatbio.com/dataset/ic50/beta-1-adrenergic-receptor_f8aba9f3e7e7e52b2b80d93116b3a61f.svg) | 1-(Isopropylamino)-3-(1-naphthyloxy)-2-propanol | IC50 | 2.5 [1] |
![](https://images.aatbio.com/dataset/ic50/beta-1-adrenergic-receptor_f8aba9f3e7e7e52b2b80d93116b3a61f.svg) | 1-(Isopropylamino)-3-(1-naphthyloxy)-2-propanol | Ki | 1.1 [1] |
![](https://images.aatbio.com/dataset/ic50/beta-1-adrenergic-receptor_5ca006686077869ce71ef3ba92f19c4b.svg) | 1-Phenylpiperazine | IC50 | 19000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/beta-1-adrenergic-receptor_5ca006686077869ce71ef3ba92f19c4b.svg) | 1-Phenylpiperazine | Ki | 1348.96 [1] |
![](https://images.aatbio.com/dataset/ic50/beta-1-adrenergic-receptor_77389a2801f3f65ad7dd698c44ce344c.svg) | CID 9829836 | IC50 | 200.0 [1] |
![](https://images.aatbio.com/dataset/ic50/beta-1-adrenergic-receptor_77389a2801f3f65ad7dd698c44ce344c.svg) | CID 9829836 | Ki | 570.0 [1] |
![](https://images.aatbio.com/dataset/ic50/beta-1-adrenergic-receptor_824101334aceee05a0a19e8d83914735.svg) | 4-Methyl-2-piperazin-1-yl-quinoline | Ki | 220.0 [1], 223.87 [2] |
![](https://images.aatbio.com/dataset/ic50/beta-1-adrenergic-receptor_1c659afb0f779ac15328cb556219387a.svg) | 4-(3-Hexyl-2-oxoimidazol-1-yl)-N-[4-[2-[[(2R)-2-hydroxy-2-pyridin-3-ylethyl]amino]ethyl]phenyl]benzenesulfonamide | IC50 | 18000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/beta-1-adrenergic-receptor_0f3d930da4d764c4bb9f7b0c1f35b8a5.svg) | 4-(1-Piperazinyl)-1H-indole | Ki | 67.61 [1], 68.0 [2] |
![](https://images.aatbio.com/dataset/ic50/beta-1-adrenergic-receptor_35015a3a7e91981c9ac0411f78b352b7.svg) | 1-Hexyl-3-[4-[[4-[2-[[(2R)-2-hydroxy-2-pyridin-3-ylethyl]amino]ethyl]phenyl]sulfamoyl]phenyl]urea | IC50 | 8000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/beta-1-adrenergic-receptor_a43f6005721c3392a7794fcc40d79826.svg) | 4-(3-Hexyl-2-oxoimidazolidin-1-yl)-N-[4-[2-[[(2R)-2-hydroxy-2-pyridin-3-ylethyl]amino]ethyl]phenyl]benzenesulfonamide | IC50 | 5000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/beta-1-adrenergic-receptor_ae1260fb5a29888431ee8d07c9f8d636.svg) | 1-(3,5-Diiodo-4-methoxybenzyl)-1,2,3,4-tetrahydroisoquinoline-6,7-diol | Ki | 2.04 [1], 79.43 [2] |
![](https://images.aatbio.com/dataset/ic50/beta-1-adrenergic-receptor_0376c90955414a1d4ca596b3885abe22.svg) | [3-[(2R)-2-[[(2R)-2-Hydroxy-2-[3-(thiophen-2-ylsulfonylamino)phenyl]ethyl]amino]propyl]-1H-indol-7-yl] methanesulfonate | Ki | 66.0 [1] |
![](https://images.aatbio.com/dataset/ic50/beta-1-adrenergic-receptor_d3c2de7965cf3b7a3390588074cd1be4.svg) | N-[4-[2-[[(2R)-2-Hydroxy-2-pyridin-3-ylethyl]amino]ethyl]phenyl]-4-(3-octyl-2-oxoimidazolidin-1-yl)benzenesulfonamide | IC50 | 580.0 [1] |
![](https://images.aatbio.com/dataset/ic50/beta-1-adrenergic-receptor_b9052dd293ceb39192e43d89b3c1e26c.svg) | CID 16118894 | IC50 | 170.0 [1] |
![](https://images.aatbio.com/dataset/ic50/beta-1-adrenergic-receptor_96c1edb906479ed0ab40654c1dda160b.svg) | N-[4-[2-[[(2R)-2-Hydroxy-2-pyridin-3-ylethyl]amino]ethyl]phenyl]-4-(3-octyl-2-oxoimidazol-1-yl)benzenesulfonamide | IC50 | 5500.0 [1] |
