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AMP-activated protein kinase, AMPK Inhibitors (IC50, Ki)

Structure
▲
▼
Compound Name
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▼
Standard Type
▲
▼
Standard Values (in nM)
▲
▼
DorsomorphinIC5041.0 [1], 230.0 [2]
3-(1H-Indol-5-yl)-5-(4-((4-methylpiperazin-1-yl)methyl)phenyl)-1H-pyrrolo[2,3-b]pyridineIC501512.0 [1]
JNK Inhibitor VIIIKi9800.0 [1]
4-[2-[4-(3-Phenylpyrazolo[1,5-a]pyrimidin-6-yl)phenoxy]ethyl]morpholineIC501800.0 [1]
N-(4-Amino-5-cyano-6-ethoxypyridin-2-yl)acetamideKi9800.0 [1]
4-Amino-5-chloro-6-ethoxy-pyridine-2-carboxylic acid 4-methanesulfonyl-benzylamideKi9800.0 [1]
1-({4-[(3,4-Dichlorophenyl)methoxy]phenyl}methyl)azetidine-3-carboxylic acidIC5010000.0 [1]
4-[2-[4-(3-Pyridin-4-ylpyrazolo[1,5-a]pyrimidin-6-yl)phenoxy]ethyl]morpholineIC50280.0 [1]
N-(4-Amino-5-cyano-6-ethoxypyridin-2-yl)-2-(2,5-dimethoxy-4-methylsulfonylphenyl)acetamideKi9800.0 [1]
N-(4-Amino-5-chloro-6-ethoxypyridin-2-yl)-2-(4-methanesulfonyl-2,5-dimethoxyphenyl)acetamideKi9800.0 [1]
N-(4-Amino-5-cyano-6-isopropoxypyridin-2-yl)-2-(4-methanesulfonyl-2,5-dimethoxyphenyl)acetamideKi9800.0 [1]
N-(4-Amino-5-cyano-6-phenylpyridin-2-yl)acetamideKi9800.0 [1]
N-Propyl-4-({4-[(2,2,2-trifluoroethyl)amino]-1H-pyrrolo[2,3-d]pyrimidin-2-yl}amino)benzamideIC501400.0 [1]
5-(3-Tert-butyl-[1,2,4]triazolo[4,3-a]pyridin-6-yl)-4-(2,4-difluorophenyl)-1,3-oxazoleIC5010000.0 [1]
5-(3-Propan-2-yl-[1,2,4]triazolo[4,3-a]pyridin-6-yl)-4-(2,4,5-trifluorophenyl)-1,3-oxazoleIC5010000.0 [1]
(2S)-2-[[4-(3-Chloro-2-fluoroanilino)-7-methoxyquinazolin-6-yl]methyl-methylamino]-3-hydroxypropanamideIC5010000.0 [1]
(S)-1-((4-(3-Chloro-2-fluorophenylamino)-7-methoxyquinazolin-6-yl)methyl)pyrrolidine-2-carboxamideIC5010000.0 [1]
(R)-1-((4-(3-Chloro-2-fluorophenylamino)-7-methoxyquinazolin-6-yl)methyl)pyrrolidine-2-carboxamideIC5010000.0 [1]
(R)-2-((4-(3-Chloro-2-fluorophenylamino)-7-methoxyquinazolin-6-yl)methylamino)propanamideIC5010000.0 [1]
3-[[4-(3-Chloro-2-fluoroanilino)-7-methoxyquinazolin-6-yl]methyl-methylamino]-1-(2-methoxyethyl)azetidine-3-carboxamideIC5010000.0 [1]
(R)-2-(((4-(3-Chloro-2-fluorophenylamino)-7-methoxyquinazolin-6-yl)methyl)(methyl)amino)propanamideIC5010000.0 [1]
