 | Clozapine | Ki | 3.7 [1], 11.0 [2], 23.0 [3], 47.86 [4] |
 | Olanzapine | Ki | 7.3 [1], 14.0 [2], 15.0 [3], 60.0 [4] |
 | Ziprasidone | IC50 | 11.0 [1] |
| Ziprasidone | Ki | 1.9 [1], 11.0 [2], 12.0 [3] |
 | N-(4,5-Dihydro-1H-imidazol-2-yl)-5-methylquinoxalin-6-amine | Ki | 1400.0 [1] |
 | Risperidone | Ki | 0.69 [1], 1.0 [2], 2.3 [3] |
 | Prazosin | IC50 | 0.17 [1], 0.2 [2], 0.86 [3] |
 | Brimonidine | Ki | 1800.0 [1], 1900.0 [2] |
 | 2-Naphthalenecarboxamide, N-(4-(4-(2-methoxyphenyl)-1-piperazinyl)butyl)- | Ki | 5.0 [1], 25.0 [2] |
 | N-[4-[4-(2,3-Dichlorophenyl)piperazin-1-yl]butyl]-1-benzothiophene-2-carboxamide | Ki | 370.0 [1], 2000.0 [2] |
 | N-(4,5-Dihydro-1H-imidazol-2-yl)-5-methyl-1,2,3,4-tetrahydroquinoxalin-6-amine | Ki | 8700.0 [1], 8900.0 [2] |
 | Clonidine | Ki | 510.0 [1] |
 | Haloperidol | Ki | 5.7 [1], 19.0 [2] |
 | Quetiapine | Ki | 4.5 [1], 58.0 [2] |
 | Cisapride | IC50 | 30.0 [1] |
 | 4-Amino-5-chloro-N-((hexahydro-1H-pyrrolizin-1-yl)methyl)-2-methoxybenzamide hydrochloride | IC50 | 10000.0 [1] |
| 4-Amino-5-chloro-N-((hexahydro-1H-pyrrolizin-1-yl)methyl)-2-methoxybenzamide hydrochloride | Ki | 10000.0 [1] |
 | (2R)-1-[4-(4-Methylbenzyl)piperazinoacetyl]-2-methylindoline | IC50 | 1118.0 [1] |
| (2R)-1-[4-(4-Methylbenzyl)piperazinoacetyl]-2-methylindoline | Ki | 1118.0 [1] |
 | 4-Amino-N-[(4R)-1-azatricyclo[3.3.1.03,7]nonan-4-yl]-5-chloro-2-methoxybenzamide | IC50 | 10000.0 [1] |
 | 7-Nitro-3-{[2-(phenyloxy)phenyl]amino}-4H-1,2,4-benzothiadiazin-5-ol 1,1-dioxide | IC50 | 1000.0 [1], 25000.0 [2] |
 | N-(4,5-Dihydro-1H-imidazol-2-yl)-5-methyl-3,4-dihydro-2H-1,4-benzoxazin-6-amine | Ki | 470.0 [1] |
 | (7-Chloro-2,3-dihydro-benzo[1,4]dioxin-2-ylmethyl)-[1-(2-methoxy-phenyl)-piperidin-4-ylmethyl]-amine | Ki | 53.0 [1], 181.0 [2] |
 | N-(4,5-Dihydro-1H-imidazol-2-yl)quinoxalin-6-amine | Ki | 11000.0 [1] |
 | Dopamine | Ki | 2511.89 [1] |
 | Norepinephrine | Ki | 2600.0 [1] |
 | Atenolol | IC50 | 230.0 [1] |
 | Terfenadine | IC50 | 2340.0 [1] |
 | Fenoldopam | Ki | 151.36 [1] |
 | Zafirlukast | IC50 | 10000.0 [1] |
 | Moxonidine | Ki | 30000.0 [1] |
 | Apraclonidine | Ki | 180.0 [1] |
 | Sertindole | Ki | 1.8 [1] |
 | Ipsapirone | IC50 | 500.0 [1] |
 | Ebastine | IC50 | 183.0 [1] |
 | Pizotifen | Ki | 75.0 [1] |
 | Zotepine | Ki | 3.4 [1] |
 | GR-127935 | Ki | 1000.0 [1] |
 | Sarpogrelate hydrochloride | IC50 | 1000.0 [1] |
 | 4-[(1R,2S)-3-(4-Benzylpiperidin-1-yl)-1-hydroxy-2-methylpropyl]phenol | Ki | 180.0 [1] |
 | Vilazodone | IC50 | 1980.0 [1] |
 | 4-[2-(Dipropylamino)ethyl]benzene-1,2-diol | Ki | 1995.26 [1] |
 | 7-Methyl-6,7,8,9,14,15-hexahydro-5H-benz[d]indolo[2,3-g]azecine | Ki | 11.0 [1] |
 | 3-[[4-(4-Chlorophenyl)piperazin-1-yl]methyl]pyrazolo[1,5-a]pyridine | Ki | 240.0 [1] |
