 | Crizotinib | IC50 | 165.0 [1] |
| Crizotinib | Ki | 0.74 [1], 8.2 [2] |
 | Ceritinib | IC50 | 14.0 [1] |
 | Unii-76pnd635L1 | IC50 | 3.5 [1] |
| Unii-76pnd635L1 | Ki | 0.1 [1], 0.2 [2] |
 | Staurosporine | IC50 | 2.36 [1] |
 | Lorlatinib | IC50 | 9.0 [1] |
| Lorlatinib | Ki | 0.07 [1], 0.7 [2], 8.2 [3] |
 | 6,6-Dimethyl-8-[1-(oxan-4-ylmethyl)piperidin-4-yl]-11-oxo-5H-benzo[b]carbazole-3-carbonitrile | IC50 | 3.9 [1] |
 | 4-(4-Methylphenoxy)-7-(1-piperidin-4-ylpyrazol-4-yl)quinoline | IC50 | 50.2 [1] |
| 4-(4-Methylphenoxy)-7-(1-piperidin-4-ylpyrazol-4-yl)quinoline | Ki | 21.99 [1], 729046655.0 [2] |
 | Nvp-tae 684 | IC50 | 3.0 [1] |
 | 5-Chloro-2-N-[2-methoxy-4-[4-[(4-methylpiperazin-1-yl)methyl]triazol-1-yl]phenyl]-4-N-(2-propan-2-ylsulfonylphenyl)pyrimidine-2,4-diamine | IC50 | 3.0 [1] |
 | 4-[7-(1-Piperidin-4-ylpyrazol-4-yl)quinolin-4-yl]oxyphenol | IC50 | 11.5 [1] |
 | 4-(4-Methoxyphenoxy)-7-(1-piperidin-4-ylpyrazol-4-yl)quinoline | IC50 | 42.2 [1] |
 | N-[2-[3-[[5-Chloro-4-(2-propan-2-ylsulfonylanilino)pyrimidin-2-yl]amino]-4-methoxyanilino]-2-oxoethyl]-2,4-dihydroxy-5-propan-2-ylbenzamide | IC50 | 2.7 [1] |
 | 5-(1,3-Dimethylpyrazol-4-yl)-3-[(1R)-1-[5-fluoro-2-(triazol-2-yl)phenyl]ethoxy]pyridin-2-amine | IC50 | 14.0 [1], 176.0 [2] |
| 5-(1,3-Dimethylpyrazol-4-yl)-3-[(1R)-1-[5-fluoro-2-(triazol-2-yl)phenyl]ethoxy]pyridin-2-amine | Ki | 0.2 [1], 2.6 [2] |
 | 3-[(1R)-1-[5-Fluoro-2-(triazol-2-yl)phenyl]ethoxy]-5-(3-methyltriazol-4-yl)pyridin-2-amine | IC50 | 249.0 [1], 2650.0 [2] |
| 3-[(1R)-1-[5-Fluoro-2-(triazol-2-yl)phenyl]ethoxy]-5-(3-methyltriazol-4-yl)pyridin-2-amine | Ki | 9.0 [1], 70.0 [2] |
 | 5-Chloro-2-N-[4-[2-(dimethylamino)ethyl]-2-methoxy-5-methylphenyl]-4-N-(2-propan-2-ylsulfonylphenyl)pyrimidine-2,4-diamine | IC50 | 1.1 [1] |
 | Alectinib | IC50 | 1.9 [1], 5.3 [2], 11.5 [3], 15.2 [4], 19.0 [5] |
 | Entrectinib | IC50 | 12.0 [1], 55.0 [2] |
| Entrectinib | Ki | 6.2 [1] |
 | CID 25229528 | IC50 | 14.0 [1], 45.0 [2], 225.0 [3] |
 | N-[5-[[5-Chloro-4-(2-propan-2-ylsulfonylanilino)pyrimidin-2-yl]amino]-4-methoxy-2-(4-methyl-1,4-diazepan-1-yl)phenyl]prop-2-enamide | IC50 | 0.59 [1], 0.82 [2], 0.92 [3], 1.0 [4], 9.8 [5] |
 | 5-[1-(7-Azaspiro[3.5]nonan-2-yl)pyrazol-4-yl]-3-[(1R)-1-(2,6-dichloro-3-fluorophenyl)ethoxy]pyridin-2-amine | IC50 | 1.2 [1], 1.4 [2], 1.5 [3], 1.8 [4] |
 | Cep-37440 | IC50 | 3.1 [1], 22.0 [2], 85.0 [3], 175.0 [4] |
