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Bcl-2-related protein A1 Inhibitors (IC50, Ki)

Structure
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Compound Name
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Standard Type
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Standard Values (in nM)
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5-Benzyl-2-(5-benzyl-1,4,6,7-tetrahydroxy-3-methylnaphthalen-2-yl)-3-methylnaphthalene-1,4,6,7-tetroneIC50122.0 [1], 650.0 [2]
5-Benzyl-2-(5-benzyl-1,4,6,7-tetrahydroxy-3-methylnaphthalen-2-yl)-3-methylnaphthalene-1,4,6,7-tetroneKi430.0 [1]
ApogossypoloneIC502170.0 [1]
ApogossypoloneKi1470.0 [1]
2,3,5-Trihydroxy-7-methyl-N-(2-phenylpropyl)-6-[1,6,7-trihydroxy-3-methyl-5-(2-phenylpropylcarbamoyl)naphthalen-2-yl]naphthalene-1-carboxamideIC50420.0 [1], 730.0 [2]
3-Chloro-1-(3,4-dichlorophenyl)-4-morpholino-1H-pyrrole-2,5-dioneIC50450.0 [1], 800.0 [2]
3-Chloro-1-(3,4-dichlorophenyl)-4-(4-methylpiperazin-1-yl)pyrrole-2,5-dioneIC50600.0 [1], 800.0 [2]
3-Chloro-1-(3-chlorophenyl)-4-(4-methylpiperazin-1-yl)pyrrole-2,5-dioneIC501200.0 [1], 2100.0 [2]
3-Chloro-1-(3,4-dichlorophenyl)-4-(dimethylamino)pyrrole-2,5-dioneIC50300.0 [1], 400.0 [2]
CID 1180669IC5050000.0 [1]
3-Chloro-1-(3,4-dichlorophenyl)-4-piperidin-1-ylpyrrole-2,5-dioneIC5050000.0 [1]
N-[2-(4-Ethylphenyl)ethyl]-6-[5-[2-(4-ethylphenyl)ethylcarbamoyl]-3-methyl-1,4,6,7-tetraoxonaphthalen-2-yl]-2,3,5,8-tetrahydroxy-7-methylnaphthalene-1-carboxamideIC501250.0 [1]
N-[2-(4-Ethylphenyl)ethyl]-6-[5-[2-(4-ethylphenyl)ethylcarbamoyl]-3-methyl-1,4,6,7-tetraoxonaphthalen-2-yl]-2,3,5,8-tetrahydroxy-7-methylnaphthalene-1-carboxamideKi870.0 [1]
3-Methyl-5-(2-phenylacetyl)-2-[1,4,6,7-tetrahydroxy-3-methyl-5-(2-phenylacetyl)naphthalen-2-yl]naphthalene-1,4,6,7-tetroneIC50690.0 [1]
3-Methyl-5-(2-phenylacetyl)-2-[1,4,6,7-tetrahydroxy-3-methyl-5-(2-phenylacetyl)naphthalen-2-yl]naphthalene-1,4,6,7-tetroneKi460.0 [1]
2,3,5,8-Tetrahydroxy-7-methyl-6-[3-methyl-1,4,6,7-tetraoxo-5-(2-phenylpropylcarbamoyl)naphthalen-2-yl]-N-(2-phenylpropyl)naphthalene-1-carboxamideIC50710.0 [1]
2,3,5,8-Tetrahydroxy-7-methyl-6-[3-methyl-1,4,6,7-tetraoxo-5-(2-phenylpropylcarbamoyl)naphthalen-2-yl]-N-(2-phenylpropyl)naphthalene-1-carboxamideKi470.0 [1]
3-Methyl-5-(2-phenylethyl)-2-[1,4,6,7-tetrahydroxy-3-methyl-5-(2-phenylethyl)naphthalen-2-yl]naphthalene-1,4,6,7-tetroneIC509720.0 [1]
3-Methyl-5-(2-phenylethyl)-2-[1,4,6,7-tetrahydroxy-3-methyl-5-(2-phenylethyl)naphthalen-2-yl]naphthalene-1,4,6,7-tetroneKi6470.0 [1]