 | N-Desmethylolanzapine | Ki | 80.0 [1] |
 | N-[4-[4-(2-Methoxyphenyl)piperazin-1-yl]butyl]pyrazolo[1,5-a]pyridine-2-carboxamide | Ki | 26.0 [1] |
 | 1-[4-(4-Chlorobenzyl)piperazinoacetyl]indoline | IC50 | 88.0 [1] |
 | N-(4-(4-(2-Methoxyphenyl)piperazin-1-yl)butyl)benzo[b]thiophene-2-carboxamide | Ki | 15.0 [1] |
 | N-(4-(4-(2-Methoxyphenyl)piperazin-1-yl)butyl)benzofuran-2-carboxamide | Ki | 8.6 [1] |
 | Unii-N4Y2V13I7F | Ki | 6.75 [1] |
 | 1-[2-(3,4-Dihydro-1H-2-benzopyran-1-yl)ethyl]-4-(4-fluorophenyl)piperazine | Ki | 38.0 [1] |
 | N-(4-(4-(2,3-Dichlorophenyl)piperazin-1-yl)butyl)benzofuran-2-carboxamide | Ki | 10000.0 [1] |
 | Eptapirone | Ki | 10000.0 [1] |
 | Mazapertine | Ki | 1.3 [1] |
 | 2-(1-Benzofuran-6-yl)-N-[[(1R)-5-methoxy-1,2,3,4-tetrahydronaphthalen-1-yl]methyl]-N-methylethanamine | Ki | 1000.0 [1] |
 | 3-Isopropyl-bicyclo[2.2.1]hept-2-ylamine | Ki | 100000.0 [1] |
 | 3-[2-(Benzylamino)ethoxy]phenol | Ki | 5291.0 [1] |
 | N-((Hexahydro-1H-pyrrolizin-1-yl)methyl)-6-chloroimidazo(1,2-a)pyridine-8-carboxamide hydrochloride | IC50 | 10000.0 [1] |
 | 2-(1,4-Benzodioxan-6-ylamino)-2-imidazoline | Ki | 2400.0 [1] |
 | 1-(2,3-Dihydro-1,4-benzodioxin-6-yl)-4-(2,3-dihydro-1H-inden-2-ylmethyl)piperazine | Ki | 967.0 [1] |
 | 3-(4-Benzyl-piperazin-1-yl)-phenol | Ki | 1000.0 [1] |
 | 4-(5-Fluoro-2-indanylmethyl)-2-imidazoline | Ki | 1000.0 [1] |
 | 2-Hydroxymethyl Olanzapine | Ki | 12.0 [1] |
 | Imidazolidine, 2-(2-methylphenylimino)- | Ki | 2500.0 [1] |
 | (3R,3As)-7,8-dimethoxy-3-[[4-[(E)-3-phenylprop-2-enyl]piperazin-1-yl]methyl]-3a,4-dihydro-3H-chromeno[4,3-c][1,2]oxazole | Ki | 1000.0 [1] |
 | (3R,3As)-7,8-dimethoxy-3-[[4-[(E)-2-methyl-3-phenylprop-2-enyl]piperazin-1-yl]methyl]-3a,4-dihydro-3H-chromeno[4,3-c][1,2]oxazole | Ki | 380.0 [1] |
 | (3R,3As)-7,8-dimethoxy-3-[[4-[(E)-3-phenylbut-2-enyl]piperazin-1-yl]methyl]-3a,4-dihydro-3H-chromeno[4,3-c][1,2]oxazole | Ki | 1000.0 [1] |
 | N-[4-[4-(2-Methoxyphenyl)piperazin-1-yl]butyl]pyrazolo[1,5-a]pyridine-4-carboxamide | Ki | 28.0 [1] |
 | N-[4-[4-(2-Methoxyphenyl)piperazin-1-yl]butyl]pyrazolo[1,5-a]pyridine-7-carboxamide | Ki | 18.0 [1] |
 | N-[4-[4-(2-Methoxyphenyl)piperazin-1-yl]butyl]pyrazolo[1,5-a]pyridine-5-carboxamide | Ki | 32.0 [1] |
 | 2-{[4-(2-Methoxyphenyl)piperazino]methyl}imidazo[1,2-a]pyridine | Ki | 98.0 [1] |
 | 1-[2-[4-(6-Fluoro-1H-indol-3-yl)-3,6-dihydro-2H-pyridin-1-yl]ethyl]-3,4-dihydro-1H-isochromene-6-carboxamide | Ki | 16.0 [1] |
 | 5-[2-[4-(2,3-Dimethylphenyl)piperazin-1-yl]ethyl]-2H-benzotriazole | Ki | 67.61 [1] |
 | N-[4-[4-(2,3-Dichlorophenyl)piperazin-1-yl]butyl]-5-iodo-1-benzofuran-2-carboxamide | Ki | 300.0 [1] |
