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Aldo-keto reductase family 1 member B10 Inhibitors (IC50, Ki)

Structure
▲
▼
Compound Name
▲
▼
Standard Type
▲
▼
Standard Values (in nM)
▲
▼
2-Methoxy-4-hydroxycinnamic acid 3-(3-hydroxyphenyl)propyl esterIC506.2 [1], 300.0 [2]
2-Methoxy-4-hydroxycinnamic acid 3-(3-hydroxyphenyl)propyl esterKi5.8 [1]
Oleanolic acidIC5090.0 [1], 4000.0 [2]
Oleanolic acidKi72.0 [1], 160.0 [2], 660.0 [3], 940.0 [4], 3560.0 [5]
Ursolic acidIC504000.0 [1]
Ursolic acidKi2000.0 [1], 2100.0 [2], 2800.0 [3], 3700.0 [4], 6000.0 [5]
N-Benzyl-7-hydroxy-2-(4-methoxyphenyl)iminochromene-3-carboxamideIC504.7 [1]
N-Benzyl-7-hydroxy-2-(4-methoxyphenyl)iminochromene-3-carboxamideKi1.3 [1], 3.8 [2], 51.0 [3]
TolrestatIC5011.6 [1], 54.0 [2]
TolrestatKi50.0 [1]
ApigeninIC506600.0 [1], 37100.0 [2]
ApigeninKi6000.0 [1]
Flufenamic acidIC50760.0 [1], 96000.0 [2]
(2Z)-7-Hydroxy-2-[(4-methoxyphenyl)imino]-N-(pyridin-2-yl)-2H-chromene-3-carboxamideIC506.0 [1]
(2Z)-7-Hydroxy-2-[(4-methoxyphenyl)imino]-N-(pyridin-2-yl)-2H-chromene-3-carboxamideKi2.7 [1]
LuteolinIC509200.0 [1], 107800.0 [2]
Isolithocholic acidIC5027.0 [1]
Isolithocholic acidKi15.0 [1]
Caffeic acid phenethyl esterIC5080.0 [1]
Caffeic acid phenethyl esterKi46.0 [1]
EpalrestatIC50330.0 [1]
7-HydroxyflavoneIC508300.0 [1], 160000.0 [2]
ZopolrestatIC50620.0 [1], 2360.0 [2]
3-((4-(Trifluoromethyl)Phenyl)Amino)Benzoic AcidIC5050000.0 [1]
(2Z)-2-[(2,5-Dimethoxyphenyl)imino]-7-hydroxy-N-(pyridin-2-yl)-2H-chromene-3-carboxamideIC5022.0 [1]
(2Z)-2-[(2,5-Dimethoxyphenyl)imino]-7-hydroxy-N-(pyridin-2-yl)-2H-chromene-3-carboxamideKi16.0 [1]
3-[(4-Nitrophenyl)amino]benzoic AcidIC5046000.0 [1]
3-(4-Acetylanilino)benzoic acidIC5037100.0 [1]
3-[(4-Bromophenyl)Amino]Benzoic AcidIC5050000.0 [1]
3-(4-Tert-butylanilino)benzoic acidIC5015000.0 [1]
(2Z)-2-[(3,4-Dimethoxyphenyl)imino]-7-hydroxy-N-(6-methylpyridin-2-yl)-2H-chromene-3-carboxamideIC5036.0 [1]
(2Z)-2-[(3,4-Dimethoxyphenyl)imino]-7-hydroxy-N-(6-methylpyridin-2-yl)-2H-chromene-3-carboxamideKi24.0 [1]
(2Z)-2-[(2,4-Dimethoxyphenyl)imino]-7-hydroxy-N-(pyridin-2-yl)-2H-chromene-3-carboxamideIC5015.0 [1]
(2Z)-2-[(2,4-Dimethoxyphenyl)imino]-7-hydroxy-N-(pyridin-2-yl)-2H-chromene-3-carboxamideKi12.0 [1]
7-Hydroxy-N-[3-(4-hydroxyphenyl)propyl]-2-oxochromene-3-carboxamideIC504.2 [1]
7-Hydroxy-N-[3-(4-hydroxyphenyl)propyl]-2-oxochromene-3-carboxamideKi2.3 [1]
DiclofenacIC501900.0 [1]
DaidzeinIC5032200.0 [1]