 | (1S,2S,3R,4R)-3-[[5-Chloro-2-[[(7S)-4-methoxy-7-morpholin-4-yl-6,7,8,9-tetrahydro-5H-benzo[7]annulen-3-yl]amino]pyrimidin-4-yl]amino]bicyclo[2.2.1]hept-5-ene-2-carboxamide | IC50 | 1.9 [1], 20.0 [2] |
 | 2-Amino-N-[3-[[5-chloro-4-(2-propan-2-ylsulfonylanilino)pyrimidin-2-yl]amino]phenyl]acetamide | IC50 | 2.7 [1], 15.3 [2] |
 | 5-Chloro-2-N-(5-methyl-4-piperidin-4-yl-2-propan-2-yloxyphenyl)-4-N-(1-methyl-3-propan-2-ylsulfonylpyrazol-4-yl)pyrimidine-2,4-diamine | IC50 | 6.0 [1], 8.0 [2], 16.0 [3], 20.0 [4] |
 | 5-Chloro-2-N-[2-cyclopropyloxy-5-methyl-4-(1-methylpiperidin-4-yl)phenyl]-4-N-(1-methyl-3-propan-2-ylsulfonylpyrazol-4-yl)pyrimidine-2,4-diamine | IC50 | 1.0 [1], 2.0 [2], 4.0 [3] |
 | 8-[1-[(4-Hydroxyoxan-4-yl)methyl]piperidin-4-yl]-6,6-dimethyl-11-oxo-5H-benzo[b]carbazole-3-carbonitrile | IC50 | 16.4 [1], 100.0 [2] |
 | 2-[8-[[5-Chloro-4-(2-methoxy-4-morpholin-4-ylanilino)pyrimidin-2-yl]amino]-7-methoxy-1,2,4,5-tetrahydro-3-benzazepin-3-yl]-N,N-dimethylacetamide | IC50 | 4.0 [1], 30.0 [2] |
 | 5-Chloro-2-N-[7-methoxy-3-(2-methoxyethyl)-1,2,4,5-tetrahydro-3-benzazepin-8-yl]-4-N-(2-methoxy-4-morpholin-4-ylphenyl)pyrimidine-2,4-diamine | IC50 | 7.0 [1], 150.0 [2] |
 | 5-Chloro-2-N-[2-cyclopropyloxy-4-[4-(diethylamino)cyclohexyl]-5-methylphenyl]-4-N-(1-methyl-3-propan-2-ylsulfonylpyrazol-4-yl)pyrimidine-2,4-diamine | IC50 | 8.0 [1], 9.0 [2], 12.0 [3], 17.0 [4] |
 | 5-Chloro-2-N-[4-[4-(cyclopropylamino)cyclohexyl]-2-cyclopropyloxy-5-methylphenyl]-4-N-(1-methyl-3-propan-2-ylsulfonylpyrazol-4-yl)pyrimidine-2,4-diamine | IC50 | 8.0 [1], 9.0 [2], 18.0 [3], 20.0 [4] |
 | 5-Chloro-2-N-[2-cyclopropyloxy-5-methyl-4-[4-(propan-2-ylamino)cyclohexyl]phenyl]-4-N-(1-methyl-3-propan-2-ylsulfonylpyrazol-4-yl)pyrimidine-2,4-diamine | IC50 | 5.0 [1], 9.0 [2], 10.0 [3] |
 | 3-[(1r)-1-(5-Fluoro-2-Methoxyphenyl)ethoxy]-5-(1-Methyl-1h-1,2,3-Triazol-5-Yl)pyridin-2-Amine | IC50 | 95.0 [1], 3200.0 [2] |
| 3-[(1r)-1-(5-Fluoro-2-Methoxyphenyl)ethoxy]-5-(1-Methyl-1h-1,2,3-Triazol-5-Yl)pyridin-2-Amine | Ki | 4.0 [1], 38.0 [2] |
 | 19-Amino-13-fluoro-3,5,8-trimethyl-17-oxa-4,5,8,20-tetrazatetracyclo[16.3.1.02,6.010,15]docosa-1(22),2(6),3,10(15),11,13,18,20-octaen-9-one | IC50 | 6.4 [1], 97.0 [2] |
| 19-Amino-13-fluoro-3,5,8-trimethyl-17-oxa-4,5,8,20-tetrazatetracyclo[16.3.1.02,6.010,15]docosa-1(22),2(6),3,10(15),11,13,18,20-octaen-9-one | Ki | 0.2 [1], 1.9 [2] |
