![](https://images.aatbio.com/dataset/ic50/alpha-1-6-mannosyl-glycoprotein-2-beta-n-acetylglucosaminyltransferase_a33ac9aa8864cb9c5427f6c8ee0cff16.svg) | N-Tert-butyl-8-[[[(1S,2S)-2-(3-methyl-1,2,4-oxadiazol-5-yl)cyclopropanecarbonyl]amino]methyl]-5-[3-(trifluoromethoxy)phenyl]-3,4-dihydro-1H-isoquinoline-2-carboxamide | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/alpha-1-6-mannosyl-glycoprotein-2-beta-n-acetylglucosaminyltransferase_67fb993ac1cbdbfc372ebb9b9519102a.svg) | (3S)-N-(2,4-Difluorophenyl)-3-ethyl-3-methyl-2,5-dioxo-1,4-dihydro-1,4-benzodiazepine-7-sulfonamide | IC50 | 6.31 [1], 12.59 [2] |
![](https://images.aatbio.com/dataset/ic50/alpha-1-6-mannosyl-glycoprotein-2-beta-n-acetylglucosaminyltransferase_48bca7da5238fe2ac449dea121fdff1b.svg) | N-(4-Methoxyphenyl)-4-(4-methylphenyl)-6-oxo-2-[4-(4,4,4-trifluorobutoxy)phenyl]-2-(trifluoromethyl)-1,3-dihydropyridine-5-carboxamide | IC50 | 55.0 [1], 4264.0 [2] |
![](https://images.aatbio.com/dataset/ic50/alpha-1-6-mannosyl-glycoprotein-2-beta-n-acetylglucosaminyltransferase_4d711a968e1a760df09fb07d77437d02.svg) | 5-(2-Ethyltetrazol-5-yl)-4-(4-methylphenyl)-2-[4-(4,4,4-trifluorobutoxy)phenyl]-2-(trifluoromethyl)-1,3-dihydropyridin-6-one | IC50 | 121.0 [1], 33330.0 [2] |
![](https://images.aatbio.com/dataset/ic50/alpha-1-6-mannosyl-glycoprotein-2-beta-n-acetylglucosaminyltransferase_adb7731cfa53bc06bfda4175d55d8444.svg) | 6-Methyl-4-(4-methylphenyl)-2-oxo-6-pentyl-1,3-dihydropyridine-3-carbonitrile | IC50 | 651.0 [1], 2049.0 [2] |
![](https://images.aatbio.com/dataset/ic50/alpha-1-6-mannosyl-glycoprotein-2-beta-n-acetylglucosaminyltransferase_b4b71c78af1f520390129d6a20bc461f.svg) | (6R)-N-(4-Methoxyphenyl)-4-(4-methylphenyl)-2-oxo-6-[4-(4,4,4-trifluorobutoxy)phenyl]-6-(trifluoromethyl)piperidine-3-carboxamide | IC50 | 416.0 [1], 8430.0 [2] |
![](https://images.aatbio.com/dataset/ic50/alpha-1-6-mannosyl-glycoprotein-2-beta-n-acetylglucosaminyltransferase_245963b81a55f03fefad76e42f914446.svg) | 2-(4-Methoxyphenyl)-4-(4-methylphenyl)-6-oxo-2-(trifluoromethyl)-1,3-dihydropyridine-5-carbonitrile | IC50 | 20.0 [1], 401.0 [2] |
![](https://images.aatbio.com/dataset/ic50/alpha-1-6-mannosyl-glycoprotein-2-beta-n-acetylglucosaminyltransferase_270c930a84683a517899dd04576b2d01.svg) | 4-(4-Methylphenyl)-2-[4-[2-[(2-methylpropan-2-yl)oxy]ethoxy]phenyl]-6-oxo-2-(trifluoromethyl)-1,3-dihydropyridine-5-carbonitrile | IC50 | 126.0 [1], 656.0 [2] |
![](https://images.aatbio.com/dataset/ic50/alpha-1-6-mannosyl-glycoprotein-2-beta-n-acetylglucosaminyltransferase_b01cf56f89f3d54166e3b803d61a737e.svg) | 4-(4-Methylphenyl)-6-oxo-2-[4-(3-phenylpropoxy)phenyl]-2-(trifluoromethyl)-1,3-dihydropyridine-5-carbonitrile | IC50 | 13.0 [1], 5199.0 [2] |
![](https://images.aatbio.com/dataset/ic50/alpha-1-6-mannosyl-glycoprotein-2-beta-n-acetylglucosaminyltransferase_892ac2f828b787a4781e7993bdb16ed4.svg) | 2-[4-(2-Cyclopentylethoxy)phenyl]-4-(4-methylphenyl)-6-oxo-2-(trifluoromethyl)-1,3-dihydropyridine-5-carbonitrile | IC50 | 57.0 [1], 396.0 [2] |
![](https://images.aatbio.com/dataset/ic50/alpha-1-6-mannosyl-glycoprotein-2-beta-n-acetylglucosaminyltransferase_6f44e997ee1c413c16f8d16b949b29e1.svg) | 2-[4-(3-Methylbutoxy)phenyl]-4-(4-methylphenyl)-6-oxo-2-(trifluoromethyl)-1,3-dihydropyridine-5-carbonitrile | IC50 | 15.0 [1], 263.0 [2] |
![](https://images.aatbio.com/dataset/ic50/alpha-1-6-mannosyl-glycoprotein-2-beta-n-acetylglucosaminyltransferase_dbb7c1ddfe5ad6675a87ac47733d24ab.svg) | 2-[4-(4-Methoxyphenyl)phenyl]-4-(4-methylphenyl)-6-oxo-2-(trifluoromethyl)-1,3-dihydropyridine-5-carbonitrile | IC50 | 164.0 [1], 2546.0 [2] |
![](https://images.aatbio.com/dataset/ic50/alpha-1-6-mannosyl-glycoprotein-2-beta-n-acetylglucosaminyltransferase_8e5c23cd7195f176e32d9ff5cf0bfd45.svg) | N-(4-Fluorophenyl)-2-(4-methoxyphenyl)-4-(4-methylphenyl)-6-oxo-2-(trifluoromethyl)-1,3-dihydropyridine-5-carboxamide | IC50 | 15.0 [1], 170.0 [2] |