(R)-1-((4-(3-Chloro-4-fluorophenylamino)-7-methoxyquinazolin-6-yl)methyl)pyrrolidine-2-carboxamideIC5010000.0 [1]
3-[[4-(3-Chloro-2-fluoroanilino)-7-methoxyquinazolin-6-yl]methyl-methylamino]-1-methylazetidine-3-carboxamideIC5010000.0 [1]
(S)-1-((4-(3-Chloro-4-fluorophenylamino)-7-methoxyquinazolin-6-yl)methyl)pyrrolidine-2-carboxamideIC5010000.0 [1]
2-[3-(3-Piperidin-4-ylpropoxy)phenyl]-N-[4-(1H-pyrrolo[2,3-b]pyridin-3-yl)-1,3-thiazol-2-yl]acetamideKi2000.0 [1]
3-[[4-(3-Chloro-2-fluoroanilino)-7-methoxyquinazolin-6-yl]methyl-methylamino]-1-propan-2-ylazetidine-3-carboxamideIC5010000.0 [1]
(S)-2-(((4-(3-Chloro-2-fluorophenylamino)-7-methoxyquinazolin-6-yl)methyl)(methyl)amino)propanamideIC5010000.0 [1]
4-[[4-(3-Chloro-2-fluoroanilino)-7-methoxyquinazolin-6-yl]methyl-methylamino]-1-methylpiperidine-4-carboxamideIC5010000.0 [1]
(2R)-2-[[4-(3-Chloro-2-fluoroanilino)-7-methoxyquinazolin-6-yl]methyl-methylamino]-N-methylpropanamideIC5010000.0 [1]
2-(((4-(3-Chloro-2-fluorophenylamino)-7-methoxyquinazolin-6-yl)methyl)(methyl)amino)acetamideIC5010000.0 [1]
2-[3-(Methanesulfonamido)phenyl]-N-[4-(1H-pyrrolo[2,3-b]pyridin-3-yl)-1,3-thiazol-2-yl]acetamideKi2000.0 [1]
(2S)-2-[[4-(3-Chloro-2-fluoroanilino)-7-methoxyquinazolin-6-yl]methyl-methylamino]-4-methoxybutanamideIC5010000.0 [1]
2-[3-[3-(4-Methylpiperazin-1-yl)propoxy]phenyl]-N-[4-(1H-pyrrolo[2,3-b]pyridin-3-yl)-1,3-thiazol-2-yl]acetamideKi10000.0 [1]
(2S)-2-[[4-(3-Chloro-2-fluoroanilino)-7-methoxyquinazolin-6-yl]methyl-methylamino]-3-methoxypropanamideIC5010000.0 [1]
Nintedanib impurity EKi4.2 [1]
Melk-IN-1Ki9.2 [1]
2-Hydroxy-3-[N-[4-[methyl-[2-(4-methylpiperazin-1-yl)acetyl]amino]phenyl]-C-phenylcarbonimidoyl]-1H-indole-5-carboxylic acidKi4.9 [1]
5,5-Dimethyl-8-[[4-(2,2,2-trifluoroethylamino)furo[3,2-d]pyrimidin-2-yl]amino]-1H-4,1-benzoxazepin-2-oneIC5010000.0 [1]
(2E)-2-[(3,4-Dihydroxyphenyl)methylidene]-1-benzofuran-3-oneIC5019500.0 [1]
4-(2-Chloro-4-fluorophenyl)-5-(3-propan-2-yl-[1,2,4]triazolo[4,3-a]pyridin-6-yl)-1,3-oxazoleIC5010000.0 [1]
N-Ethyl-6-[4-(4-fluorophenyl)-1,3-oxazol-5-yl]-[1,2,4]triazolo[4,3-a]pyridin-3-amineIC5010000.0 [1]
6-[5-(2,5-Difluorophenyl)-1H-pyrazol-4-yl]-3-propan-2-yl-[1,2,4]triazolo[4,3-a]pyridineIC5010000.0 [1]
(R)-1-((4-(3-Chloro-2-fluorophenylamino)-7-methoxyquinazolin-6-yl)methyl)piperidine-2-carboxamideIC5010000.0 [1]
