| Propranolol | IC50 | 4.0 [1], 12.0 [2] |
| Olanzapine | Ki | 10000.0 [1] |
| Sotalol | IC50 | 7200.0 [1] |
| Cisapride | IC50 | 10000.0 [1] |
| Sotalol hydrochloride | IC50 | 7200.0 [1] |
| Alprenolol | IC50 | 2.3 [1] |
| Zafirlukast | IC50 | 10000.0 [1] |
| Sematilide | IC50 | 7000000.0 [1] |
| 4-Amino-5-chloro-N-((hexahydro-1H-pyrrolizin-1-yl)methyl)-2-methoxybenzamide hydrochloride | Ki | 10000.0 [1] |
| Naluzotan | Ki | 2000.0 [1] |
| N-Desmethylolanzapine | Ki | 10000.0 [1] |
| 4-(3-Tert-Butylamino-propoxy)-3-methyl-benzofuran-2-carboxylic acid ethyl ester | IC50 | 25000.0 [1] |
| 2-Hydroxymethyl Olanzapine | Ki | 10000.0 [1] |
| Ethyl 4-[2-hydroxy-3-(isopropylamino)propoxy]-3-methyl-1-benzofuran-2-carboxylate | IC50 | 98.0 [1] |
| Ethyl 3-methyl-4-{3-[(methylethyl)amino]propoxy}benzo[d]furan-2-carboxylate | IC50 | 38000.0 [1] |
| Ethyl 4-{3-[(tert-butyl)amino]-2-hydroxypropoxy}-3-methylbenzo[d]furan-2-carboxylate | IC50 | 4.3 [1] |
| 4-Amino-N-[(4R)-1-azatricyclo[3.3.1.03,7]nonan-4-yl]-5-chloro-2-methoxybenzamide | IC50 | 10000.0 [1] |
| N-[2-[(2-Hydroxy-3-naphthalen-1-yloxypropyl)amino]ethyl]-4-(methanesulfonamido)benzamide | IC50 | 150.0 [1] |
| N-[2-[[2-Hydroxy-3-(4-methoxyphenoxy)propyl]amino]ethyl]-4-(methanesulfonamido)benzamide | IC50 | 43800.0 [1] |
| N-[2-[(2-Hydroxy-3-phenoxypropyl)amino]ethyl]-4-(methanesulfonamido)benzamide | IC50 | 3900.0 [1] |
| N-[2-[[3-(2-Cyanophenoxy)-2-hydroxypropyl]amino]ethyl]-4-(methanesulfonamido)benzamide | IC50 | 2900.0 [1] |
| N-[2-[(2-Hydroxy-3-phenoxypropyl)amino]cyclohexyl]-4-(methanesulfonamido)benzamide | IC50 | 192000.0 [1] |
| N-[2-[[2-Hydroxy-3-[4-(2-methoxyethyl)phenoxy]propyl]amino]ethyl]-4-imidazol-1-ylbenzamide | IC50 | 12400.0 [1] |
| N-[2-[[2-Hydroxy-3-(4-methoxyphenoxy)propyl]amino]ethyl]-4-imidazol-1-ylbenzamide | IC50 | 61400.0 [1] |
| N-[2-[(2-Hydroxy-3-naphthalen-1-yloxypropyl)amino]ethyl]-4-imidazol-1-ylbenzamide | IC50 | 420.0 [1] |
| N-[2-[[2-Hydroxy-3-[4-(methanesulfonamido)phenoxy]propyl]amino]ethyl]-4-imidazol-1-ylbenzamide | IC50 | 227000.0 [1] |
| 1-[2-Hydroxy-3-(1-naphthalenyloxy)propyl]-4-[4-[(methylsulfonyl)amino]benzoyl]piperazine | IC50 | 30900.0 [1] |
| 1-[4-(Methylsulfonylamino)benzoyl]-4-[2-hydroxy-3-phenoxypropyl]piperazine | IC50 | 12200.0 [1] |
| 1-[4-(Methylsulfonylamino)benzoyl]-4-[2-hydroxy-3-[4-(2-methoxyethyl)phenoxy]propyl]piperazine | IC50 | 360000.0 [1] |
| 1-[4-(Methylsulfonylamino)benzylamino]-3-(3-methylphenoxy)-2-propanol | IC50 | 990.0 [1] |