![](https://images.aatbio.com/dataset/ic50/alpha-1-6-mannosyl-glycoprotein-2-beta-n-acetylglucosaminyltransferase_6b43850f07f30abf5687e22d67b551af.svg) | 4-(4-Methylphenyl)-6-oxo-2-(4-pentylphenyl)-2-(trifluoromethyl)-1,3-dihydropyridine-5-carbonitrile | IC50 | 77.0 [1], 403.0 [2] |
![](https://images.aatbio.com/dataset/ic50/alpha-1-6-mannosyl-glycoprotein-2-beta-n-acetylglucosaminyltransferase_fd1e1017df63afe9a55aaff90730fb85.svg) | 4-(4-Methylphenyl)-6-oxo-2-(4-pyridin-2-ylphenyl)-2-(trifluoromethyl)-1,3-dihydropyridine-5-carbonitrile | IC50 | 60.0 [1], 5387.0 [2] |
![](https://images.aatbio.com/dataset/ic50/alpha-1-6-mannosyl-glycoprotein-2-beta-n-acetylglucosaminyltransferase_82e49a8ead2a1c2af000df5e7dda45fb.svg) | N-(4-Fluorophenyl)-4-(4-methylphenyl)-6-oxo-2-(4-phenoxyphenyl)-2-(trifluoromethyl)-1,3-dihydropyridine-5-carboxamide | IC50 | 8.0 [1], 60.0 [2] |
![](https://images.aatbio.com/dataset/ic50/alpha-1-6-mannosyl-glycoprotein-2-beta-n-acetylglucosaminyltransferase_7a60e29442ee104885d6c2fcaf3b6705.svg) | N-(4-Fluorophenyl)-4-(4-methylphenyl)-6-oxo-2-(4-pyrimidin-4-yloxyphenyl)-2-(trifluoromethyl)-1,3-dihydropyridine-5-carboxamide | IC50 | 64.0 [1], 127.0 [2] |
![](https://images.aatbio.com/dataset/ic50/alpha-1-6-mannosyl-glycoprotein-2-beta-n-acetylglucosaminyltransferase_824dec7e6c9b6749e3204a6ae2076852.svg) | N-(4-Fluorophenyl)-4-(4-methylphenyl)-6-oxo-2-(4-pyrazin-2-ylphenyl)-2-(trifluoromethyl)-1,3-dihydropyridine-5-carboxamide | IC50 | 95.0 [1], 242.0 [2] |
![](https://images.aatbio.com/dataset/ic50/alpha-1-6-mannosyl-glycoprotein-2-beta-n-acetylglucosaminyltransferase_242867666db47b947e5a95d48af7c542.svg) | N-(4-Fluorophenyl)-4-(4-methylphenyl)-6-oxo-2-(4-pentylphenyl)-2-(trifluoromethyl)-1,3-dihydropyridine-5-carboxamide | IC50 | 13.0 [1], 63.0 [2] |
![](https://images.aatbio.com/dataset/ic50/alpha-1-6-mannosyl-glycoprotein-2-beta-n-acetylglucosaminyltransferase_a2c9927cd55dd1afbb87b766e68769ba.svg) | N-(4-Fluorophenyl)-4-(4-methylphenyl)-6-oxo-2-(4-pyrimidin-2-yloxyphenyl)-2-(trifluoromethyl)-1,3-dihydropyridine-5-carboxamide | IC50 | 99.0 [1], 477.0 [2] |
![](https://images.aatbio.com/dataset/ic50/alpha-1-6-mannosyl-glycoprotein-2-beta-n-acetylglucosaminyltransferase_49bb60b2b25c38015b578d46f5714b19.svg) | N-(4-Fluorophenyl)-4-(4-methylphenyl)-6-oxo-2-(4-phenylmethoxyphenyl)-2-(trifluoromethyl)-1,3-dihydropyridine-5-carboxamide | IC50 | 20.0 [1], 258.0 [2] |
![](https://images.aatbio.com/dataset/ic50/alpha-1-6-mannosyl-glycoprotein-2-beta-n-acetylglucosaminyltransferase_8059efa6158151c1acdada47fec46a3b.svg) | 4-(4-Methylphenyl)-6-oxo-N-pentyl-2-[4-(4,4,4-trifluorobutoxy)phenyl]-2-(trifluoromethyl)-1,3-dihydropyridine-5-carboxamide | IC50 | 20.0 [1], 846.0 [2] |
![](https://images.aatbio.com/dataset/ic50/alpha-1-6-mannosyl-glycoprotein-2-beta-n-acetylglucosaminyltransferase_1e4b2e7843add6f046fe09d4893238d0.svg) | 4-(4-Methylphenyl)-6-oxo-N-(2-phenylethyl)-2-[4-(4,4,4-trifluorobutoxy)phenyl]-2-(trifluoromethyl)-1,3-dihydropyridine-5-carboxamide | IC50 | 16.0 [1], 412.0 [2] |
![](https://images.aatbio.com/dataset/ic50/alpha-1-6-mannosyl-glycoprotein-2-beta-n-acetylglucosaminyltransferase_a8143f85fea4ad96990d7b1186f24ad0.svg) | N-(3-Methoxyphenyl)-4-(4-methylphenyl)-6-oxo-2-[4-(4,4,4-trifluorobutoxy)phenyl]-2-(trifluoromethyl)-1,3-dihydropyridine-5-carboxamide | IC50 | 29.0 [1], 275.0 [2] |
![](https://images.aatbio.com/dataset/ic50/alpha-1-6-mannosyl-glycoprotein-2-beta-n-acetylglucosaminyltransferase_ae28fd2e6bd21429da0b6f0ca4f1c6b6.svg) | 4-(4-Methylphenyl)-6-oxo-N-phenyl-2-[4-(4,4,4-trifluorobutoxy)phenyl]-2-(trifluoromethyl)-1,3-dihydropyridine-5-carboxamide | IC50 | 4.0 [1], 53.0 [2] |
