![](https://images.aatbio.com/dataset/ic50/adrenergic-receptor-beta_c70f5b79af37726016ec15cea0b55e94.svg) | Propranolol | IC50 | 4.0 [1], 12.0 [2] |
![](https://images.aatbio.com/dataset/ic50/adrenergic-receptor-beta_8b78ef0953132cb6729f40caa0d6bbea.svg) | Olanzapine | Ki | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/adrenergic-receptor-beta_9c9b6aadd4f8caa0bf86f9d7bbd70a7c.svg) | Sotalol | IC50 | 7200.0 [1] |
![](https://images.aatbio.com/dataset/ic50/adrenergic-receptor-beta_01a74ff12e6bf089ced324ef974b490e.svg) | Cisapride | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/adrenergic-receptor-beta_69119f40d0cfa359f19beacacddd1dc5.svg) | Sotalol hydrochloride | IC50 | 7200.0 [1] |
![](https://images.aatbio.com/dataset/ic50/adrenergic-receptor-beta_21a5e343431c845430d5c459f3e32ffb.svg) | Alprenolol | IC50 | 2.3 [1] |
![](https://images.aatbio.com/dataset/ic50/adrenergic-receptor-beta_10e671aa0c2e8af205d779ba113db7f0.svg) | Zafirlukast | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/adrenergic-receptor-beta_adfb749019985c1f8d769dcf4cc2178b.svg) | Sematilide | IC50 | 7000000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/adrenergic-receptor-beta_df20649e63f6814da658fbc9fd2ea41a.svg) | 4-Amino-5-chloro-N-((hexahydro-1H-pyrrolizin-1-yl)methyl)-2-methoxybenzamide hydrochloride | Ki | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/adrenergic-receptor-beta_25f5e25b0dad5fba18d7a0a972a7ad5f.svg) | Naluzotan | Ki | 2000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/adrenergic-receptor-beta_404ee23e4ae97a72a8990c4ff78f508e.svg) | N-Desmethylolanzapine | Ki | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/adrenergic-receptor-beta_5c33b6895b51be2fb2353c9a2cc7ab40.svg) | 4-(3-Tert-Butylamino-propoxy)-3-methyl-benzofuran-2-carboxylic acid ethyl ester | IC50 | 25000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/adrenergic-receptor-beta_1a25fd3b14cdd6366b9860277ee1d8db.svg) | 2-Hydroxymethyl Olanzapine | Ki | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/adrenergic-receptor-beta_d59ce514cb743faa8901da9019b43d12.svg) | Ethyl 4-[2-hydroxy-3-(isopropylamino)propoxy]-3-methyl-1-benzofuran-2-carboxylate | IC50 | 98.0 [1] |
![](https://images.aatbio.com/dataset/ic50/adrenergic-receptor-beta_902d9f8450dbf5e6c0fdbf3e2ba493f7.svg) | Ethyl 3-methyl-4-{3-[(methylethyl)amino]propoxy}benzo[d]furan-2-carboxylate | IC50 | 38000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/adrenergic-receptor-beta_ff207c208d28dd5a66e80b5c36e10c36.svg) | Ethyl 4-{3-[(tert-butyl)amino]-2-hydroxypropoxy}-3-methylbenzo[d]furan-2-carboxylate | IC50 | 4.3 [1] |
![](https://images.aatbio.com/dataset/ic50/adrenergic-receptor-beta_760c3502a4edf61c27018ca53a36c234.svg) | 4-Amino-N-[(4R)-1-azatricyclo[3.3.1.03,7]nonan-4-yl]-5-chloro-2-methoxybenzamide | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/adrenergic-receptor-beta_c19d0ac38f1af2179d31460833b8a096.svg) | N-[2-[(2-Hydroxy-3-naphthalen-1-yloxypropyl)amino]ethyl]-4-(methanesulfonamido)benzamide | IC50 | 150.0 [1] |
![](https://images.aatbio.com/dataset/ic50/adrenergic-receptor-beta_d7ff1eaae84953a42a1129e772fc8ae0.svg) | N-[2-[[2-Hydroxy-3-(4-methoxyphenoxy)propyl]amino]ethyl]-4-(methanesulfonamido)benzamide | IC50 | 43800.0 [1] |
![](https://images.aatbio.com/dataset/ic50/adrenergic-receptor-beta_b8af37a6027640c9500c3ee5d293b315.svg) | N-[2-[(2-Hydroxy-3-phenoxypropyl)amino]ethyl]-4-(methanesulfonamido)benzamide | IC50 | 3900.0 [1] |