5-[(4-Chlorophenyl)methyl]-2-[5-[(4-chlorophenyl)methyl]-1,4,6,7-tetrahydroxy-3-methylnaphthalen-2-yl]-3-methylnaphthalene-1,4,6,7-tetroneIC50700.0 [1]
5-[(4-Chlorophenyl)methyl]-2-[5-[(4-chlorophenyl)methyl]-1,4,6,7-tetrahydroxy-3-methylnaphthalen-2-yl]-3-methylnaphthalene-1,4,6,7-tetroneKi470.0 [1]
3-Methyl-5-(2-methylpropyl)-2-[1,4,6,7-tetrahydroxy-3-methyl-5-(2-methylpropyl)naphthalen-2-yl]naphthalene-1,4,6,7-tetroneIC501410.0 [1]
3-Methyl-5-(2-methylpropyl)-2-[1,4,6,7-tetrahydroxy-3-methyl-5-(2-methylpropyl)naphthalen-2-yl]naphthalene-1,4,6,7-tetroneKi930.0 [1]
3-Methyl-5-[2-(4-methylphenyl)ethyl]-2-[1,4,6,7-tetrahydroxy-3-methyl-5-[2-(4-methylphenyl)ethyl]naphthalen-2-yl]naphthalene-1,4,6,7-tetroneIC5014700.0 [1]
3-Methyl-5-[2-(4-methylphenyl)ethyl]-2-[1,4,6,7-tetrahydroxy-3-methyl-5-[2-(4-methylphenyl)ethyl]naphthalen-2-yl]naphthalene-1,4,6,7-tetroneKi9330.0 [1]
3-Methyl-5-(3-phenylpropyl)-2-[1,4,6,7-tetrahydroxy-3-methyl-5-(3-phenylpropyl)naphthalen-2-yl]naphthalene-1,4,6,7-tetroneIC505270.0 [1]
3-Methyl-5-(3-phenylpropyl)-2-[1,4,6,7-tetrahydroxy-3-methyl-5-(3-phenylpropyl)naphthalen-2-yl]naphthalene-1,4,6,7-tetroneKi3530.0 [1]
3-Chloro-1-(3,4-dichlorophenyl)-4-(4-phenylpiperazin-1-yl)pyrrole-2,5-dioneIC504100.0 [1], 4900.0 [2]
3-Chloro-1-(3,5-dichlorophenyl)-4-(4-methylpiperazin-1-yl)pyrrole-2,5-dioneIC501900.0 [1], 2400.0 [2]
3-Chloro-1-(3,4-dichlorophenyl)-4-(pyrrolidino)-1H-pyrrole-2,5-dioneIC5050000.0 [1]
CID 16654638IC502600.0 [1], 8700.0 [2]
CID 16654639IC5011100.0 [1], 23900.0 [2]
3-Chloranyl-1-(2-chlorophenyl)-4-(4-methylpiperazin-1-yl)pyrrole-2,5-dioneIC501000.0 [1], 3300.0 [2]
3-Chloro-1-(3,4-dichlorophenyl)-4-[4-(3-methylphenyl)piperazin-1-yl]pyrrole-2,5-dioneIC5010000.0 [1]
CID 16654652IC50300.0 [1], 400.0 [2]
CID 16654653IC50600.0 [1], 800.0 [2]
3-Chloranyl-1-(3,4-dichlorophenyl)-4-[(3S)-3-methylpiperazin-1-yl]pyrrole-2,5-dioneIC501100.0 [1], 2200.0 [2]
CID 16654655IC50250.0 [1], 690.0 [2]
3-Chloranyl-1-(3,4-dichlorophenyl)-4-(4-ethylpiperazin-1-yl)pyrrole-2,5-dioneIC501000.0 [1], 1700.0 [2]
3-Chloro-1-(3,4-dichlorophenyl)-4-(4-piperonylpiperazino)-3-pyrroline-2,5-quinoneIC502100.0 [1], 4100.0 [2]
CID 16654662IC501300.0 [1], 2400.0 [2]
3-Chloro-1-(3,4-dichlorophenyl)-4-[4-[3-(trifluoromethyl)phenyl]piperazin-1-yl]pyrrole-2,5-dioneIC5010000.0 [1]
CID 16654669IC50240.0 [1], 620.0 [2]
CID 16654670IC506200.0 [1], 9600.0 [2]
CID 16654672IC508300.0 [1], 10000.0 [2]
CID 16654674IC503300.0 [1], 10500.0 [2]