![](https://images.aatbio.com/dataset/ic50/alpha-1-6-mannosyl-glycoprotein-2-beta-n-acetylglucosaminyltransferase_954cecc44c8cca5ea3e871b4df069ec4.svg) | N-(2-Chlorophenyl)-4-(4-methylphenyl)-6-oxo-2-[4-(4,4,4-trifluorobutoxy)phenyl]-2-(trifluoromethyl)-1,3-dihydropyridine-5-carboxamide | IC50 | 12.0 [1], 441.0 [2] |
![](https://images.aatbio.com/dataset/ic50/alpha-1-6-mannosyl-glycoprotein-2-beta-n-acetylglucosaminyltransferase_f23de0869049cf76ef4a3a5e9f7c7fbc.svg) | N-(4-Chlorophenyl)-4-(4-methylphenyl)-6-oxo-2-[4-(4,4,4-trifluorobutoxy)phenyl]-2-(trifluoromethyl)-1,3-dihydropyridine-5-carboxamide | IC50 | 24.0 [1], 156.0 [2] |
![](https://images.aatbio.com/dataset/ic50/alpha-1-6-mannosyl-glycoprotein-2-beta-n-acetylglucosaminyltransferase_975abf8f45751f76b9b72dd40c8129d9.svg) | 4-(3-Methoxyphenyl)-6-oxo-2-[4-(4,4,4-trifluorobutoxy)phenyl]-2-(trifluoromethyl)-1,3-dihydropyridine-5-carbonitrile | IC50 | 280.0 [1], 761.0 [2] |
![](https://images.aatbio.com/dataset/ic50/alpha-1-6-mannosyl-glycoprotein-2-beta-n-acetylglucosaminyltransferase_337e0637b084061018c0a9c26ab69335.svg) | 4-(4-Methoxyphenyl)-6-oxo-2-[4-(4,4,4-trifluorobutoxy)phenyl]-2-(trifluoromethyl)-1,3-dihydropyridine-5-carbonitrile | IC50 | 27.0 [1], 89.0 [2] |
![](https://images.aatbio.com/dataset/ic50/alpha-1-6-mannosyl-glycoprotein-2-beta-n-acetylglucosaminyltransferase_9f3e031663c27eada5aef09f66fcdde6.svg) | 4-(4-Cyanophenyl)-6-oxo-2-[4-(4,4,4-trifluorobutoxy)phenyl]-2-(trifluoromethyl)-1,3-dihydropyridine-5-carbonitrile | IC50 | 414.0 [1], 731.0 [2] |
![](https://images.aatbio.com/dataset/ic50/alpha-1-6-mannosyl-glycoprotein-2-beta-n-acetylglucosaminyltransferase_6e2703bd0431624e1e8cf80e1826a5c0.svg) | 4-(4-Fluorophenyl)-6-oxo-2-[4-(4,4,4-trifluorobutoxy)phenyl]-2-(trifluoromethyl)-1,3-dihydropyridine-5-carbonitrile | IC50 | 697.0 [1], 2476.0 [2] |
![](https://images.aatbio.com/dataset/ic50/alpha-1-6-mannosyl-glycoprotein-2-beta-n-acetylglucosaminyltransferase_92449eac85936beb5a74d7fa4b4da389.svg) | 4-(3-Chlorophenyl)-6-oxo-2-[4-(4,4,4-trifluorobutoxy)phenyl]-2-(trifluoromethyl)-1,3-dihydropyridine-5-carbonitrile | IC50 | 1282.0 [1], 7523.0 [2] |
![](https://images.aatbio.com/dataset/ic50/alpha-1-6-mannosyl-glycoprotein-2-beta-n-acetylglucosaminyltransferase_ccab7a82fbd8bcd79c249089820c7d37.svg) | 4-(3-Cyanophenyl)-6-oxo-2-[4-(4,4,4-trifluorobutoxy)phenyl]-2-(trifluoromethyl)-1,3-dihydropyridine-5-carbonitrile | IC50 | 983.0 [1], 9230.0 [2] |
![](https://images.aatbio.com/dataset/ic50/alpha-1-6-mannosyl-glycoprotein-2-beta-n-acetylglucosaminyltransferase_d5722f97947aac60f2251f56c3082cdf.svg) | 6-Oxo-4-phenyl-2-[4-(4,4,4-trifluorobutoxy)phenyl]-2-(trifluoromethyl)-1,3-dihydropyridine-5-carbonitrile | IC50 | 1917.0 [1], 2931.0 [2] |
![](https://images.aatbio.com/dataset/ic50/alpha-1-6-mannosyl-glycoprotein-2-beta-n-acetylglucosaminyltransferase_b515ea0734fef9268be5ce8b43d17898.svg) | 4-(4-Chlorophenyl)-6-oxo-2-[4-(4,4,4-trifluorobutoxy)phenyl]-2-(trifluoromethyl)-1,3-dihydropyridine-5-carbonitrile | IC50 | 214.0 [1], 3519.0 [2] |
![](https://images.aatbio.com/dataset/ic50/alpha-1-6-mannosyl-glycoprotein-2-beta-n-acetylglucosaminyltransferase_063402a4198a86b5ee5b5d593cd5c1a3.svg) | 4-Naphthalen-2-yl-6-oxo-2-[4-(4,4,4-trifluorobutoxy)phenyl]-2-(trifluoromethyl)-1,3-dihydropyridine-5-carbonitrile | IC50 | 25.0 [1], 397.0 [2] |
![](https://images.aatbio.com/dataset/ic50/alpha-1-6-mannosyl-glycoprotein-2-beta-n-acetylglucosaminyltransferase_3c76b029c8ac3e2de75517b6cf882709.svg) | 6-Oxo-2-[4-(4,4,4-trifluorobutoxy)phenyl]-2-(trifluoromethyl)-4-[4-(trifluoromethyl)phenyl]-1,3-dihydropyridine-5-carbonitrile | IC50 | 209.0 [1], 873.0 [2] |
![](https://images.aatbio.com/dataset/ic50/alpha-1-6-mannosyl-glycoprotein-2-beta-n-acetylglucosaminyltransferase_a3b609675f8a70f7b8802701f6f62a0d.svg) | 6-Oxo-2-[4-(4,4,4-trifluorobutoxy)phenyl]-4-[4-(trifluoromethoxy)phenyl]-2-(trifluoromethyl)-1,3-dihydropyridine-5-carbonitrile | IC50 | 45.0 [1], 1856.0 [2] |