![](https://images.aatbio.com/dataset/ic50/beta-1-adrenergic-receptor_9a9877a4c06d68b876831ac2faa1633b.svg) | 7-((R)-2-((1S,2S)-2-(Benzyloxy)cyclopentylamino)-1-hydroxyethyl)-4-hydroxybenzo[d]thiazol-2(3H)-one | Ki | 70.0 [1], 107.0 [2] |
![](https://images.aatbio.com/dataset/ic50/beta-1-adrenergic-receptor_147e629938e079c1fe13f62367c5be8a.svg) | 4-[4-(3,4-Difluorophenyl)-1,3-thiazol-2-yl]-N-[4-[2-[[(2R)-2-hydroxy-2-pyridin-3-ylethyl]amino]ethyl]phenyl]benzenesulfonamide | IC50 | 1700.0 [1] |
![](https://images.aatbio.com/dataset/ic50/beta-1-adrenergic-receptor_897c90be6f0b54afe7dd9d619ae3bc59.svg) | 7-[(1R)-2-[[(1R,2R)-2-Cyclopentylcyclopentyl]amino]-1-hydroxyethyl]-4-hydroxy-3H-1,3-benzothiazol-2-one | Ki | 17.0 [1], 17.8 [2] |
![](https://images.aatbio.com/dataset/ic50/beta-1-adrenergic-receptor_5d76064ddc2dff8b46597ab1ba156fa1.svg) | (6S)-N-[4-[[(2S,5R)-5-[(R)-Hydroxy(pyridin-3-yl)methyl]pyrrolidin-2-yl]methyl]phenyl]-5,6-dihydro-4H-pyrrolo[1,2-b]pyrazole-6-carboxamide | IC50 | 20000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/beta-1-adrenergic-receptor_722c621ffb02e379ed12b3dedfac01e8.svg) | (4R)-N-[4-[[(2S,5R)-5-[(R)-Hydroxy(pyridin-3-yl)methyl]pyrrolidin-2-yl]methyl]phenyl]-5,6-dihydro-4H-cyclopenta[d][1,3]thiazole-4-carboxamide | IC50 | 20000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/beta-1-adrenergic-receptor_c9a0c15c13f721a0f2337b7fea62daca.svg) | 4-(3,5-Diiodo-4-methoxybenzyl)-4,5,6,7-tetrahydrothiazolo[5,4-c]pyridine-2-amine | IC50 | 780.0 [1] |
![](https://images.aatbio.com/dataset/ic50/beta-1-adrenergic-receptor_c9a0c15c13f721a0f2337b7fea62daca.svg) | 4-(3,5-Diiodo-4-methoxybenzyl)-4,5,6,7-tetrahydrothiazolo[5,4-c]pyridine-2-amine | Ki | 724.44 [1] |
![](https://images.aatbio.com/dataset/ic50/beta-1-adrenergic-receptor_1ab128e95c5a93c9f00ec10177d1795d.svg) | Ethyl (1S,5R)-3-[4-[[(2S,5R)-5-[(R)-hydroxy(phenyl)methyl]pyrrolidin-2-yl]methyl]benzoyl]-3-azabicyclo[3.1.0]hexane-6-carboxylate | IC50 | 20000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/beta-1-adrenergic-receptor_d5e2cd733d4afe021c278ea28af921da.svg) | 2-[[1-[2-Hydroxy-3-(5-methyl-2-propan-2-ylphenoxy)propyl]piperidin-4-yl]methyl]benzo[de]isoquinoline-1,3-dione | IC50 | 377.0 [1] |
![](https://images.aatbio.com/dataset/ic50/beta-1-adrenergic-receptor_d5e2cd733d4afe021c278ea28af921da.svg) | 2-[[1-[2-Hydroxy-3-(5-methyl-2-propan-2-ylphenoxy)propyl]piperidin-4-yl]methyl]benzo[de]isoquinoline-1,3-dione | Ki | 1000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/beta-1-adrenergic-receptor_32a0612a648044dbc4831a7d07460b80.svg) | Dexpropranolol | Ki | 214.0 [1] |
![](https://images.aatbio.com/dataset/ic50/beta-1-adrenergic-receptor_f28ce47318433f5c984060ce11c4a797.svg) | Tamoxifen | Ki | 9984.0 [1] |
![](https://images.aatbio.com/dataset/ic50/beta-1-adrenergic-receptor_81af8877c0a8c32165f86d729092ee41.svg) | Amiodarone | Ki | 25202.0 [1] |
![](https://images.aatbio.com/dataset/ic50/beta-1-adrenergic-receptor_adf25e33d7987b11abe6dedf76999efd.svg) | Diethylstilbestrol | Ki | 12755.0 [1] |
![](https://images.aatbio.com/dataset/ic50/beta-1-adrenergic-receptor_b245c9e25780678ea441c35a3d085042.svg) | Bromocriptine | Ki | 1386.0 [1] |