CID 16654677IC501200.0 [1], 5000.0 [2]
CID 16654679IC502000.0 [1], 5600.0 [2]
CID 16654730IC5010800.0 [1], 12600.0 [2]
CID 16654772IC503900.0 [1], 6800.0 [2]
3-Chloro-1-(2,4-dichlorophenyl)-4-(4-methylpiperazin-1-yl)pyrrole-2,5-dioneIC501400.0 [1], 2600.0 [2]
1-(4-Chlorophenyl)-3-(4-methylpiperazin-1-yl)-1H-pyrrole-2,5-dioneIC5010000.0 [1]
1-(3,4-Dichlorophenyl)-3-(4-methylpiperazin-1-yl)pyrrolidine-2,5-dioneIC5010000.0 [1]
3-Chloro-1-(3,4-dichlorophenyl)-4-(2-hydroxyethylamino)pyrrole-2,5-dioneIC5050000.0 [1]
3-Chloro-1-(3-chloropyridin-4-yl)-4-(4-methylpiperazin-1-yl)pyrrole-2,5-dioneIC5029000.0 [1], 35600.0 [2]
Abt-737Ki20000.0 [1]
(2Z)-2-[(5Z)-5-[(3,5-Dimethyl-1H-pyrrol-2-yl)methylidene]-4-methoxypyrrol-2-ylidene]indoleKi1000.0 [1]
ApogossypolIC5010000.0 [1]
2-[4-[(4-Bromophenyl)sulfonylamino]-1-hydroxynaphthalen-2-yl]sulfanylacetic acidKi5330.0 [1]
SabutoclaxIC50620.0 [1]
2-(1-Hydroxy-4-(thiophene-2-sulfonamido)naphthalen-2-ylthio)acetic acidKi6140.0 [1]
2-[1-Hydroxy-4-[[(4-phenoxyphenyl)sulfonyl]amino]-2-naphthylthio]acetic acidKi3360.0 [1]
7-[1,3-Dimethyl-5-[[4-(4-methylsulfonylpiperazin-1-yl)phenoxy]methyl]pyrazol-4-yl]-1-(2-morpholin-4-ylethyl)-3-(3-naphthalen-1-yloxypropyl)indole-2-carboxylic acidKi660.0 [1]
(4S)-4-[[(2S)-2-[[(2S)-2-[[(2S,3S)-2-[[(2S)-2-[[(2S,3S)-2-Acetamido-3-methylpentanoyl]amino]-3-(prop-2-enoylamino)propanoyl]amino]-3-methylpentanoyl]amino]propanoyl]amino]-5-amino-5-oxopentanoyl]amino]-5-[[(2S)-1-[[(2S)-1-[[(3S,9S,12S,21S)-21-[[(2S)-1-[[(2S)-4-amino-1-[[(2S)-1-[[(2S)-1-[[(2S)-1-[[(2S)-1-[[(2S)-1-[[(2S)-1-amino-5-carbamimidamido-1-oxopentan-2-yl]amino]-5-carbamimidamido-1-oxopentan-2-yl]amino]-1-oxopropan-2-yl]amino]-3-(4-hydroxyphenyl)-1-oxopropan-2-yl]amino]-3-(4-hydroxyphenyl)-1-oxopropan-2-yl]amino]-1-oxopropan-2-yl]amino]-1,4-dioxobutan-2-yl]amino]-1-oxo-3-phenylpropan-2-yl]carbamoyl]-9-[(2S)-butan-2-yl]-3-(carboxymethyl)-12,21-dimethyl-2,5,8,11-tetraoxo-1,4,7,10-tetrazacyclohenicos-16-en-12-yl]amino]-5-carbamimidamido-1-oxopentan-2-yl]amino]-4-methyl-1-oxopentan-2-yl]amino]-5-oxopentanoic acidIC508.5 [1]
(4S)-4-[[(2S)-2-[[(2S)-2-[[(2S,3S)-2-[[(2S)-2-[[(2S,3S)-2-Acetamido-3-methylpentanoyl]amino]-3-(1H-indol-3-yl)propanoyl]amino]-3-methylpentanoyl]amino]propanoyl]amino]-5-amino-5-oxopentanoyl]amino]-5-[[(2S)-1-[[(2S)-1-[[(3S,9S,12S,21S)-21-[[(2S)-1-[[(2S)-4-amino-1-[[(2S)-1-[[(2S)-1-[[(2S)-1-[[(2S)-1-[[(2S)-1-[[(2S)-1-amino-5-carbamimidamido-1-oxopentan-2-yl]amino]-5-carbamimidamido-1-oxopentan-2-yl]amino]-1-oxopropan-2-yl]amino