![](https://images.aatbio.com/dataset/ic50/alpha-1-6-mannosyl-glycoprotein-2-beta-n-acetylglucosaminyltransferase_a266f0e1b0da144cfc262b398cede34a.svg) | 4-(4-Ethoxyphenyl)-6-oxo-2-[4-(4,4,4-trifluorobutoxy)phenyl]-2-(trifluoromethyl)-1,3-dihydropyridine-5-carbonitrile | IC50 | 25.0 [1], 130.0 [2] |
![](https://images.aatbio.com/dataset/ic50/alpha-1-6-mannosyl-glycoprotein-2-beta-n-acetylglucosaminyltransferase_1ee57007a7d4d63c05d1d34d8e60fc40.svg) | 4-(2-Fluoro-4-methoxyphenyl)-6-oxo-2-[4-(4,4,4-trifluorobutoxy)phenyl]-2-(trifluoromethyl)-1,3-dihydropyridine-5-carbonitrile | IC50 | 2.0 [1], 916.0 [2] |
![](https://images.aatbio.com/dataset/ic50/alpha-1-6-mannosyl-glycoprotein-2-beta-n-acetylglucosaminyltransferase_76c48956013850efeb86f9d5e1e6dd69.svg) | N,4-Bis(4-methylphenyl)-6-oxo-2-[4-(4,4,4-trifluorobutoxy)phenyl]-2-(trifluoromethyl)-1,3-dihydropyridine-5-carboxamide | IC50 | 2.0 [1], 133.0 [2] |
![](https://images.aatbio.com/dataset/ic50/alpha-1-6-mannosyl-glycoprotein-2-beta-n-acetylglucosaminyltransferase_ee4a42b7db5077ada75866e429d74c31.svg) | N-(3-Fluoro-4-methoxyphenyl)-4-(4-methylphenyl)-6-oxo-2-[4-(4,4,4-trifluorobutoxy)phenyl]-2-(trifluoromethyl)-1,3-dihydropyridine-5-carboxamide | IC50 | 2.0 [1], 115.0 [2] |
![](https://images.aatbio.com/dataset/ic50/alpha-1-6-mannosyl-glycoprotein-2-beta-n-acetylglucosaminyltransferase_f095644f62b4c7d10b9b64ea18504e2e.svg) | N-(3-Fluoro-4-methylphenyl)-4-(4-methylphenyl)-6-oxo-2-[4-(4,4,4-trifluorobutoxy)phenyl]-2-(trifluoromethyl)-1,3-dihydropyridine-5-carboxamide | IC50 | 7.0 [1], 1465.0 [2] |
![](https://images.aatbio.com/dataset/ic50/alpha-1-6-mannosyl-glycoprotein-2-beta-n-acetylglucosaminyltransferase_5143c9c6c1107e402a4c067d37914c7e.svg) | N-(4-Methoxyphenyl)-4-(4-methylphenyl)-6-oxo-2-[4-(2,2,2-trifluoroethoxy)phenyl]-2-(trifluoromethyl)-1,3-dihydropyridine-5-carboxamide | IC50 | 5.0 [1], 28.0 [2] |
![](https://images.aatbio.com/dataset/ic50/alpha-1-6-mannosyl-glycoprotein-2-beta-n-acetylglucosaminyltransferase_44dfb4dbb58f0e21f2545009f56c0502.svg) | 4-(4-Methylphenyl)-6-oxo-2-[4-(2,2,2-trifluoroethoxy)phenyl]-2-(trifluoromethyl)-1,3-dihydropyridine-5-carbonitrile | IC50 | 20.0 [1], 731.0 [2] |
![](https://images.aatbio.com/dataset/ic50/alpha-1-6-mannosyl-glycoprotein-2-beta-n-acetylglucosaminyltransferase_f5e2cf3bebfada40e7a1b4fef42087dc.svg) | 4-(4-Methylphenyl)-5-(2H-tetrazol-5-yl)-2-[4-(2,2,2-trifluoroethoxy)phenyl]-2-(trifluoromethyl)-1,3-dihydropyridin-6-one | IC50 | 78.0 [1], 815.0 [2] |
![](https://images.aatbio.com/dataset/ic50/alpha-1-6-mannosyl-glycoprotein-2-beta-n-acetylglucosaminyltransferase_ba543c13cc1f74ea5c1b94a48e05b913.svg) | 4-[4-(Difluoromethoxy)phenyl]-5-(2H-tetrazol-5-yl)-2-[4-(4,4,4-trifluorobutoxy)phenyl]-2-(trifluoromethyl)-1,3-dihydropyridin-6-one | IC50 | 37.0 [1], 46.0 [2] |
![](https://images.aatbio.com/dataset/ic50/alpha-1-6-mannosyl-glycoprotein-2-beta-n-acetylglucosaminyltransferase_cc2af1df907ba86ed4e3621e1c91d517.svg) | 4-(4-Methylphenyl)-2-[4-(4,4,4-trifluorobutoxy)phenyl]-5-[4-(trifluoromethoxy)phenyl]-2-(trifluoromethyl)-1,3-dihydropyridin-6-one | IC50 | 4.0 [1], 32.0 [2] |
![](https://images.aatbio.com/dataset/ic50/alpha-1-6-mannosyl-glycoprotein-2-beta-n-acetylglucosaminyltransferase_ce8c01e9afe3d57699689c25f6779ec0.svg) | 4-(2-Fluoro-4-methoxyphenyl)-5-(2H-tetrazol-5-yl)-2-[4-(4,4,4-trifluorobutoxy)phenyl]-2-(trifluoromethyl)-1,3-dihydropyridin-6-one | IC50 | 43.0 [1], 95.0 [2] |
![](https://images.aatbio.com/dataset/ic50/alpha-1-6-mannosyl-glycoprotein-2-beta-n-acetylglucosaminyltransferase_07337d972cb3724ed10f5ca6fb9b6ace.svg) | 5-(2H-Tetrazol-5-yl)-2-[4-(4,4,4-trifluorobutoxy)phenyl]-2-(trifluoromethyl)-4-[4-(trifluoromethyl)phenyl]-1,3-dihydropyridin-6-one | IC50 | 69.0 [1], 154.0 [2] |
![](https://images.aatbio.com/dataset/ic50/alpha-1-6-mannosyl-glycoprotein-2-beta-n-acetylglucosaminyltransferase_ceb5dc78cb3c56600ac0f7dfd170162d.svg) | 4-(4-Chlorophenyl)-5-(2H-tetrazol-5-yl)-2-[4-(4,4,4-trifluorobutoxy)phenyl]-2-(trifluoromethyl)-1,3-dihydropyridin-6-one | IC50 | 108.0 [1], 379.0 [2] |