 | 14-Fluoro-3-methyl-10,18-dioxa-3,4,21-triazatetracyclo[17.3.1.02,6.011,16]tricosa-1(23),2(6),4,11(16),12,14,19,21-octaen-20-amine | IC50 | 86.0 [1], 654.0 [2] |
| 14-Fluoro-3-methyl-10,18-dioxa-3,4,21-triazatetracyclo[17.3.1.02,6.011,16]tricosa-1(23),2(6),4,11(16),12,14,19,21-octaen-20-amine | Ki | 0.38 [1], 29.0 [2] |
 | 20-Amino-14-fluoro-10,18-dioxa-4,5,21-triazatetracyclo[17.3.1.02,6.011,16]tricosa-1(23),2(6),3,11(16),12,14,19,21-octaene-3-carbonitrile | IC50 | 15.0 [1], 112.0 [2] |
| 20-Amino-14-fluoro-10,18-dioxa-4,5,21-triazatetracyclo[17.3.1.02,6.011,16]tricosa-1(23),2(6),3,11(16),12,14,19,21-octaene-3-carbonitrile | Ki | 0.1 [1], 0.22 [2] |
 | 19-Amino-13-fluoro-9,17-dioxa-4,5,20-triazatetracyclo[16.3.1.02,6.010,15]docosa-1(22),2(6),3,10(15),11,13,18,20-octaene-3-carbonitrile | IC50 | 22.0 [1], 101.0 [2] |
| 19-Amino-13-fluoro-9,17-dioxa-4,5,20-triazatetracyclo[16.3.1.02,6.010,15]docosa-1(22),2(6),3,10(15),11,13,18,20-octaene-3-carbonitrile | Ki | 0.36 [1], 1.6 [2] |
 | 15-Fluoro-3-methyl-11,19-dioxa-3,4,22-triazatetracyclo[18.3.1.02,6.012,17]tetracosa-1(24),2(6),4,12(17),13,15,20,22-octaen-21-amine | IC50 | 524.0 [1], 3655.0 [2] |
| 15-Fluoro-3-methyl-11,19-dioxa-3,4,22-triazatetracyclo[18.3.1.02,6.012,17]tetracosa-1(24),2(6),4,12(17),13,15,20,22-octaen-21-amine | Ki | 5.0 [1], 36.0 [2] |
 | 2-[(1r)-1-{[3-Amino-6-(2-Methoxypyridin-3-Yl)pyrazin-2-Yl]oxy}ethyl]-4-Fluoro-N-Methylbenzamide | IC50 | 16.0 [1], 312.0 [2] |
| 2-[(1r)-1-{[3-Amino-6-(2-Methoxypyridin-3-Yl)pyrazin-2-Yl]oxy}ethyl]-4-Fluoro-N-Methylbenzamide | Ki | 0.85 [1], 8.2 [2] |
 | 3-[(1R)-1-[5-Fluoro-2-(triazol-2-yl)phenyl]ethoxy]-5-(3-methylsulfonylphenyl)pyridin-2-amine | IC50 | 4.6 [1], 54.0 [2] |
| 3-[(1R)-1-[5-Fluoro-2-(triazol-2-yl)phenyl]ethoxy]-5-(3-methylsulfonylphenyl)pyridin-2-amine | Ki | 0.2 [1], 1.4 [2] |
 | 3-[(1R)-1-[5-Fluoro-2-(triazol-2-yl)phenyl]ethoxy]-5-(2-methoxypyridin-3-yl)pyrazin-2-amine | IC50 | 9.7 [1], 53.0 [2] |
| 3-[(1R)-1-[5-Fluoro-2-(triazol-2-yl)phenyl]ethoxy]-5-(2-methoxypyridin-3-yl)pyrazin-2-amine | Ki | 0.2 [1], 0.7 [2] |
 | (16R)-19-Amino-13-fluoro-3-methoxy-5,8,16-trimethyl-17-oxa-4,5,8,20-tetrazatetracyclo[16.3.1.02,6.010,15]docosa-1(22),2(6),3,10(15),11,13,18,20-octaen-9-one | IC50 | 0.18 [1], 2.1 [2] |
| (16R)-19-Amino-13-fluoro-3-methoxy-5,8,16-trimethyl-17-oxa-4,5,8,20-tetrazatetracyclo[16.3.1.02,6.010,15]docosa-1(22),2(6),3,10(15),11,13,18,20-octaen-9-one | Ki | 0.1 [1], 0.2 [2] |