| 1-[4-(Methylsulfonylamino)benzylamino]-3-phenoxy-2-propanol | IC50 | 2900.0 [1] |
| 1-[4-(Methylsulfonylamino)benzylamino]-3-[4-(2-methoxyethyl)phenoxy]-2-propanol | IC50 | 25800.0 [1] |
| 1-(4-Imidazol-1-yl-benzylamino)-3-o-tolyloxy-propan-2-ol | IC50 | 780.0 [1] |
| 1-[4-[4-(Methylsulfonylamino)phenyl]-1-piperazinyl]-3-phenoxy-2-propanol | IC50 | 15800.0 [1] |
| 1-[4-[4-(Methylsulfonylamino)phenyl]-1-piperazinyl]-3-(3-methylphenoxy)-2-propanol | IC50 | 15700.0 [1] |
| 1-[4-[4-(Methylsulfonylamino)phenyl]-1-piperazinyl]-3-[4-(2-methoxyethyl)phenoxy]-2-propanol | IC50 | 109000.0 [1] |
| N-[4-[2-Hydroxy-3-[4-[4-(methanesulfonamido)phenyl]piperazin-1-yl]propoxy]phenyl]acetamide | IC50 | 293000.0 [1] |
| N-[4-[4-[2-Hydroxy-3-[(5-oxo-7,8-dihydro-6H-naphthalen-1-yl)oxy]propyl]piperazin-1-yl]phenyl]methanesulfonamide | IC50 | 8400.0 [1] |
| 1-[4-[4-(Methylsulfonylamino)phenyl]-1-piperazinyl]-3-(2-methylphenoxy)-2-propanol | IC50 | 2300.0 [1] |
| 1-[[2-[4-(1H-Imidazol-1-yl)phenoxy]ethyl]amino]-3-phenoxy-2-propanol | IC50 | 40.0 [1] |
| 1-[[2-[4-(1H-Imidazol-1-yl)phenoxy]ethyl]amino]-3-[4-(2-methoxyethyl)phenoxy]-2-propanol | IC50 | 270.0 [1] |
| 1-{2-[4-(3H-Imidazol-1-yl)-phenoxy]-ethylamino}-3-m-tolyloxy-propan-2-ol | IC50 | 90.0 [1] |
| 2-[2-[4-(1H-Imidazol-1-yl)phenoxy]ethylamino]-1-[4-(methylsulfonylamino)phenyl]ethanol | IC50 | 3600.0 [1] |
| alpha-[[[2-[4-(1H-Imidazol-1-yl)phenoxy]ethyl]amino]methyl]-2-methoxybenzenemethanol | IC50 | 3700.0 [1] |
| 4-Amino-N-(1-azatricyclo[3.3.1.13,7]decan-4-yl)-5-chloro-2-methoxybenzamide | IC50 | 10000.0 [1] |
| N-[4-[4-[3-(Dicyclopropylmethylamino)oxy-2-hydroxypropyl]piperazin-1-yl]phenyl]methanesulfonamide | IC50 | 15700.0 [1] |
| 1-(Dicyclopropylmethylamino)oxy-3-[2-(4-imidazol-1-ylphenoxy)ethylamino]propan-2-ol | IC50 | 300.0 [1] |
| (5R)-3-(3-Methyl-1-benzofuran-5-yl)spiro[1,3-oxazolidine-5,3'-1-azabicyclo[2.2.2]octane]-2-one | IC50 | 10000.0 [1] |
| 1-[2-Hydroxy-2-[4-[(methylsulfonyl)amino]phenyl]ethyl]-3-methyl-1H-imidazol-3-ium | IC50 | 2350000.0 [1] |
| 4-Amino-N-(1-azatricyclo[3.3.1.03,7]nonan-4-yl)-5-chloro-2-methoxybenzamide | IC50 | 10000.0 [1] |
| 4-Amino-N-(1-azatricyclo[3.3.1.13,7]decan-4-ylmethyl)-5-chloro-2-methoxybenzamide | IC50 | 10000.0 [1] |
| Olanzapine N-Oxide | Ki | 10000.0 [1] |
| 5-Fluoro-2-[(E)-2-[3-[[4-(2-methylimidazo[4,5-c]pyridin-1-yl)phenoxy]methyl]phenyl]ethenyl]-1,3-benzothiazole | IC50 | 10000.0 [1] |
| 7-Chloro-2-[(E)-2-[3-[[4-(2-methylimidazo[4,5-c]pyridin-1-yl)phenoxy]methyl]phenyl]ethenyl]quinoline | IC50 | 10000.0 [1] |