![](https://images.aatbio.com/dataset/ic50/beta-1-adrenergic-receptor_b7b8a734145b81caa9a4a7ab9953506c.svg) | Metoprolol | Ki | 102.0 [1] |
![](https://images.aatbio.com/dataset/ic50/beta-1-adrenergic-receptor_69f1e2f0b60a6951de28604d3a1311ba.svg) | Dobutamine | Ki | 1123.0 [1] |
![](https://images.aatbio.com/dataset/ic50/beta-1-adrenergic-receptor_71814b7cfaffdb246739fb46903a8181.svg) | Lysergide | Ki | 140.0 [1] |
![](https://images.aatbio.com/dataset/ic50/beta-1-adrenergic-receptor_22ca1744345a750f98669f67193f6275.svg) | Carvedilol | Ki | 0.1 [1] |
![](https://images.aatbio.com/dataset/ic50/beta-1-adrenergic-receptor_b4f76a216efed394b41035ecb49dec98.svg) | Miconazole | Ki | 7296.0 [1] |
![](https://images.aatbio.com/dataset/ic50/beta-1-adrenergic-receptor_6c5a78e8ca55529a3f6c3b506ecb26d6.svg) | Clotrimazole | Ki | 6513.0 [1] |
![](https://images.aatbio.com/dataset/ic50/beta-1-adrenergic-receptor_92de0750be5ed5be0d0c9ea65877cc94.svg) | Labetalol | Ki | 5.84 [1] |
![](https://images.aatbio.com/dataset/ic50/beta-1-adrenergic-receptor_450c13a75b3dc6366b9bf225bd270c46.svg) | Ergotamine | Ki | 2392.0 [1] |
![](https://images.aatbio.com/dataset/ic50/beta-1-adrenergic-receptor_01a74ff12e6bf089ced324ef974b490e.svg) | Cisapride | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/beta-1-adrenergic-receptor_89fd1058473b46f547fd6ef0c68156d1.svg) | Propafenone | Ki | 205.0 [1] |
![](https://images.aatbio.com/dataset/ic50/beta-1-adrenergic-receptor_92d5e1170d4cc2a475fe08d4ff8a00c8.svg) | Clenbuterol | Ki | 69.0 [1] |
![](https://images.aatbio.com/dataset/ic50/beta-1-adrenergic-receptor_21a5e343431c845430d5c459f3e32ffb.svg) | Alprenolol | IC50 | 4.88 [1] |
![](https://images.aatbio.com/dataset/ic50/beta-1-adrenergic-receptor_227772c6b35181ad4f999c7ec25d9175.svg) | Harmine | Ki | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/beta-1-adrenergic-receptor_4b9c1f50c88f6f316f4ab191bc3b47c0.svg) | 1-(3-Chlorophenyl)piperazine | IC50 | 2000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/beta-1-adrenergic-receptor_e2827ec41e052d65c1bbfd99d08fc9a9.svg) | Acebutolol | Ki | 422.0 [1] |
![](https://images.aatbio.com/dataset/ic50/beta-1-adrenergic-receptor_15457e4c21c33a24f91603d479b4d435.svg) | Esmolol | Ki | 113.7 [1] |
![](https://images.aatbio.com/dataset/ic50/beta-1-adrenergic-receptor_3b7395ec254589f5d3f9a4cc5434da86.svg) | Lisuride | Ki | 323.0 [1] |
![](https://images.aatbio.com/dataset/ic50/beta-1-adrenergic-receptor_f67d9004e24bf13185c0a0543b060ab0.svg) | Astemizole | Ki | 10037.0 [1] |
![](https://images.aatbio.com/dataset/ic50/beta-1-adrenergic-receptor_0e06682e28b9fadd6faa1c46a98e31f5.svg) | Econazole | Ki | 7404.0 [1] |
![](https://images.aatbio.com/dataset/ic50/beta-1-adrenergic-receptor_8a8d97b767839368361933650518caa1.svg) | Quipazine | Ki | 6309.57 [1] |
![](https://images.aatbio.com/dataset/ic50/beta-1-adrenergic-receptor_4f2f56c4220db9379d1f14f08c53f040.svg) | Betaxolol | IC50 | 37.1 [1] |
![](https://images.aatbio.com/dataset/ic50/beta-1-adrenergic-receptor_dcb6fe4082f8fb0defd50ea385ab64f9.svg) | 4-[(2S)-3-(Tert-butylamino)-2-hydroxypropoxy]-1,3-dihydrobenzimidazol-2-one | Ki | 0.25 [1] |