![](https://images.aatbio.com/dataset/ic50/alpha-1-6-mannosyl-glycoprotein-2-beta-n-acetylglucosaminyltransferase_3b8e7017d688a2024caa160e641a4a40.svg) | 4-(4-Methylphenyl)-6-oxo-N-[6-(2H-tetrazol-5-yl)pyridin-3-yl]-2-[4-(4,4,4-trifluorobutoxy)phenyl]-2-(trifluoromethyl)-1,3-dihydropyridine-5-carboxamide | IC50 | 7.0 [1], 9.0 [2] |
![](https://images.aatbio.com/dataset/ic50/alpha-1-6-mannosyl-glycoprotein-2-beta-n-acetylglucosaminyltransferase_faeff26c94c580e053fbebdc50257cb4.svg) | 2-(4-Bromophenyl)-4-(4-methylphenyl)-5-(2H-tetrazol-5-yl)-2-(trifluoromethyl)-1,3-dihydropyridin-6-one | IC50 | 639.0 [1], 1297.0 [2] |
![](https://images.aatbio.com/dataset/ic50/alpha-1-6-mannosyl-glycoprotein-2-beta-n-acetylglucosaminyltransferase_29475d389c338e05e9112c595e2903b7.svg) | 4-(4-Methylphenyl)-5-(5H-tetrazol-5-yl)-2-[4-(4,4,4-trifluorobutoxy)phenyl]-2-(trifluoromethyl)-1,3-dihydropyridin-6-one | IC50 | 8.0 [1], 158.0 [2] |
![](https://images.aatbio.com/dataset/ic50/alpha-1-6-mannosyl-glycoprotein-2-beta-n-acetylglucosaminyltransferase_4f83754e23400c9408ce6219604f5c84.svg) | 4-(4-Methylphenyl)-2-[4-(4,4,5,5,5-pentafluoropentoxy)phenyl]-5-(2H-tetrazol-5-yl)-2-(trifluoromethyl)-1,3-dihydropyridin-6-one | IC50 | 4.0 [1], 32.0 [2] |
![](https://images.aatbio.com/dataset/ic50/alpha-1-6-mannosyl-glycoprotein-2-beta-n-acetylglucosaminyltransferase_94b2d67be0926b415278cb5cf452956a.svg) | N-Cyclobutyl-4-(4-methylphenyl)-6-oxo-2-[4-(4,4,4-trifluorobutoxy)phenyl]-2-(trifluoromethyl)-1,3-dihydropyridine-5-carboxamide | IC50 | 6.0 [1], 58.0 [2] |
![](https://images.aatbio.com/dataset/ic50/alpha-1-6-mannosyl-glycoprotein-2-beta-n-acetylglucosaminyltransferase_355c5bf7706834a6a7d0953c39d66f97.svg) | N-Cyclohexyl-4-(4-methylphenyl)-6-oxo-2-[4-(4,4,4-trifluorobutoxy)phenyl]-2-(trifluoromethyl)-1,3-dihydropyridine-5-carboxamide | IC50 | 20.0 [1], 231.0 [2] |
![](https://images.aatbio.com/dataset/ic50/alpha-1-6-mannosyl-glycoprotein-2-beta-n-acetylglucosaminyltransferase_2ad0ffe75219473a9536332ff7458688.svg) | N-Methyl-4-(4-methylphenyl)-6-oxo-2-[4-(4,4,4-trifluorobutoxy)phenyl]-2-(trifluoromethyl)-1,3-dihydropyridine-5-carboxamide | IC50 | 5.0 [1], 743.0 [2] |
![](https://images.aatbio.com/dataset/ic50/alpha-1-6-mannosyl-glycoprotein-2-beta-n-acetylglucosaminyltransferase_1d16fe6ef56aa2214d725f0e91bc5c17.svg) | 2-[4-(Cyclopenten-1-yl)phenyl]-4-(4-methylphenyl)-6-oxo-N-(2H-tetrazol-5-yl)-2-(trifluoromethyl)-1,3-dihydropyridine-5-carboxamide | IC50 | 33.0 [1], 1874.0 [2] |
![](https://images.aatbio.com/dataset/ic50/alpha-1-6-mannosyl-glycoprotein-2-beta-n-acetylglucosaminyltransferase_c7db025a19a9163c3ee863842267465a.svg) | 2-[3-(Cyclohexen-1-yl)phenyl]-4-(4-methylphenyl)-6-oxo-N-(2H-tetrazol-5-yl)-2-(trifluoromethyl)-1,3-dihydropyridine-5-carboxamide | IC50 | 10.0 [1], 655.0 [2] |
![](https://images.aatbio.com/dataset/ic50/alpha-1-6-mannosyl-glycoprotein-2-beta-n-acetylglucosaminyltransferase_16e7a88044d29b35f7b825eab622ef34.svg) | 4-(4-Methylphenyl)-N-(1,2-oxazol-5-yl)-6-oxo-2-(trifluoromethyl)-2-[4-(3,3,3-trifluoropropoxy)phenyl]-1,3-dihydropyridine-5-carboxamide | IC50 | 1.0 [1], 20.0 [2] |
![](https://images.aatbio.com/dataset/ic50/alpha-1-6-mannosyl-glycoprotein-2-beta-n-acetylglucosaminyltransferase_d115dc3781c863221de792df99b96b81.svg) | 5,5-Difluoro-N-(4-methoxyphenyl)-4-(4-methylphenyl)-2-oxo-6-(trifluoromethyl)-6-[4-(3,3,3-trifluoropropoxy)phenyl]-1H-pyridine-3-carboxamide | IC50 | 127.0 [1], 1518.0 [2] |
![](https://images.aatbio.com/dataset/ic50/alpha-1-6-mannosyl-glycoprotein-2-beta-n-acetylglucosaminyltransferase_7548284686ee1eb22e33a02ca36fcd5f.svg) | 4-(2-Fluoro-4-methoxyphenyl)-5-(tetrazol-1-yl)-2-[4-(4,4,4-trifluorobutoxy)phenyl]-2-(trifluoromethyl)-1,3-dihydropyridin-6-one | IC50 | 10.0 [1], 93.0 [2] |