4-((4-(3-Chloro-2-fluorophenylamino)-7-methoxyquinazolin-6-yl)methyl)morpholine-3-carboxamideIC5010000.0 [1]
(2R)-2-[[4-(3-Chloro-2-fluoroanilino)-7-methoxyquinazolin-6-yl]methyl-methylamino]-N,N-dimethylpropanamideIC5010000.0 [1]
1-((4-(3-Chloro-2-fluorophenylamino)-7-methoxyquinazolin-6-yl)methyl)azetidine-3-carboxamideIC5010000.0 [1]
CID 44410844IC5010000.0 [1]
1-((4-(3-Chloro-2-fluorophenylamino)-7-methoxyquinazolin-6-yl)methyl)azetidine-2-carboxamideIC5010000.0 [1]
(2R,4R)-1-[[4-(3-Chloro-2-fluoroanilino)-7-methoxyquinazolin-6-yl]methyl]-4-methoxypyrrolidine-2-carboxamideIC5010000.0 [1]
3-(((4-(3-Chloro-2-fluorophenylamino)-7-methoxyquinazolin-6-yl)methyl)(methyl)amino)pyrrolidin-2-oneIC5010000.0 [1]
(2S)-2-[[4-(3-Chloro-2-fluoroanilino)-7-methoxyquinazolin-6-yl]methyl-propan-2-ylamino]propanamideIC5010000.0 [1]
(2R)-1-[[4-(3-Chloro-2-fluoroanilino)-7-methoxyquinazolin-6-yl]methyl]-N-methylpyrrolidine-2-carboxamideIC5010000.0 [1]
(2S)-2-[[4-(3-Chloro-2-fluoroanilino)-7-methoxyquinazolin-6-yl]methyl-[2-(dimethylamino)ethyl]amino]propanamideIC5010000.0 [1]
(2R)-1-[[4-(3-Chloro-2-fluoroanilino)-7-methoxyquinazolin-6-yl]methyl]-N,N-dimethylpyrrolidine-2-carboxamideIC5010000.0 [1]
(2S)-2-[[4-(3-Chloro-2-fluoroanilino)-7-methoxyquinazolin-6-yl]methyl-(2-methoxyethyl)amino]propanamideIC5010000.0 [1]
2-[(2S)-1-[[4-(3-Chloro-2-fluoroanilino)-7-methoxyquinazolin-6-yl]methyl]pyrrolidin-2-yl]acetamideIC5010000.0 [1]
1-[[4-(3-Chloro-2-fluoroanilino)-7-methoxyquinazolin-6-yl]methyl]-4-methylpiperazine-2-carboxamideIC5010000.0 [1]
(S)-1-((4-(3-Chloro-2-fluorophenylamino)-7-methoxyquinazolin-6-yl)methyl)pyrrolidine-3-carboxamideIC5010000.0 [1]
(2S)-2-[[4-(3-Chloro-2-fluoroanilino)-7-methoxyquinazolin-6-yl]methyl-methylamino]-3-(dimethylamino)propanamideIC5010000.0 [1]
4-[[4-(3-Chloro-2-fluoroanilino)-7-methoxyquinazolin-6-yl]methyl-methylamino]-1-propan-2-ylpiperidine-4-carboxamideIC5010000.0 [1]
2-[9-(4-Amino-3-methoxyphenyl)-6-oxo-5,11-dihydrobenzo[b][1,4]benzodiazepin-3-yl]-N-(4-morpholin-4-ylphenyl)acetamideIC5050000.0 [1]
2-[9-(4-Amino-3-methoxyphenyl)-6-oxo-5,11-dihydrobenzo[b][1,4]benzodiazepin-3-yl]-2-methyl-N-(4-morpholin-4-ylphenyl)propanamideIC5010000.0 [1]
5-[6-[4-(2-Morpholin-4-ylethoxy)phenyl]pyrazolo[1,5-a]pyrimidin-3-yl]-1H-pyridin-2-oneIC5060.0 [1]