 | (17R)-20-Amino-14-fluoro-9,17-dimethyl-4-methylsulfonyl-18-oxa-9,21-diazatetracyclo[17.3.1.02,7.011,16]tricosa-1(23),2(7),3,5,11(16),12,14,19,21-nonaen-10-one | IC50 | 1.3 [1], 21.0 [2] |
| (17R)-20-Amino-14-fluoro-9,17-dimethyl-4-methylsulfonyl-18-oxa-9,21-diazatetracyclo[17.3.1.02,7.011,16]tricosa-1(23),2(7),3,5,11(16),12,14,19,21-nonaen-10-one | Ki | 0.07 [1], 0.4 [2] |
 | (16R)-19-Amino-13-fluoro-3,5,8,16-tetramethyl-17-oxa-4,5,8,20-tetrazatetracyclo[16.3.1.02,6.010,15]docosa-1(22),2(6),3,10(15),11,13,18,20-octaen-9-one | IC50 | 0.7 [1], 14.0 [2] |
| (16R)-19-Amino-13-fluoro-3,5,8,16-tetramethyl-17-oxa-4,5,8,20-tetrazatetracyclo[16.3.1.02,6.010,15]docosa-1(22),2(6),3,10(15),11,13,18,20-octaen-9-one | Ki | 0.2 [1], 0.29 [2] |
 | 2-[(1R)-1-[2-Amino-5-(1,3-dimethylpyrazol-4-yl)pyridin-3-yl]oxyethyl]-4-fluoro-N-methylbenzamide | IC50 | 116.0 [1], 1665.0 [2] |
| 2-[(1R)-1-[2-Amino-5-(1,3-dimethylpyrazol-4-yl)pyridin-3-yl]oxyethyl]-4-fluoro-N-methylbenzamide | Ki | 2.8 [1], 35.0 [2] |
 | (16R)-19-Amino-13-fluoro-4,16-dimethyl-9,17-dioxa-4,5,20-triazatetracyclo[16.3.1.02,6.010,15]docosa-1(22),2,5,10(15),11,13,18,20-octaene-3-carbonitrile | IC50 | 1.0 [1], 20.0 [2] |
| (16R)-19-Amino-13-fluoro-4,16-dimethyl-9,17-dioxa-4,5,20-triazatetracyclo[16.3.1.02,6.010,15]docosa-1(22),2,5,10(15),11,13,18,20-octaene-3-carbonitrile | Ki | 0.1 [1], 0.57 [2] |
 | (17R)-20-Amino-14-fluoro-4,17-dimethyl-10,18-dioxa-4,5,21-triazatetracyclo[17.3.1.02,6.011,16]tricosa-1(23),2,5,11(16),12,14,19,21-octaene-3-carbonitrile | IC50 | 0.9 [1], 21.0 [2] |
| (17R)-20-Amino-14-fluoro-4,17-dimethyl-10,18-dioxa-4,5,21-triazatetracyclo[17.3.1.02,6.011,16]tricosa-1(23),2,5,11(16),12,14,19,21-octaene-3-carbonitrile | Ki | 0.1 [1], 0.62 [2] |
 | (16R)-19-Amino-13-fluoro-3,5,8,16-tetramethyl-17-oxa-4,5,8,20,22-pentazatetracyclo[16.3.1.02,6.010,15]docosa-1(21),2(6),3,10(15),11,13,18(22),19-octaen-9-one | IC50 | 0.21 [1], 1.4 [2] |
| (16R)-19-Amino-13-fluoro-3,5,8,16-tetramethyl-17-oxa-4,5,8,20,22-pentazatetracyclo[16.3.1.02,6.010,15]docosa-1(21),2(6),3,10(15),11,13,18(22),19-octaen-9-one | Ki | 0.1 [1], 0.2 [2] |
 | (16S)-19-Amino-13-fluoro-3,5,8,16-tetramethyl-17-oxa-4,5,8,20,22-pentazatetracyclo[16.3.1.02,6.010,15]docosa-1(21),2(6),3,10(15),11,13,18(22),19-octaen-9-one | IC50 | 156.0 [1], 1230.0 [2] |
| (16S)-19-Amino-13-fluoro-3,5,8,16-tetramethyl-17-oxa-4,5,8,20,22-pentazatetracyclo[16.3.1.02,6.010,15]docosa-1(21),2(6),3,10(15),11,13,18(22),19-octaen-9-one | Ki | 17.0 [1], 61.0 [2] |