 | 2-N-[2-(4-Fluorophenoxy)ethyl]-4-N-[(1S)-1-phenylethyl]pyridine-2,4-diamine | Ki | 8.0 [1] |
 | N-[4-[4-(2-Methoxyphenyl)piperazin-1-yl]butyl]pyrazolo[1,5-a]pyridine-6-carboxamide | Ki | 19.0 [1] |
 | N-[4-[4-(2-Methoxyphenyl)piperazin-1-yl]butyl]pyrazolo[1,5-a]pyridine-3-carboxamide | Ki | 48.0 [1] |
 | 1-[1-(6-Chloro-1,3-benzodioxole-5-ylmethyl)-4-piperidinyl]-1H-benzimidazole-2(3H)-one | IC50 | 1330.0 [1] |
 | 3-[1-[(6-Chloro-1,3-benzodioxol-5-yl)methyl]piperidin-4-yl]-5-methyl-1H-benzimidazol-2-one | IC50 | 4920.0 [1] |
 | 8-(2,1,3-Benzothiadiazol-5-ylmethyl)-1-phenyl-1,3,8-triazaspiro[4.5]decan-4-one | IC50 | 4250.0 [1] |
 | 1-[3-(6-Chloro-1,3-benzodioxole-5-ylmethylamino)propyl]-1H-benzimidazole-2(3H)-one | IC50 | 174.0 [1] |
 | (6-Chloro-1,3-benzodioxol-5-yl)methyl 4-(2-oxo-3H-benzimidazol-1-yl)piperidine-1-carboxylate | IC50 | 1340.0 [1] |
 | 5-(2-(4-(1-Naphthyl)piperazinyl)ethyl)oxindole | IC50 | 45.0 [1] |
 | N-[4-[4-(2-Methoxyphenyl)piperazin-1-yl]butyl]tricyclo[8.2.2.24,7]hexadeca-1(13),4,6,10(14),11,15-hexaene-5-carboxamide | Ki | 3.9 [1] |
 | 2-[4-[4-(7-Hydroxynaphthalen-1-yl)piperazin-1-yl]butyl]-4-methyl-1,2,4-triazine-3,5-dione | Ki | 24.5 [1] |
 | 2-[4-[4-(7-(111C)Methoxynaphthalen-1-yl)piperazin-1-yl]butyl]-4-methyl-1,2,4-triazine-3,5-dione | Ki | 32.2 [1] |
 | 6-(4-Chlorophenyl)-3-[2-[4-(2-chlorophenyl)piperazin-1-yl]ethyl]-1,7-dihydropyrrolo[2,3-d]pyrimidine-2,4-dione | Ki | 2.64 [1] |
 | 3-[2-[4-(2-Chlorophenyl)piperazin-1-yl]ethyl]-6-(4-methylphenyl)-1,5-dihydropyrrolo[3,2-d]pyrimidine-2,4-dione | Ki | 17.26 [1] |
 | 8-(3-Phenoxybenzyl)-1-phenyl-1,3,8-triazaspiro[4.5]decane-4-one | IC50 | 2830.0 [1] |
 | N-(Diaminomethylidene)-9-hydroxy-9-methylfluorene-2-carboxamide;hydrochloride | Ki | 1000.0 [1] |
 | 1-[(Dimethylamino)methyl]-2,3-dihydro-1H-indene-4,5-diol | Ki | 6900.0 [1] |
 | 1H-Indene-4,5-diol, 2,3-dihydro-1-[(methylamino)methyl]- | Ki | 2000.0 [1] |
 | 1H-Indene-4,5-diol, 1-(aminomethyl)-2,3-dihydro- | Ki | 2250.0 [1] |
 | 1-[(Dipropylamino)methyl]-2,3-dihydro-1H-indene-4,5-diol | Ki | 7400.0 [1] |
 | 1H-Indene-5,6-diol, 1-(aminomethyl)-2,3-dihydro- | Ki | 26000.0 [1] |
 | 4-[2-Hydroxy-3-[4-hydroxy-4-(4-methylbenzyl)piperidino]propyl]phenol | Ki | 5915.0 [1] |
 | 2-[10-[3-[4-(1,3-Dimethyl-2,6-dioxopyrimidin-4-yl)piperazin-1-yl]propyl]phenothiazin-2-yl]acetic acid | IC50 | 430.0 [1] |
 | 2-[4-(4-Chloro-benzyl)-piperazin-1-yl]-N-methyl-N-phenyl-acetamide | Ki | 10000.0 [1] |
 | (3R,3As)-7,8-dimethoxy-3-[[4-(naphthalen-2-ylmethyl)piperazin-1-yl]methyl]-3a,4-dihydro-3H-chromeno[4,3-c][1,2]oxazole | Ki | 1000.0 [1] |
 | 5-Iodo-N-[4-[4-(2-methoxyphenyl)piperazin-1-yl]butyl]-1-benzofuran-2-carboxamide | Ki | 5.9 [1] |
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