]-3-(4-hydroxyphenyl)-1-oxopropan-2-yl]amino]-3-(4-hydroxyphenyl)-1-oxopropan-2-yl]amino]-1-oxopropan-2-yl]amino]-1,4-dioxobutan-2-yl]amino]-1-oxo-3-phenylpropan-2-yl]carbamoyl]-9-[(2S)-butan-2-yl]-3-(carboxymethyl)-12,21-dimethyl-2,5,8,11-tetraoxo-1,4,7,10-tetrazacyclohenicos-16-en-12-yl]amino]-5-carbamimidamido-1-oxopentan-2-yl]amino]-4-methyl-1-oxopentan-2-yl]amino]-5-oxopentanoic acidIC50110.0 [1]
2,3,5-Trihydroxy-7-methyl-N-(2-phenylethyl)-6-[1,6,7-trihydroxy-3-methyl-5-(2-phenylethylcarbamoyl)naphthalen-2-yl]naphthalene-1-carboxamideIC50550.0 [1]
N-[2-(4-Ethylphenyl)ethyl]-6-[5-[2-(4-ethylphenyl)ethylcarbamoyl]-1,6,7-trihydroxy-3-methylnaphthalen-2-yl]-2,3,5-trihydroxy-7-methylnaphthalene-1-carboxamideIC501300.0 [1]
N-(2,3-Dihydro-1H-inden-2-yl)-6-[5-(2,3-dihydro-1H-inden-2-ylcarbamoyl)-1,6,7-trihydroxy-3-methylnaphthalen-2-yl]-2,3,5-trihydroxy-7-methylnaphthalene-1-carboxamideIC50670.0 [1]
3-Methyl-5-(2-phenylethyl)-2-[1,6,7-trihydroxy-3-methyl-5-(2-phenylethyl)naphthalen-2-yl]naphthalene-1,6,7-triolIC505000.0 [1]
N-[1-(4-Chlorophenyl)ethyl]-6-[5-[1-(4-chlorophenyl)ethylcarbamoyl]-1,6,7-trihydroxy-3-methylnaphthalen-2-yl]-2,3,5-trihydroxy-7-methylnaphthalene-1-carboxamideIC50400.0 [1]
N-(Cyclohexylmethyl)-6-[5-(cyclohexylmethylcarbamoyl)-1,6,7-trihydroxy-3-methylnaphthalen-2-yl]-2,3,5-trihydroxy-7-methylnaphthalene-1-carboxamideIC502000.0 [1]
2-[1-Hydroxy-4-[(4-phenylphenyl)sulfonylamino]naphthalen-2-yl]sulfanylacetic acidKi2340.0 [1]
2,3,5-Trihydroxy-7-methyl-N-[(2S)-2-phenylpropyl]-6-[1,6,7-trihydroxy-3-methyl-5-[[(2S)-2-phenylpropyl]carbamoyl]naphthalen-2-yl]naphthalene-1-carboxamideIC50750.0 [1]
2-[4-[[4-(4-Chlorophenyl)phenyl]sulfonylamino]-1-hydroxynaphthalen-2-yl]sulfanylacetic acidKi1110.0 [1]
2-[1-Hydroxy-4-[(3-phenylphenyl)sulfonylamino]naphthalen-2-yl]sulfanylacetic acidKi3180.0 [1]
2-[1-Hydroxy-4-[(2-phenylphenyl)sulfonylamino]naphthalen-2-yl]sulfanylacetic acidKi17260.0 [1]
Items per page: 1 - 10 of 76
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References

This online tool may be cited as follows

MLA

"Quest Database™ Bcl-2-related protein A1 Inhibitors (IC50, Ki)." AAT Bioquest, Inc., 20 Feb. 2025, https://www.aatbio.com/data-sets/bcl-2-related-protein-a1-inhibitors-ic50-ki.

APA

AAT Bioquest, Inc. (2025, February 20). Quest Database™ Bcl-2-related protein A1 Inhibitors (IC50, Ki). AAT Bioquest. https://www.aatbio.com/data-sets/bcl-2-related-protein-a1-inhibitors-ic50-ki.
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