5-[6-[4-(2-Morpholin-4-ylethoxy)phenyl]pyrazolo[1,5-a]pyrimidin-3-yl]pyridin-2-amineIC502100.0 [1]
4-(5-(3,4-Dihydroxyphenyl)oxazol-2-ylamino)benzenesulfonamideIC502900.0 [1]
4-[6-[4-(2-Morpholin-4-ylethoxy)phenyl]pyrazolo[1,5-a]pyrimidin-3-yl]benzene-1,2-diolIC501100.0 [1]
4-[6-[4-(2-Morpholin-4-ylethoxy)phenyl]pyrazolo[1,5-a]pyrimidin-3-yl]-1H-pyridin-2-oneIC50270.0 [1]
4-[2-[4-(3-Bromopyrazolo[1,5-a]pyrimidin-6-yl)phenoxy]ethyl]morpholineIC503500.0 [1]
4-[2-[4-[3-(1H-Pyrazol-4-yl)pyrazolo[1,5-a]pyrimidin-6-yl]phenoxy]ethyl]morpholineIC50140.0 [1]
4-[6-[4-(2-Morpholin-4-ylethoxy)phenyl]pyrazolo[1,5-a]pyrimidin-3-yl]pyridin-2-amineIC50220.0 [1]
4-(3-Bromopyrazolo[1,5-a]pyrimidin-6-yl)phenolIC507700.0 [1]
4-(5-(6-Oxo-1,6-dihydropyridin-3-yl)oxazol-2-ylamino)benzenesulfonamideIC505000.0 [1]
4-[2-[4-[3-(3,4-Dimethoxyphenyl)pyrazolo[1,5-a]pyrimidin-6-yl]phenoxy]ethyl]morpholineIC502200.0 [1]
2-[3-(3-Piperazin-1-ylpropoxy)phenyl]-N-(4-pyridin-4-yl-1,3-thiazol-2-yl)acetamideIC5010000.0 [1]
2-N-(1H-Indazol-6-yl)-4-N-(2,2,2-trifluoroethyl)furo[3,2-d]pyrimidine-2,4-diamineIC5010000.0 [1]
N~4~-Cyclopropyl-N~2~-(3-Methyl-1h-Indazol-6-Yl)furo[3,2-D]pyrimidine-2,4-DiamineIC5010000.0 [1]
2-N-(3-Chloro-4-morpholin-4-ylphenyl)-4-N-(2,2,2-trifluoroethyl)furo[3,2-d]pyrimidine-2,4-diamineIC5010000.0 [1]
2-(2,6-Dichloroanilino)-7-[(E)-3-(diethylamino)prop-1-enyl]-1,6-dimethyl-8H-imidazo[4,5-h]isoquinolin-9-oneIC501000.0 [1]
3-Isopropyl-6-(4-phenyl-oxazol-5-yl)-[1,2,4]triazolo[4,3-a]pyridineIC5010000.0 [1]
5-(3-Tert-butyl-[1,2,4]triazolo[4,3-a]pyridin-6-yl)-4-(2,4,5-trifluorophenyl)-1,3-oxazoleIC5010000.0 [1]
Items per page: 1 - 10 of 80
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References

This online tool may be cited as follows

MLA

"Quest Database™ AMP-activated protein kinase, AMPK Inhibitors (IC50, Ki)." AAT Bioquest, Inc., 22 Feb. 2025, https://www.aatbio.com/data-sets/amp-activated-protein-kinase-ampk-inhibitors-ic50-ki.

APA

AAT Bioquest, Inc. (2025, February 22). Quest Database™ AMP-activated protein kinase, AMPK Inhibitors (IC50, Ki). AAT Bioquest. https://www.aatbio.com/data-sets/amp-activated-protein-kinase-ampk-inhibitors-ic50-ki.
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