![](https://images.aatbio.com/dataset/ic50/adrenergic-receptor-beta_8b85bdb4e802c91b072fb0cc962b8b1a.svg) | N-[2-[[3-(2-Cyanophenoxy)-2-hydroxypropyl]amino]ethyl]-4-(methanesulfonamido)benzamide | IC50 | 2900.0 [1] |
![](https://images.aatbio.com/dataset/ic50/adrenergic-receptor-beta_28e4199d4801885941c047dc3755fcae.svg) | N-[2-[(2-Hydroxy-3-phenoxypropyl)amino]cyclohexyl]-4-(methanesulfonamido)benzamide | IC50 | 192000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/adrenergic-receptor-beta_495543d0c5c6a45d04d023db3f1941d6.svg) | N-[2-[[2-Hydroxy-3-[4-(2-methoxyethyl)phenoxy]propyl]amino]ethyl]-4-imidazol-1-ylbenzamide | IC50 | 12400.0 [1] |
![](https://images.aatbio.com/dataset/ic50/adrenergic-receptor-beta_a57ac07fce9fa5282ba33d64faf5138b.svg) | N-[2-[[2-Hydroxy-3-(4-methoxyphenoxy)propyl]amino]ethyl]-4-imidazol-1-ylbenzamide | IC50 | 61400.0 [1] |
![](https://images.aatbio.com/dataset/ic50/adrenergic-receptor-beta_04aaa3d39abe8ea85fa23273d67e5207.svg) | N-[2-[(2-Hydroxy-3-naphthalen-1-yloxypropyl)amino]ethyl]-4-imidazol-1-ylbenzamide | IC50 | 420.0 [1] |
![](https://images.aatbio.com/dataset/ic50/adrenergic-receptor-beta_0cf56e473c5f4ec33ca22f66c9256dfd.svg) | N-[2-[[2-Hydroxy-3-[4-(methanesulfonamido)phenoxy]propyl]amino]ethyl]-4-imidazol-1-ylbenzamide | IC50 | 227000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/adrenergic-receptor-beta_7b13fbeefe8a3a21c1d02dcc597a03f7.svg) | 1-[2-Hydroxy-3-(1-naphthalenyloxy)propyl]-4-[4-[(methylsulfonyl)amino]benzoyl]piperazine | IC50 | 30900.0 [1] |
![](https://images.aatbio.com/dataset/ic50/adrenergic-receptor-beta_f8ad60a31b7fe0f5b0d97bb419f82f23.svg) | 1-[4-(Methylsulfonylamino)benzoyl]-4-[2-hydroxy-3-phenoxypropyl]piperazine | IC50 | 12200.0 [1] |
![](https://images.aatbio.com/dataset/ic50/adrenergic-receptor-beta_db4f0286d94e07c6b8664c404e759c86.svg) | 1-[4-(Methylsulfonylamino)benzoyl]-4-[2-hydroxy-3-[4-(2-methoxyethyl)phenoxy]propyl]piperazine | IC50 | 360000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/adrenergic-receptor-beta_fe478243de8eb2aa32bfc6b6d379e046.svg) | 1-[4-(Methylsulfonylamino)benzylamino]-3-(3-methylphenoxy)-2-propanol | IC50 | 990.0 [1] |
![](https://images.aatbio.com/dataset/ic50/adrenergic-receptor-beta_73ab41177a8fc26426829b85c554d1bd.svg) | 1-[4-(Methylsulfonylamino)benzylamino]-3-phenoxy-2-propanol | IC50 | 2900.0 [1] |
![](https://images.aatbio.com/dataset/ic50/adrenergic-receptor-beta_ce234fb1cfe7c623f4441dc73c2a3da1.svg) | 1-[4-(Methylsulfonylamino)benzylamino]-3-[4-(2-methoxyethyl)phenoxy]-2-propanol | IC50 | 25800.0 [1] |
![](https://images.aatbio.com/dataset/ic50/adrenergic-receptor-beta_81a4773cd3eef7e737a403d3a88aaf57.svg) | 1-(4-Imidazol-1-yl-benzylamino)-3-o-tolyloxy-propan-2-ol | IC50 | 780.0 [1] |
![](https://images.aatbio.com/dataset/ic50/adrenergic-receptor-beta_27eb37ae53f40b0756b1171f31b1da9c.svg) | 1-[4-[4-(Methylsulfonylamino)phenyl]-1-piperazinyl]-3-phenoxy-2-propanol | IC50 | 15800.0 [1] |
![](https://images.aatbio.com/dataset/ic50/adrenergic-receptor-beta_d5c50c5fad317db0f349441abe507d90.svg) | 1-[4-[4-(Methylsulfonylamino)phenyl]-1-piperazinyl]-3-(3-methylphenoxy)-2-propanol | IC50 | 15700.0 [1] |
![](https://images.aatbio.com/dataset/ic50/adrenergic-receptor-beta_415e7befba24ceeef17ddb0c4e4f25c7.svg) | 1-[4-[4-(Methylsulfonylamino)phenyl]-1-piperazinyl]-3-[4-(2-methoxyethyl)phenoxy]-2-propanol | IC50 | 109000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/adrenergic-receptor-beta_587469c8cd5f3aa10eb9de514ac3cb13.svg) | N-[4-[2-Hydroxy-3-[4-[4-(methanesulfonamido)phenyl]piperazin-1-yl]propoxy]phenyl]acetamide | IC50 | 293000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/adrenergic-receptor-beta_aa3a82dab627802582385dd2395f0c0e.svg) | N-[4-[4-[2-Hydroxy-3-[(5-oxo-7,8-dihydro-6H-naphthalen-1-yl)oxy]propyl]piperazin-1-yl]phenyl]methanesulfonamide | IC50 | 8400.0 [1] |