EnoxoloneIC504900.0 [1]
Chlorogenic acidIC507900.0 [1]
Caffeic acidIC5090000.0 [1]
Mefenamic acidIC501600.0 [1]
Betulinic acidIC502000.0 [1]
4-Hydroxycinnamic acidIC5063000.0 [1]
SorbinilIC509600.0 [1]
Biochanin AIC5036100.0 [1]
Maslinic acidIC50630.0 [1]
Asiatic acidIC505900.0 [1]
BisdemethoxycurcuminIC5060.0 [1]
3,5-Dicaffeoylquinic acidIC50130.0 [1]
Artepillin CIC5053000.0 [1]
3,4-Dicaffeoylquinic acidIC50240.0 [1]
ErythrodiolIC5030000.0 [1]
Benzyl caffeateIC50210.0 [1]
MinalrestatIC50740.0 [1]
(E)-3-(4-Hydroxy-3-(3-methyl-2-butenyl)phenyl)-2-propenoic acidIC5049000.0 [1]
Phenethyl cinnamateIC5018000.0 [1]
(3-Thioxo-2,3-Dihydro-5h-[1,2,4]triazino[5,6-B]indol-5-Yl)acetic AcidIC5021400.0 [1]
(E)-Benzyl 3-(4-hydroxyphenyl)acrylateIC50130.0 [1]
Isopropyl p-hydroxycinnamateIC50920.0 [1]
7-Hydroxy-N-[2-(4-hydroxyphenyl)ethyl]-2-oxochromene-3-carboxamideIC5020.0 [1]
4-Hydroxycinnamic acid phenethyl esterIC5069.0 [1]
2-Benzyl-9-(carboxymethyl)-1-sulfanylidene-3,4-dihydropyrido[3,4-b]indole-6-carboxylic acidIC5040000.0 [1]
N-[3-(4-Hydroxyphenyl)propyl]-2-oxochromene-3-carboxamideIC502700.0 [1]
3-Hydroxycinnamic acid phenethyl esterIC5019000.0 [1]
2-(2-(Ethoxycarbonyl)-8-methoxy-3,4-dihydro-1H-pyrido[4,3-b]indol-5(2H)-yl)acetic acidIC509434.0 [1]
{5-Chloro-2-[(Pentabromobenzyl)carbamoyl]phenoxy}acetic AcidIC5080.0 [1]
(3S,5R,6R,8S,9S,10R,13S,14S)-10-(Hydroxymethyl)-13-methyl-1,2,3,4,6,7,8,9,11,12,14,15,16,17-tetradecahydrocyclopenta[a]phenanthrene-3,5,6-triolIC50830.0 [1]
(2Z)-7-Hydroxy-2-(phenylimino)-N-(pyridin-2-yl)-2H-chromene-3-carboxamideIC5012.0 [1]
(2Z)-7-Hydroxy-2-[(4-methylphenyl)imino]-N-(pyridin-2-yl)-2H-chromene-3-carboxamideIC508.6 [1]
7-Hydroxy-2-(4-methoxyphenyl)imino-N-(2-methylpropyl)chromene-3-carboxamideIC5016.0 [1]
2-(4-Bromophenyl)imino-7-hydroxy-N-pyridin-2-ylchromene-3-carboxamideIC5014.0 [1]
7-Hydroxy-2-(4-hydroxyphenyl)imino-N-pyridin-2-ylchromene-3-carboxamideIC506.8 [1]
4-[[7-Hydroxy-3-(pyridin-2-ylcarbamoyl)chromen-2-ylidene]amino]benzoic acidIC507.6 [1]
7-Hydroxy-2-(4-iodophenyl)imino-N-pyridin-2-ylchromene-3-carboxamideIC5013.0 [1]
2-[4-[[7-Hydroxy-3-(pyridin-2-ylcarbamoyl)chromen-2-ylidene]amino]phenyl]acetic acidIC5013.0 [1]
7-Hydroxy-2-(4-methoxyphenyl)imino-N-propan-2-ylchromene-3-carboxamideIC509.7 [1]
N-Butyl-7-hydroxy-2-(4-methoxyphenyl)iminochromene-3-carboxamideIC5018.0 [1]
N-Cyclohexyl-7-hydroxy-2-(4-methoxyphenyl)iminochromene-3-carboxamideIC5011.0 [1]
