| 1-(1,3-Benzothiazol-2-yl)-3,4-dimethyl-1H-pyrazol-5-ol | IC50 | 10000.0 [1] |
| 4-Benzyl-5-methyl-2-(6-methyl-1H-benzimidazol-2-yl)-1H-pyrazol-3-one | IC50 | 670.0 [1] |
| DMT1 blocker 1 | IC50 | 1700.0 [1] |
| 2,3-Bis(4-methylphenyl)-5-methyl-1H-indene-1-one | IC50 | 50000.0 [1] |
| 2-Bromo-3-(4-methoxyphenyl)-5-methylinden-1-one | IC50 | 43170.0 [1] |
| 2-(3,5-Dimethoxyphenyl)-3-(4-methoxyphenyl)-5-(4-methylphenyl)inden-1-one | IC50 | 50000.0 [1] |
| 2-Chloro-3-(4-methoxyphenyl)-5-phenylinden-1-one | IC50 | 50000.0 [1] |
| 2-Bromo-3-(3,5-dimethoxyphenyl)-5-methylinden-1-one | IC50 | 50000.0 [1] |
| 2,3-Bis(3,4-dichlorophenyl)-5-methylinden-1-one | IC50 | 32300.0 [1] |
| 2,3-Bis(3,4-dimethoxyphenyl)-5-phenylinden-1-one | IC50 | 50000.0 [1] |
| 2-Chloro-3-(4-methoxyphenyl)-5-(4-methylphenyl)inden-1-one | IC50 | 9800.0 [1] |
| 2,3-Bis(3-methoxyphenyl)-5-phenylinden-1-one | IC50 | 50000.0 [1] |
| 2,3-Bis(3-methoxyphenyl)-5-(4-methylphenyl)inden-1-one | IC50 | 13100.0 [1] |
| 2-(3,5-Dimethoxyphenyl)-3-(4-methoxyphenyl)-5-phenylinden-1-one | IC50 | 50000.0 [1] |
| 2-Bromo-5-methyl-3-naphthalen-1-ylinden-1-one | IC50 | 50000.0 [1] |
| 2,3-Bis(4-methoxyphenyl)-5-phenylinden-1-one | IC50 | 50000.0 [1] |
| 2,3-Bis(4-methoxyphenyl)-5-methylinden-1-one | IC50 | 50000.0 [1] |
| 2,3-Bis(3-methoxyphenyl)-5-methylinden-1-one | IC50 | 50000.0 [1] |
| 3-(3,5-Dimethoxyphenyl)-2-(4-methoxyphenyl)-5-methylinden-1-one | IC50 | 50000.0 [1] |
| 2,3-Bis(3,4-dimethoxyphenyl)-5-(4-methylphenyl)inden-1-one | IC50 | 50000.0 [1] |
| 2-Chloro-3-(4-methoxyphenyl)-5-methylinden-1-one | IC50 | 50000.0 [1] |
| 2-Bromo-5-methyl-3-(4-methylphenyl)inden-1-one | IC50 | 50000.0 [1] |
| 2,3-Bis(3,4-dimethoxyphenyl)-5-methylinden-1-one | IC50 | 50000.0 [1] |
| 2-(3,5-Dimethoxyphenyl)-3-(4-methoxyphenyl)-5-methylinden-1-one | IC50 | 50000.0 [1] |
| 2-Bromo-3-(3,4-dimethoxyphenyl)-5-methylinden-1-one | IC50 | 50000.0 [1] |
| 1-(1H-Benzimidazol-2-yl)-4-(4-tert-butylbenzyl)-3-methyl-1H-pyrazol-5-ol | IC50 | 4100.0 [1] |
| 1-(1H-Benzimidazol-2-yl)-3,4-dimethyl-1H-pyrazol-5-ol | IC50 | 4000.0 [1] |
| 1-(1H-Benzimidazol-2-yl)-4-(2-chlorobenzyl)-3-methyl-1H-pyrazol-5-ol | IC50 | 10000.0 [1] |