![](https://images.aatbio.com/dataset/ic50/alpha-1-6-mannosyl-glycoprotein-2-beta-n-acetylglucosaminyltransferase_6dba7498a58d4d42a035470ee7f1ed9d.svg) | 4-(4-Methoxyphenyl)-5-(tetrazol-1-yl)-2-[4-(4,4,4-trifluorobutoxy)phenyl]-2-(trifluoromethyl)-1,3-dihydropyridin-6-one | IC50 | 4.0 [1], 156.0 [2] |
![](https://images.aatbio.com/dataset/ic50/alpha-1-6-mannosyl-glycoprotein-2-beta-n-acetylglucosaminyltransferase_db071585ba758ffc8cd90c967c4d93fa.svg) | 4-(2,4-Dimethylphenyl)-N-(4-methoxyphenyl)-6-oxo-2-[4-(4,4,4-trifluorobutoxy)phenyl]-2-(trifluoromethyl)-1,3-dihydropyridine-5-carboxamide | IC50 | 9.0 [1], 102.0 [2] |
![](https://images.aatbio.com/dataset/ic50/alpha-1-6-mannosyl-glycoprotein-2-beta-n-acetylglucosaminyltransferase_fc0e6b55460f709e999ddc4614da16d9.svg) | N-[5,5-Difluoro-4-(4-methylphenyl)-2-oxo-6-[4-(4,4,4-trifluorobutoxy)phenyl]-6-(trifluoromethyl)-1H-pyridin-3-yl]-3-methyl-1,2-oxazole-5-carboxamide | IC50 | 3.0 [1], 11.0 [2] |
![](https://images.aatbio.com/dataset/ic50/alpha-1-6-mannosyl-glycoprotein-2-beta-n-acetylglucosaminyltransferase_55883388c0511eaab4d2a019a683b8f8.svg) | 4-Methyl-N-[4-(4-methylphenyl)-6-oxo-2-[4-(4,4,4-trifluorobutoxy)phenyl]-2-(trifluoromethyl)-1,3-dihydropyridin-5-yl]-1,2-oxazole-5-carboxamide | IC50 | 84.0 [1], 168.0 [2] |
![](https://images.aatbio.com/dataset/ic50/alpha-1-6-mannosyl-glycoprotein-2-beta-n-acetylglucosaminyltransferase_338a6d82fb64bec15c2234b80fcf555c.svg) | 6-Chloro-N-[4-(4-methylphenyl)-6-oxo-2-[4-(4,4,4-trifluorobutoxy)phenyl]-2-(trifluoromethyl)-1,3-dihydropyridin-5-yl]pyridazine-3-carboxamide | IC50 | 75.0 [1], 302.0 [2] |
![](https://images.aatbio.com/dataset/ic50/alpha-1-6-mannosyl-glycoprotein-2-beta-n-acetylglucosaminyltransferase_3c4ca341896e2cfe64b4d9fd64c85b75.svg) | N-[5,5-Difluoro-4-(4-methylphenyl)-2-oxo-6-[4-(4,4,4-trifluorobutoxy)phenyl]-6-(trifluoromethyl)-1H-pyridin-3-yl]-4-methoxybenzamide | IC50 | 47.0 [1], 1176.0 [2] |
![](https://images.aatbio.com/dataset/ic50/alpha-1-6-mannosyl-glycoprotein-2-beta-n-acetylglucosaminyltransferase_eec11baca18d387f583adc7afe080032.svg) | N-[4-[4-(Difluoromethoxy)phenyl]-6-oxo-2-[4-(4,4,4-trifluorobutoxy)phenyl]-2-(trifluoromethyl)-1,3-dihydropyridin-5-yl]-1,2-oxazole-5-carboxamide | IC50 | 2.0 [1], 8.0 [2] |
![](https://images.aatbio.com/dataset/ic50/alpha-1-6-mannosyl-glycoprotein-2-beta-n-acetylglucosaminyltransferase_a44d41bc55458706b57ac064ede1f9c7.svg) | 2-Chloro-5-fluoro-N-[4-(4-methylphenyl)-6-oxo-2-[4-(4,4,4-trifluorobutoxy)phenyl]-2-(trifluoromethyl)-1,3-dihydropyridin-5-yl]benzamide | IC50 | 57.0 [1], 724.0 [2] |
![](https://images.aatbio.com/dataset/ic50/alpha-1-6-mannosyl-glycoprotein-2-beta-n-acetylglucosaminyltransferase_195ccbb5fd22bbee814a0baf1fcc0411.svg) | N-[2-(4-Butoxyphenyl)-4-(4-methoxyphenyl)-6-oxo-2-(trifluoromethyl)-1,3-dihydropyridin-5-yl]-1,2-oxazole-5-carboxamide | IC50 | 3.0 [1], 16.0 [2] |
![](https://images.aatbio.com/dataset/ic50/alpha-1-6-mannosyl-glycoprotein-2-beta-n-acetylglucosaminyltransferase_40c311ad9b33c5fd92a8f96e2e9d9a77.svg) | 2-N-Hexadecyl-5-N-(4-methoxyphenyl)-2-methyl-4-(4-methylphenyl)-6-oxo-1,3-dihydropyridine-2,5-dicarboxamide | IC50 | 43.0 [1], 63.0 [2] |
![](https://images.aatbio.com/dataset/ic50/alpha-1-6-mannosyl-glycoprotein-2-beta-n-acetylglucosaminyltransferase_800299fda15ebfa55442c36d30930448.svg) | 5-N-(4-Methoxyphenyl)-2-methyl-4-(4-methylphenyl)-2-N-octyl-6-oxo-1,3-dihydropyridine-2,5-dicarboxamide | IC50 | 60.0 [1], 237.0 [2] |
![](https://images.aatbio.com/dataset/ic50/alpha-1-6-mannosyl-glycoprotein-2-beta-n-acetylglucosaminyltransferase_e2fe8f7517006c711d81f76f88395863.svg) | 5-N-(4-Methoxyphenyl)-2-methyl-4-(4-methylphenyl)-6-oxo-2-N-(4-phenylbutyl)-1,3-dihydropyridine-2,5-dicarboxamide | IC50 | 47.0 [1], 78.0 [2] |