![](https://images.aatbio.com/dataset/ic50/adrenergic-receptor-beta_8f5ca8410bd13ec754c957a49e34e425.svg) | 1-[4-[4-(Methylsulfonylamino)phenyl]-1-piperazinyl]-3-(2-methylphenoxy)-2-propanol | IC50 | 2300.0 [1] |
![](https://images.aatbio.com/dataset/ic50/adrenergic-receptor-beta_0e1a0b77c2cbf4145dc606d931f032e7.svg) | 1-[[2-[4-(1H-Imidazol-1-yl)phenoxy]ethyl]amino]-3-phenoxy-2-propanol | IC50 | 40.0 [1] |
![](https://images.aatbio.com/dataset/ic50/adrenergic-receptor-beta_cadfe1cae1ebe935c223f24c9688a9d7.svg) | 1-[[2-[4-(1H-Imidazol-1-yl)phenoxy]ethyl]amino]-3-[4-(2-methoxyethyl)phenoxy]-2-propanol | IC50 | 270.0 [1] |
![](https://images.aatbio.com/dataset/ic50/adrenergic-receptor-beta_573f88e8a0226ed7536b66c9c4ca9d12.svg) | 1-{2-[4-(3H-Imidazol-1-yl)-phenoxy]-ethylamino}-3-m-tolyloxy-propan-2-ol | IC50 | 90.0 [1] |
![](https://images.aatbio.com/dataset/ic50/adrenergic-receptor-beta_ff06f854c92ba7d91f5613fc9ead478f.svg) | 2-[2-[4-(1H-Imidazol-1-yl)phenoxy]ethylamino]-1-[4-(methylsulfonylamino)phenyl]ethanol | IC50 | 3600.0 [1] |
![](https://images.aatbio.com/dataset/ic50/adrenergic-receptor-beta_5e3f4908203eccfafbd7f63490b53721.svg) | alpha-[[[2-[4-(1H-Imidazol-1-yl)phenoxy]ethyl]amino]methyl]-2-methoxybenzenemethanol | IC50 | 3700.0 [1] |
![](https://images.aatbio.com/dataset/ic50/adrenergic-receptor-beta_48b356b985bd7092f7cca34a9917e214.svg) | 4-Amino-N-(1-azatricyclo[3.3.1.13,7]decan-4-yl)-5-chloro-2-methoxybenzamide | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/adrenergic-receptor-beta_661698f214ede3677cafa0ebc11ae5fd.svg) | N-[4-[4-[3-(Dicyclopropylmethylamino)oxy-2-hydroxypropyl]piperazin-1-yl]phenyl]methanesulfonamide | IC50 | 15700.0 [1] |
![](https://images.aatbio.com/dataset/ic50/adrenergic-receptor-beta_1493fdc64b9f16499e0004a679f2f158.svg) | 1-(Dicyclopropylmethylamino)oxy-3-[2-(4-imidazol-1-ylphenoxy)ethylamino]propan-2-ol | IC50 | 300.0 [1] |
![](https://images.aatbio.com/dataset/ic50/adrenergic-receptor-beta_f129a59986c2b776c652f279787c4183.svg) | (5R)-3-(3-Methyl-1-benzofuran-5-yl)spiro[1,3-oxazolidine-5,3'-1-azabicyclo[2.2.2]octane]-2-one | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/adrenergic-receptor-beta_d25e94149787af9b3b05d1433400ec2f.svg) | 1-[2-Hydroxy-2-[4-[(methylsulfonyl)amino]phenyl]ethyl]-3-methyl-1H-imidazol-3-ium | IC50 | 2350000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/adrenergic-receptor-beta_24dfe81a08817ea380bb78bf673314d7.svg) | 4-Amino-N-(1-azatricyclo[3.3.1.03,7]nonan-4-yl)-5-chloro-2-methoxybenzamide | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/adrenergic-receptor-beta_af626ce502ae0aa7d74cd7782941cd61.svg) | 4-Amino-N-(1-azatricyclo[3.3.1.13,7]decan-4-ylmethyl)-5-chloro-2-methoxybenzamide | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/adrenergic-receptor-beta_d0633676d54791ae6c2121b4a37658ab.svg) | Olanzapine N-Oxide | Ki | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/adrenergic-receptor-beta_0cd593c4d8e68bd2fedfa9cbe7af8fcd.svg) | 5-Fluoro-2-[(E)-2-[3-[[4-(2-methylimidazo[4,5-c]pyridin-1-yl)phenoxy]methyl]phenyl]ethenyl]-1,3-benzothiazole | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/adrenergic-receptor-beta_5a1d59942f914b250645c69607ffb388.svg) | 7-Chloro-2-[(E)-2-[3-[[4-(2-methylimidazo[4,5-c]pyridin-1-yl)phenoxy]methyl]phenyl]ethenyl]quinoline | IC50 | 10000.0 [1] |