![](https://images.aatbio.com/dataset/ic50/beta-1-adrenergic-receptor_bb1c6343edb378e5deabb6618f62dc47.svg) | Carteolol | Ki | 1.9 [1] |
![](https://images.aatbio.com/dataset/ic50/beta-1-adrenergic-receptor_4670f48ea07e5f4dfa8a4f044b78a0df.svg) | Levobunolol | Ki | 3.98 [1] |
![](https://images.aatbio.com/dataset/ic50/beta-1-adrenergic-receptor_e692cf5147fd5e48089d97db374b47b8.svg) | Cl-316243 Free diacid | Ki | 100000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/beta-1-adrenergic-receptor_c7700b890db794d7c22ab266a229bb5b.svg) | Bopindolol | Ki | 27.0 [1] |
![](https://images.aatbio.com/dataset/ic50/beta-1-adrenergic-receptor_dd63cc5758f16c2a47660cbe0516a008.svg) | 1-(2-Methoxyphenyl)piperazine | IC50 | 2000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/beta-1-adrenergic-receptor_69cdad9a7cffce891b22d99e3d466366.svg) | (+)-Dihydrexidine | Ki | 1500.0 [1] |
![](https://images.aatbio.com/dataset/ic50/beta-1-adrenergic-receptor_5bfc996f8d242d6ccd706830c48cb90d.svg) | SB 224289 | Ki | 1000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/beta-1-adrenergic-receptor_889c75941cc4ae0a55b6d028f9169fbd.svg) | alpha-Methyltryptamine | Ki | 3801.89 [1] |
![](https://images.aatbio.com/dataset/ic50/beta-1-adrenergic-receptor_c309ec30409c0092587bfcf4b098e4de.svg) | SB 204070 hydrochloride | Ki | 1000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/beta-1-adrenergic-receptor_e39e3bc989cee0b1a0a409acf38c8621.svg) | Cipargamin | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/beta-1-adrenergic-receptor_6de12df8c12a625b9ea568beff3bccc5.svg) | (4-{(R)-2-[(R)-2-(3-Chloro-phenyl)-2-hydroxy-ethylamino]-propyl}-phenoxy)-acetic acid methyl ester | Ki | 170.0 [1] |
![](https://images.aatbio.com/dataset/ic50/beta-1-adrenergic-receptor_5891a040fd88cee28fafc55091d0e612.svg) | (S)-(-)-Pindolol | Ki | 0.43 [1] |
![](https://images.aatbio.com/dataset/ic50/beta-1-adrenergic-receptor_9eb6a66c29679c2b8beec909e0d0298b.svg) | Clorprenaline | Ki | 1497.0 [1] |
![](https://images.aatbio.com/dataset/ic50/beta-1-adrenergic-receptor_90fb2a3a66730e2f70a5255e06106c8e.svg) | 4-(4-Butylpiperidin-1-yl)-1-o-tolylbutan-1-one | Ki | 1000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/beta-1-adrenergic-receptor_df20649e63f6814da658fbc9fd2ea41a.svg) | 4-Amino-5-chloro-N-((hexahydro-1H-pyrrolizin-1-yl)methyl)-2-methoxybenzamide hydrochloride | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/beta-1-adrenergic-receptor_cf93aa4f7751be8474321896d37c7b1a.svg) | 1-[3-(4-Butylpiperidino)propyl]-3,4-dihydroquinoline-2(1H)-one | Ki | 47863.01 [1] |
![](https://images.aatbio.com/dataset/ic50/beta-1-adrenergic-receptor_eb5f506f9aa282dac1c16f6df8d82d8c.svg) | 1-(4-Methoxyphenyl)piperazine | IC50 | 38000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/beta-1-adrenergic-receptor_b0c2d037b2c47e158c7b276a895192f6.svg) | Solabegron | Ki | 398.11 [1] |
![](https://images.aatbio.com/dataset/ic50/beta-1-adrenergic-receptor_5716523bfa5a770fcbe111ff599e0550.svg) | Benzonitrile, 3-fluoro-5-(2-(2-(fluoromethyl)-4-thiazolyl)ethynyl)- | Ki | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/beta-1-adrenergic-receptor_e58637f0d4a87ff8f46c8ad80ca08fcf.svg) | Vibegron | IC50 | 20000.0 [1] |