![](https://images.aatbio.com/dataset/ic50/alpha-1-6-mannosyl-glycoprotein-2-beta-n-acetylglucosaminyltransferase_323915df5f152c1cc16e665a7250b1d5.svg) | 3-Bromo-N-[4-(4-methylphenyl)-6-oxo-2-[4-(4,4,4-trifluorobutoxy)phenyl]-2-(trifluoromethyl)-1,3-dihydropyridin-5-yl]-1,2-oxazole-5-carboxamide | IC50 | 2.0 [1], 24.0 [2] |
![](https://images.aatbio.com/dataset/ic50/alpha-1-6-mannosyl-glycoprotein-2-beta-n-acetylglucosaminyltransferase_a06bce4375b502761cd6f7ab69aa5401.svg) | N-[4-(4-Methylphenyl)-6-oxo-2-[4-(4,4,4-trifluorobutoxy)phenyl]-2-(trifluoromethyl)-1,3-dihydropyridin-5-yl]-3-phenylmethoxy-1,2-oxazole-5-carboxamide | IC50 | 30.0 [1], 36.0 [2] |
![](https://images.aatbio.com/dataset/ic50/alpha-1-6-mannosyl-glycoprotein-2-beta-n-acetylglucosaminyltransferase_753f174155145214e0f68c86f0651d09.svg) | N-(5-Methoxypyrazin-2-yl)-4-(4-methylphenyl)-6-oxo-2-(trifluoromethyl)-2-[4-(5,5,5-trifluoropentoxy)phenyl]-1,3-dihydropyridine-5-carboxamide | IC50 | 10.0 [1], 21.0 [2] |
![](https://images.aatbio.com/dataset/ic50/alpha-1-6-mannosyl-glycoprotein-2-beta-n-acetylglucosaminyltransferase_cb4048c994f8ac0a29467d3d1eed335a.svg) | (2S)-N-(4-Methoxyphenyl)-4-(4-methylphenyl)-6-oxo-2-[4-(4,4,4-trifluorobutoxy)phenyl]-2-(trifluoromethyl)-1,3-dihydropyridine-5-carboxamide | IC50 | 2.0 [1], 14.0 [2] |
![](https://images.aatbio.com/dataset/ic50/alpha-1-6-mannosyl-glycoprotein-2-beta-n-acetylglucosaminyltransferase_0142d2fcc62c38e04936ff212730b9d4.svg) | 2-N-Heptyl-5-N-(4-methoxyphenyl)-2-methyl-4-(4-methylphenyl)-6-oxo-1,3-dihydropyridine-2,5-dicarboxamide | IC50 | 102.0 [1], 237.0 [2] |
![](https://images.aatbio.com/dataset/ic50/alpha-1-6-mannosyl-glycoprotein-2-beta-n-acetylglucosaminyltransferase_7970ab0fb0a4202eebf919facc5f6b2d.svg) | N-(6-Methoxypyridin-3-yl)-4-(4-methylphenyl)-6-oxo-2-[4-(4,4,4-trifluorobutoxy)phenyl]-2-(trifluoromethyl)-1,3-dihydropyridine-5-carboxamide | IC50 | 5.0 [1], 11.0 [2] |
![](https://images.aatbio.com/dataset/ic50/alpha-1-6-mannosyl-glycoprotein-2-beta-n-acetylglucosaminyltransferase_4422dda1cb3d26026e8f9811a4874ff8.svg) | N-Cyclopropyl-4-(4-methylphenyl)-6-oxo-2-[4-(4,4,4-trifluorobutoxy)phenyl]-2-(trifluoromethyl)-1,3-dihydropyridine-5-carboxamide | IC50 | 21.0 [1], 94.0 [2] |
![](https://images.aatbio.com/dataset/ic50/alpha-1-6-mannosyl-glycoprotein-2-beta-n-acetylglucosaminyltransferase_e4baed254fbd5acdfc8a64d938ed6682.svg) | 4-(4-Methylphenyl)-6-oxo-2-[4-(4,4,4-trifluorobutoxy)phenyl]-N-[4-(trifluoromethoxy)phenyl]-2-(trifluoromethyl)-1,3-dihydropyridine-5-carboxamide | IC50 | 1.0 [1], 89.0 [2] |
![](https://images.aatbio.com/dataset/ic50/alpha-1-6-mannosyl-glycoprotein-2-beta-n-acetylglucosaminyltransferase_902869d9ce2a4e85d629c17f2a99ac44.svg) | N-(4-Hydroxyphenyl)-4-(4-methylphenyl)-6-oxo-2-[4-(4,4,4-trifluorobutoxy)phenyl]-2-(trifluoromethyl)-1,3-dihydropyridine-5-carboxamide | IC50 | 1.0 [1], 14.0 [2] |
![](https://images.aatbio.com/dataset/ic50/alpha-1-6-mannosyl-glycoprotein-2-beta-n-acetylglucosaminyltransferase_cdeaa3bbb64dbcf674c4ece7eead6d9e.svg) | 4-[4-(Difluoromethoxy)phenyl]-6-oxo-2-[4-(4,4,4-trifluorobutoxy)phenyl]-2-(trifluoromethyl)-1,3-dihydropyridine-5-carbonitrile | IC50 | 16.0 [1], 175.0 [2] |
![](https://images.aatbio.com/dataset/ic50/alpha-1-6-mannosyl-glycoprotein-2-beta-n-acetylglucosaminyltransferase_60f1418a13b2f29c5cfa661398ff17c2.svg) | 4-(4-Methylphenyl)-5-(2H-tetrazol-5-yl)-2-[4-(4,4,4-trifluorobutoxy)phenyl]-2-(trifluoromethyl)-1,3-dihydropyridin-6-one | IC50 | 8.0 [1], 35.0 [2] |
![](https://images.aatbio.com/dataset/ic50/alpha-1-6-mannosyl-glycoprotein-2-beta-n-acetylglucosaminyltransferase_8c863cd9289cda355e09d83529e62488.svg) | 4-(4-Methylphenyl)-6-oxo-2-[4-(4,4,4-trifluorobutoxy)phenyl]-2-(trifluoromethyl)-1,3-dihydropyridine-5-carbonitrile | IC50 | 171.0 [1], 5073.0 [2] |
![](https://images.aatbio.com/dataset/ic50/alpha-1-6-mannosyl-glycoprotein-2-beta-n-acetylglucosaminyltransferase_775bf04ee6eaa67687ad8df57eeb4d01.svg) | 4-(4-Methylphenyl)-6-oxo-2-(trifluoromethyl)-2-[4-(3,3,3-trifluoropropoxy)phenyl]-1,3-dihydropyridine-5-carbonitrile | IC50 | 14.0 [1], 91.0 [2] |