 | (16R)-19-Amino-13-fluoro-3-methoxy-5,8,16-trimethyl-17-oxa-4,5,8,20,22-pentazatetracyclo[16.3.1.02,6.010,15]docosa-1(21),2(6),3,10(15),11,13,18(22),19-octaen-9-one | IC50 | 0.11 [1], 0.75 [2] |
| (16R)-19-Amino-13-fluoro-3-methoxy-5,8,16-trimethyl-17-oxa-4,5,8,20,22-pentazatetracyclo[16.3.1.02,6.010,15]docosa-1(21),2(6),3,10(15),11,13,18(22),19-octaen-9-one | Ki | 0.02 [1], 0.08 [2] |
 | (17R)-20-Amino-14-fluoro-9,17-dimethyl-4-methylsulfonyl-18-oxa-9,21,23-triazatetracyclo[17.3.1.02,7.011,16]tricosa-1(22),2(7),3,5,11(16),12,14,19(23),20-nonaen-10-one | IC50 | 0.34 [1], 1.9 [2] |
| (17R)-20-Amino-14-fluoro-9,17-dimethyl-4-methylsulfonyl-18-oxa-9,21,23-triazatetracyclo[17.3.1.02,7.011,16]tricosa-1(22),2(7),3,5,11(16),12,14,19(23),20-nonaen-10-one | Ki | 0.1 [1], 0.12 [2] |
 | 9-Ethyl-6,6-dimethyl-8-[4-(oxetan-3-yl)piperazin-1-yl]-11-oxo-5H-benzo[b]carbazole-3-carbonitrile | IC50 | 2.9 [1], 7.15 [2] |
 | N-[2-[2-[4-[4-[(2S)-2-Hydroxypropyl]piperazin-1-yl]-2-methoxyanilino]pyrrolo[2,1-f][1,2,4]triazin-7-yl]phenyl]-N-methylmethanesulfonamide | IC50 | 9.0 [1], 10.0 [2] |
 | 9-Ethyl-6,6-dimethyl-8-[1-(oxan-4-ylmethyl)-3,6-dihydro-2H-pyridin-4-yl]-11-oxo-5H-benzo[b]carbazole-3-carbonitrile | IC50 | 2.3 [1], 11.2 [2], 49.0 [3] |
 | 9-Ethyl-6,6-dimethyl-8-[1-(oxane-4-carbonyl)-3,6-dihydro-2H-pyridin-4-yl]-11-oxo-5H-benzo[b]carbazole-3-carbonitrile | IC50 | 1.7 [1], 18.0 [2], 126.0 [3] |
 | CID 138108958 | IC50 | 10.0 [1], 40.0 [2], 50.0 [3] |
 | 6,6-Dimethyl-8-[1-(oxetan-3-yl)piperidin-4-yl]-11-oxo-5H-benzo[b]carbazole-3-carbonitrile | IC50 | 1.5 [1], 1.53 [2] |
 | N-[2-[2-[2-[4-[4-[[5-Chloro-4-(2-propan-2-ylsulfonylanilino)pyrimidin-2-yl]amino]-3-methoxyphenyl]piperazin-1-yl]ethoxy]ethoxy]ethyl]-2-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]amino]acetamide | IC50 | 10.0 [1], 50.0 [2], 180.0 [3] |
 | N-[2-[[5-Chloro-2-[[2-methoxy-6-(4-methylpiperazin-1-yl)pyridin-3-yl]amino]pyrimidin-4-yl]amino]phenyl]methanesulfonamide | IC50 | 1300.0 [1], 2100.0 [2], 3900.0 [3] |
 | N-[1-[3-[[5-Chloro-4-(2-propan-2-ylsulfonylanilino)pyrimidin-2-yl]amino]-4-methoxyanilino]-1-oxo-3-phenylpropan-2-yl]-2,4-dihydroxy-5-propan-2-ylbenzamide | IC50 | 7.8 [1], 65.0 [2], 81.0 [3] |
 | N-[2-[3-[[5-Chloro-4-(2-dimethylphosphorylanilino)pyrimidin-2-yl]amino]-4-methoxyanilino]-2-oxoethyl]-2,4-dihydroxy-5-propan-2-ylbenzamide | IC50 | 1.5 [1], 5.0 [2], 7.8 [3] |