7-Hydroxy-N-(2-hydroxyethyl)-2-(4-methoxyphenyl)iminochromene-3-carboxamideIC5011.0 [1]
7-Hydroxy-N-(3-hydroxypropyl)-2-(4-methoxyphenyl)iminochromene-3-carboxamideIC508.8 [1]
5-Hydroxy-2-(4-methoxyphenyl)imino-N-pyridin-2-ylchromene-3-carboxamideIC50290.0 [1]
2-[9-Fluoro-5-(4-methoxyphenyl)-3-methyl-1-oxopyrimido[4,5-c]quinolin-2-yl]acetic acidIC5010000.0 [1]
2-[5-(4-Chlorophenyl)-3-methyl-1-oxopyrimido[4,5-c]quinolin-2-yl]acetic acidIC507860.0 [1]
N-[3-(3,5-Difluorophenyl)propyl]-7-hydroxy-2-oxochromene-3-carboxamideIC507.8 [1]
N-[3-(3-Fluorophenyl)propyl]-7-hydroxy-2-oxochromene-3-carboxamideIC506.0 [1]
7-Hydroxy-N-[3-(4-methylphenyl)propyl]-2-oxochromene-3-carboxamideIC507.0 [1]
7-Hydroxy-N-[4-(4-hydroxyphenyl)butyl]-2-oxochromene-3-carboxamideIC5011.0 [1]
7-Hydroxy-N-[3-(3-hydroxyphenyl)propyl]-2-oxochromene-3-carboxamideIC508.3 [1]
7-Hydroxy-N-[3-(3-hydroxyphenyl)propyl]-2-(4-methoxyphenyl)iminochromene-3-carboxamideIC507.5 [1]
N-[3-(4-Fluorophenyl)propyl]-7-hydroxy-2-oxochromene-3-carboxamideIC503.5 [1]
8-Hydroxy-N-[3-(4-hydroxyphenyl)propyl]-2-oxochromene-3-carboxamideIC501500.0 [1]
7-Hydroxy-N-[3-(4-methoxyphenyl)propyl]-2-oxochromene-3-carboxamideIC5011.0 [1]
7-Hydroxy-N-[3-(2-hydroxyphenyl)propyl]-2-oxochromene-3-carboxamideIC506.4 [1]
2-[3-Benzyl-5-(4-chlorophenyl)-1-oxopyrimido[4,5-c]quinolin-2-yl]acetic acidIC502350.0 [1]
2-[5-(4-Bromophenyl)-9-fluoro-3-methyl-1-oxopyrimido[4,5-c]quinolin-2-yl]acetic acidIC509610.0 [1]
2-[5-(4-Chlorophenyl)-1-oxo-3-propylpyrimido[4,5-c]quinolin-2-yl]acetic acidIC503330.0 [1]
2-[9-Bromo-5-(4-bromophenyl)-3-methyl-1-oxopyrimido[4,5-c]quinolin-2-yl]acetic acidIC5016320.0 [1]
2-[5-(4-Chlorophenyl)-3-ethyl-9-fluoro-1-oxopyrimido[4,5-c]quinolin-2-yl]acetic acidIC503890.0 [1]
2-[5-(4-Bromophenyl)-3-methyl-1-oxopyrimido[4,5-c]quinolin-2-yl]acetic acidIC5010000.0 [1]
Items per page: 1 - 10 of 100
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References

This online tool may be cited as follows

MLA

"Quest Database™ Aldo-keto reductase family 1 member B10 Inhibitors (IC50, Ki)." AAT Bioquest, Inc., 20 Nov. 2024, https://www.aatbio.com/data-sets/aldo-keto-reductase-family-1-member-b10-inhibitors-ic50-ki.

APA

AAT Bioquest, Inc. (2024, November 20). Quest Database™ Aldo-keto reductase family 1 member B10 Inhibitors (IC50, Ki). AAT Bioquest. https://www.aatbio.com/data-sets/aldo-keto-reductase-family-1-member-b10-inhibitors-ic50-ki.
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