AMP-activated protein kinase, beta-1 subunit Inhibitors (IC50, Ki)

Structure ▲ ▼	Compound Name ▲ ▼	Standard Type ▲ ▼	Standard Values (in nM) ▲ ▼
	Dorsomorphin	IC50	234.6 [1], 318.2 [2]
	4-(6-(4-(Piperazin-1-yl)phenyl)pyrazolo[1,5-a]pyrimidin-3-yl)quinoline	IC50	1122.0 [1]
	6-Chloro-5-(4-(1-hydroxycyclobutyl)phenyl)-1H-indole-3-carboxylic acid	IC50	400.0 [1]
	5-[6-[4-(1-Piperazinyl)phenyl]pyrazolo[1,5-a]pyrimidin-3-yl]quinoline	IC50	2520.0 [1]
	CID 59604787	IC50	10000.0 [1]
	4-[2-[4-(3-Phenylpyrazolo[1,5-a]pyrimidin-6-yl)phenoxy]ethyl]morpholine	IC50	2916.0 [1]
	7-Chloro-3-oxo-8-(1,3-thiazol-5-ylmethylamino)-11,16-dioxa-2,4,19,21-tetrazatricyclo[15.3.1.05,10]henicosa-1(20),5,7,9,17(21),18-hexaene-18-carbonitrile	Ki	1539.0 [1]
	Khk-IN-1	IC50	40000.0 [1]
	7-Chloro-9-ethyl-6-hydroxy-1H,3H,4H,9H-quinolino[2,3-c][1,2]oxazole-3,4-dione	Ki	1730.0 [1]
	4-(6-(4-Methoxyphenyl)pyrazolo[1,5-a]pyrimidin-3-yl)quinoline	IC50	7260.0 [1]
	CID 60182364	IC50	960.0 [1]
	CID 60182389	IC50	2680.0 [1]
	4-(4-(3-(1H-Pyrazol-4-yl)pyrazolo[1,5-a]pyrimidin-6-yl)phenyl)morpholine	IC50	39.9 [1]
	6-Chloro-5-[6-(Dimethylamino)-2-Methoxypyridin-3-Yl]-1h-Indole-3-Carboxylic Acid	IC50	420.0 [1]
	1-O-{6-Chloro-5-[4-(1-hydroxycyclobutyl)phenyl]-1H-indole-3-carbonyl}-beta-D-glucopyranuronic acid	IC50	11000.0 [1]
	(2S,3S,4S,5R,6S)-6-[6-Chloro-5-[6-(dimethylamino)-2-methoxypyridin-3-yl]-1H-indole-3-carbonyl]oxy-3,4,5-trihydroxyoxane-2-carboxylic acid	IC50	25000.0 [1]
	4-[2-[4-(3-Quinolin-4-ylpyrazolo[1,5-a]pyrimidin-6-yl)phenoxy]ethyl]morpholine	IC50	527.0 [1]
	6-(4-Methoxyphenyl)-3-(1H-pyrazol-4-yl)pyrazolo[1,5-a]pyrimidine	IC50	44.0 [1]
	6-(4-Piperazin-1-ylphenyl)-3-(1H-pyrazol-4-yl)pyrazolo[1,5-a]pyrimidine	IC50	82.0 [1]
	3-Phenyl-6-(4-piperazin-1-ylphenyl)pyrazolo[1,5-a]pyrimidine	IC50	1122.0 [1]
	3-(Tert-butylamino)-4-[[2-(4-pyridin-4-ylanilino)pyrimidin-4-yl]amino]cyclobut-3-ene-1,2-dione	Ki	333.0 [1]
	N,N-Dimethyl-3-[4-(3-quinolin-4-ylpyrazolo[1,5-a]pyrimidin-6-yl)phenoxy]propan-1-amine	IC50	1940.0 [1]

Entire TableStructureCompound NameStandard TypeStandard Values (in nM)

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References

This online tool may be cited as follows

MLA	"Quest Database™ AMP-activated protein kinase, beta-1 subunit Inhibitors (IC50, Ki)." AAT Bioquest, Inc., 21 Nov. 2024, https://www.aatbio.com/data-sets/amp-activated-protein-kinase-beta-1-subunit-inhibitors-ic50-ki.
APA	AAT Bioquest, Inc. (2024, November 21). Quest Database™ AMP-activated protein kinase, beta-1 subunit Inhibitors (IC50, Ki). AAT Bioquest. https://www.aatbio.com/data-sets/amp-activated-protein-kinase-beta-1-subunit-inhibitors-ic50-ki.
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