 | 4-[4-[[4-[2-[[2-[3-[[5-Chloro-4-(2-propan-2-ylsulfonylanilino)pyrimidin-2-yl]amino]-4-methoxyanilino]-2-oxoethyl]amino]-2-oxoethyl]piperazin-1-yl]methyl]phenyl]-5-(2,4-dihydroxy-5-propan-2-ylphenyl)-N-ethyl-1,2-oxazole-3-carboxamide | IC50 | 6.9 [1], 8.7 [2], 36.4 [3] |
 | 4-[4-[[4-[2-[3-[[5-Chloro-4-(2-propan-2-ylsulfonylanilino)pyrimidin-2-yl]amino]-4-methoxyanilino]-2-oxoethyl]piperazin-1-yl]methyl]phenyl]-5-(2,4-dihydroxy-5-propan-2-ylphenyl)-N-ethyl-1,2-oxazole-3-carboxamide | IC50 | 6.2 [1], 17.3 [2], 85.5 [3] |
 | N-[2-[3-[[5-Chloro-4-(2-propan-2-ylsulfonylanilino)pyrimidin-2-yl]amino]-4-fluoroanilino]-2-oxoethyl]-2,4-dihydroxy-5-propan-2-ylbenzamide | IC50 | 1.0 [1], 14.0 [2], 15.5 [3] |
 | N-[2-[[5-Chloro-2-[[6-(3-hydroxyazetidin-1-yl)-2-methoxypyridin-3-yl]amino]pyrimidin-4-yl]amino]phenyl]methanesulfonamide | IC50 | 1400.0 [1], 2000.0 [2], 5200.0 [3] |
 | N-[2-[[5-Chloro-2-[[6-(4-methylpiperazin-1-yl)-2-propan-2-yloxypyridin-3-yl]amino]pyrimidin-4-yl]amino]phenyl]methanesulfonamide | IC50 | 4200.0 [1], 4800.0 [2], 9400.0 [3] |
 | N-[2-[[5-Chloro-2-[[6-[4-(2-hydroxyethyl)piperazin-1-yl]-2-methoxypyridin-3-yl]amino]pyrimidin-4-yl]amino]phenyl]methanesulfonamide | IC50 | 2200.0 [1], 3200.0 [2], 7800.0 [3] |
 | N-[2-[[5-Chloro-2-[[2-methoxy-6-(4-methylpiperazin-1-yl)pyridin-3-yl]amino]pyrimidin-4-yl]amino]phenyl]cyclopropanesulfonamide | IC50 | 3900.0 [1], 6000.0 [2] |
 | N-[2-[[5-Chloro-2-[(2-methoxy-6-thiomorpholin-4-ylpyridin-3-yl)amino]pyrimidin-4-yl]amino]phenyl]methanesulfonamide | IC50 | 1600.0 [1], 2800.0 [2], 7900.0 [3] |
 | N-[5-[(3,5-Difluorophenyl)methyl]-1H-indazol-3-yl]-4-(4-methylpiperazin-1-yl)benzamide | IC50 | 73.0 [1], 207.0 [2] |
 | 2-(Cyclohexylamino)-N-[5-[(3,5-difluorophenyl)methyl]-1H-indazol-3-yl]-4-(4-methylpiperazin-1-yl)benzamide | IC50 | 560.0 [1], 1771.0 [2] |
 | N-[5-[(3,5-Difluorophenyl)methyl]-1H-indazol-3-yl]-2-(2-methoxyethylamino)-4-(4-methylpiperazin-1-yl)benzamide | IC50 | 210.0 [1], 411.0 [2] |
 | 3-[1-(2,5-Difluorobenzyl)-1h-Pyrazol-4-Yl]-5-(1-Methyl-1h-Pyrazol-4-Yl)-1h-Pyrrolo[2,3-B]pyridine | IC50 | 29.0 [1], 124.0 [2], 1592.0 [3] |
 | 3-[1-[(3-Fluorophenyl)methyl]pyrazol-4-yl]-5-(1-methylpyrazol-4-yl)-1H-pyrrolo[2,3-b]pyridine | IC50 | 5.6 [1], 35.0 [2], 138.5 [3] |
 | 3-[1-[(4-Fluorophenyl)methyl]pyrazol-4-yl]-5-(1-methylpyrazol-4-yl)-1H-pyrrolo[2,3-b]pyridine | IC50 | 70.0 [1], 256.4 [2], 3011.0 [3] |
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