| 1-(1H-Benzimidazol-2-yl)-4-(4-chlorobenzyl)-3-methyl-1H-pyrazol-5-ol | IC50 | 10000.0 [1] |
| 1-(1H-Benzimidazol-2-yl)-4-(3-chlorobenzyl)-3-methyl-1H-pyrazol-5-ol | IC50 | 540.0 [1] |
| 2-(1,3-Benzoxazol-2-yl)-4,5-dimethyl-1H-pyrazol-3-one | IC50 | 10000.0 [1] |
| 1-(1H-Benzimidazol-2-yl)-4-benzyl-3-methyl-1H-pyrazol-5-ol | IC50 | 480.0 [1] |
| 4,5-Dimethyl-2-pyridin-2-yl-1H-pyrazol-3-one | IC50 | 10000.0 [1] |
| 2,3,5-Triphenyl-1H-indene-1-one | IC50 | 50000.0 [1] |
| 3,4-Dimethyl-1-phenyl-3-pyrazolin-5-one | IC50 | 10000.0 [1] |
| 4,5-Dimethyl-2-pyrimidin-2-yl-1H-pyrazol-3-one | IC50 | 10000.0 [1] |
| 1-(1H-Benzimidazol-2-yl)-3-phenyl-1H-pyrazol-5-ol | IC50 | 7200.0 [1] |
| 2-Bromo-5-methyl-3-phenylinden-1-one | IC50 | 50000.0 [1] |
| 5-Methyl-2,3-diphenyl-1H-inden-1-one | IC50 | 50000.0 [1] |
| 1-(1H-Benzimidazol-2-yl)-3-methyl-1H-pyrazol-5-ol | IC50 | 3600.0 [1] |
| 2-[2-(1H-Benzimidazol-2-yl)-5-methyl-3-oxo-1H-pyrazol-4-yl]acetic acid | IC50 | 15000.0 [1] |
| 2-(6-Chloro-1H-benzimidazol-2-yl)-4,5-diphenyl-1H-pyrazol-3-one | IC50 | 2000.0 [1] |
| 4-Benzyl-2-(6-tert-butyl-1H-benzimidazol-2-yl)-5-methyl-1H-pyrazol-3-one | IC50 | 640.0 [1] |
| 4-[(3,4-Dichlorophenyl)methyl]-5-methyl-2-(6-methyl-1H-benzimidazol-2-yl)-1H-pyrazol-3-one | IC50 | 720.0 [1] |
| 2-(1H-Benzimidazol-2-yl)-4-[(3,4-dichlorophenyl)methyl]-5-methyl-1H-pyrazol-3-one | IC50 | 3100.0 [1] |
| 4,5-Dimethyl-2-(4-methyl-1H-benzimidazol-2-yl)-1H-pyrazol-3-one | IC50 | 10000.0 [1] |
| 2-(1H-Benzimidazol-2-yl)-4-[(2,4-dichlorophenyl)methyl]-5-methyl-1H-pyrazol-3-one | IC50 | 10000.0 [1] |
| 2-(1H-Benzimidazol-2-yl)-4-[(4-methoxyphenyl)methyl]-5-methyl-1H-pyrazol-3-one | IC50 | 630.0 [1] |
| 4-Benzyl-5-methyl-2-[6-(trifluoromethyl)-1H-benzimidazol-2-yl]-1H-pyrazol-3-one | IC50 | 610.0 [1] |
| 2-(6-Methyl-1H-benzimidazol-2-yl)-4,5-diphenyl-1H-pyrazol-3-one | IC50 | 5800.0 [1] |
| 4-[(4-Fluorophenyl)methyl]-5-methyl-2-(6-methyl-1H-benzimidazol-2-yl)-1H-pyrazol-3-one | IC50 | 780.0 [1] |
| 5-Methyl-2-(6-methyl-1H-benzimidazol-2-yl)-4-[(4-phenylphenyl)methyl]-1H-pyrazol-3-one | IC50 | 5300.0 [1] |