![](https://images.aatbio.com/dataset/ic50/alpha-1-6-mannosyl-glycoprotein-2-beta-n-acetylglucosaminyltransferase_582b9f439a6591bdc25bd89beab37eed.svg) | 4-[4-(Difluoromethoxy)phenyl]-5-(tetrazol-1-yl)-2-[4-(4,4,4-trifluorobutoxy)phenyl]-2-(trifluoromethyl)-1,3-dihydropyridin-6-one | IC50 | 6.0 [1], 53.0 [2] |
![](https://images.aatbio.com/dataset/ic50/alpha-1-6-mannosyl-glycoprotein-2-beta-n-acetylglucosaminyltransferase_85546c77ca21461831b2fb691b5563a2.svg) | 5-Methyl-N-[4-(4-methylphenyl)-6-oxo-2-[4-(4,4,4-trifluorobutoxy)phenyl]-2-(trifluoromethyl)-1,3-dihydropyridin-5-yl]-1,3,4-oxadiazole-2-carboxamide | IC50 | 8.0 [1], 34.0 [2] |
![](https://images.aatbio.com/dataset/ic50/alpha-1-6-mannosyl-glycoprotein-2-beta-n-acetylglucosaminyltransferase_1f4fc1220ed81126bbf6ddb4f925e684.svg) | 2-Methyl-N-[(2S)-4-(4-methylphenyl)-6-oxo-2-[4-(4,4,4-trifluorobutoxy)phenyl]-2-(trifluoromethyl)-1,3-dihydropyridin-5-yl]benzamide | IC50 | 24.0 [1], 672.0 [2] |
![](https://images.aatbio.com/dataset/ic50/alpha-1-6-mannosyl-glycoprotein-2-beta-n-acetylglucosaminyltransferase_d26609a46e223496cfe7b972fbcb9e6f.svg) | (2R)-4-(4-Methylphenyl)-5-(2H-tetrazol-5-yl)-2-[4-(4,4,4-trifluorobutoxy)phenyl]-2-(trifluoromethyl)-1,3-dihydropyridin-6-one | IC50 | 261.0 [1], 1400.0 [2] |
![](https://images.aatbio.com/dataset/ic50/alpha-1-6-mannosyl-glycoprotein-2-beta-n-acetylglucosaminyltransferase_b7ae7a1a89ae25f1b459e72c4def1fa3.svg) | 2-(4-Butoxyphenyl)-4-(4-methylphenyl)-6-oxo-2-(trifluoromethyl)-1,3-dihydropyridine-5-carbonitrile | IC50 | 21.0 [1], 309.0 [2] |
![](https://images.aatbio.com/dataset/ic50/alpha-1-6-mannosyl-glycoprotein-2-beta-n-acetylglucosaminyltransferase_b5b0a70992efb5db127f99a1d50978c7.svg) | 4-(4-Methylphenyl)-5-nitro-2-[4-(4,4,4-trifluorobutoxy)phenyl]-2-(trifluoromethyl)-1,3-dihydropyridin-6-one | IC50 | 35.0 [1], 3333.0 [2] |
![](https://images.aatbio.com/dataset/ic50/alpha-1-6-mannosyl-glycoprotein-2-beta-n-acetylglucosaminyltransferase_8305ce57ea3a148833ea71c20925bfa2.svg) | 4-(4-Methylphenyl)-2-[4-(4,4,4-trifluorobutoxy)phenyl]-2-(trifluoromethyl)-5-[5-(trifluoromethyl)-1,3,4-oxadiazol-2-yl]-1,3-dihydropyridin-6-one | IC50 | 138.0 [1], 2716.0 [2] |
![](https://images.aatbio.com/dataset/ic50/alpha-1-6-mannosyl-glycoprotein-2-beta-n-acetylglucosaminyltransferase_016d4505a3eb518c037c6eaa8b42c730.svg) | 4-(4-Methylphenyl)-5-(2H-tetrazol-5-yl)-2-[4-(6,6,6-trifluorohexoxy)phenyl]-2-(trifluoromethyl)-1,3-dihydropyridin-6-one | IC50 | 48.0 [1], 407.0 [2] |
![](https://images.aatbio.com/dataset/ic50/alpha-1-6-mannosyl-glycoprotein-2-beta-n-acetylglucosaminyltransferase_4f06e999c12bfe1ede0011b29f6a0223.svg) | 2-Methyl-4-(4-methylphenyl)-6-oxo-2-[4-(4,4,4-trifluorobutoxy)phenyl]-N-[4-(trifluoromethoxy)phenyl]-1,3-dihydropyridine-5-carboxamide | IC50 | 13.0 [1], 48.0 [2] |
![](https://images.aatbio.com/dataset/ic50/alpha-1-6-mannosyl-glycoprotein-2-beta-n-acetylglucosaminyltransferase_304a94d538757b109e29eab2f9c30f8a.svg) | (6S)-N-(4-Methoxyphenyl)-4-(4-methylphenyl)-2-oxo-6-[4-(4,4,4-trifluorobutoxy)phenyl]-6-(trifluoromethyl)piperidine-3-carboxamide | IC50 | 25.0 [1], 416.0 [2] |
![](https://images.aatbio.com/dataset/ic50/alpha-1-6-mannosyl-glycoprotein-2-beta-n-acetylglucosaminyltransferase_c9067cc73cc158ed70c83bbd8412663d.svg) | (6S)-3-Fluoro-4-(4-methoxyphenyl)-2-oxo-6-[4-(4,4,4-trifluorobutoxy)phenyl]-6-(trifluoromethyl)-1H-pyridine-3-carbonitrile | IC50 | 2049.0 [1], 33330.0 [2] |
![](https://images.aatbio.com/dataset/ic50/alpha-1-6-mannosyl-glycoprotein-2-beta-n-acetylglucosaminyltransferase_5f749caa02f4fa2c8a0cda3075222bc6.svg) | (6R)-3-Fluoro-4-(4-methoxyphenyl)-2-oxo-6-[4-(4,4,4-trifluorobutoxy)phenyl]-6-(trifluoromethyl)-1H-pyridine-3-carbonitrile | IC50 | 2049.0 [1], 33330.0 [2] |