| 4,5-Dimethyl-2-(1-methylbenzimidazol-2-yl)-1H-pyrazol-3-one | IC50 | 10000.0 [1] |
| 4-Benzyl-5-methyl-2-(6-phenyl-1H-benzimidazol-2-yl)-1H-pyrazol-3-one | IC50 | 810.0 [1] |
| 4-Benzyl-5-methyl-2-(4-methyl-1H-benzimidazol-2-yl)-1H-pyrazol-3-one | IC50 | 5900.0 [1] |
| 4-[(4-Chlorophenyl)methyl]-5-methyl-2-(6-methyl-1H-benzimidazol-2-yl)-1H-pyrazol-3-one | IC50 | 750.0 [1] |
| 4-[(4-Tert-butylphenyl)methyl]-5-methyl-2-(6-methyl-1H-benzimidazol-2-yl)-1H-pyrazol-3-one | IC50 | 3700.0 [1] |
| 4-Benzyl-5-methyl-2-[6-(4-methylphenyl)-1H-benzimidazol-2-yl]-1H-pyrazol-3-one | IC50 | 2100.0 [1] |
| 4,5-Dimethyl-2-(6-methyl-1H-benzimidazol-2-yl)-1H-pyrazol-3-one | IC50 | 2600.0 [1] |
| Methyl 2-[2-(1H-benzimidazol-2-yl)-5-methyl-3-oxo-1H-pyrazol-4-yl]acetate | IC50 | 4300.0 [1] |
| 2-(1H-Benzimidazol-2-yl)-4-benzyl-5-phenyl-1H-pyrazol-3-one | IC50 | 10000.0 [1] |
| 2-(1H-Benzimidazol-2-yl)-4-[(4-fluorophenyl)methyl]-5-methyl-1H-pyrazol-3-one | IC50 | 600.0 [1] |
| 2-(1H-Benzimidazol-2-yl)-5-methyl-4-[(4-phenylphenyl)methyl]-1H-pyrazol-3-one | IC50 | 720.0 [1] |
| 4-Benzyl-2-(6-chloro-1H-benzimidazol-2-yl)-5-methyl-1H-pyrazol-3-one | IC50 | 4500.0 [1] |
| 4-Benzyl-2-[6-(4-chlorophenyl)-1H-benzimidazol-2-yl]-5-methyl-1H-pyrazol-3-one | IC50 | 1500.0 [1] |
| 2-(1H-Benzimidazol-2-yl)-5-methyl-4-(naphthalen-2-ylmethyl)-1H-pyrazol-3-one | IC50 | 750.0 [1] |
| 2-(1H-Benzimidazol-2-yl)-4-methyl-5-phenyl-1H-pyrazol-3-one | IC50 | 10000.0 [1] |
| 4-Methyl-2-(6-methyl-1H-benzimidazol-2-yl)-5-phenyl-1H-pyrazol-3-one | IC50 | 3300.0 [1] |
| 2-(1H-Benzimidazol-2-yl)-5-methyl-4-[[4-(trifluoromethyl)phenyl]methyl]-1H-pyrazol-3-one | IC50 | 550.0 [1] |
| 4-Benzyl-2-(6-bromo-1H-benzimidazol-2-yl)-5-methyl-1H-pyrazol-3-one | IC50 | 490.0 [1] |
| 4-Benzyl-2-(4,5-dimethyl-1H-benzimidazol-2-yl)-5-methyl-1H-pyrazol-3-one | IC50 | 10000.0 [1] |
| 5-Methyl-2-(6-methyl-1H-benzimidazol-2-yl)-4-[[4-(trifluoromethyl)phenyl]methyl]-1H-pyrazol-3-one | IC50 | 570.0 [1] |
| 4-[(4-Methoxyphenyl)methyl]-5-methyl-2-(6-methyl-1H-benzimidazol-2-yl)-1H-pyrazol-3-one | IC50 | 680.0 [1] |
| 4-[(2-Chlorophenyl)methyl]-5-methyl-2-(6-methyl-1H-benzimidazol-2-yl)-1H-pyrazol-3-one | IC50 | 910.0 [1] |