 | 3-[[4-[3-[4-(1-Benzofuran-2-yl)anilino]-2-(4-tert-butylphenyl)-3-oxopropyl]benzoyl]amino]propanoic acid | Ki | 29.0 [1], 69.0 [2] |
 | Gra EX-25 | Ki | 254.0 [1] |
 | (2S)-N-[(2S)-1-Amino-5-(diaminomethylideneamino)-1-oxopentan-2-yl]-1-[(4R,7S,10S,13S,16R)-7-(2-amino-2-oxoethyl)-13-benzyl-20,20-dicyclopentyl-16-[(4-ethoxyphenyl)methyl]-6,9,12,15,18-pentaoxo-10-propan-2-yl-1,2-dithia-5,8,11,14,17-pentazacycloicosane-4-carbonyl]pyrrolidine-2-carboxamide | Ki | 3.9 [1] |
 | (10R,13S,16S,19S)-N-[(2S)-1-Amino-5-(diaminomethylideneamino)-1-oxopentan-2-yl]-19-(2-amino-2-oxoethyl)-13-benzyl-10-[(4-ethoxyphenyl)methyl]-8,11,14,17,20-pentaoxo-16-propan-2-yl-9,12,15,18,21-pentazaspiro[5.19]pentacosane-22-carboxamide | Ki | 4400000.0 [1] |
 | 3-[[4-[2-(4-Tert-butylphenyl)-3-oxo-3-[4-(trifluoromethoxy)anilino]propyl]benzoyl]amino]propanoic acid | Ki | 110.0 [1] |
 | 3-[[4-[2-(4-Tert-butylphenyl)-3-oxo-3-(4-phenylanilino)propyl]benzoyl]amino]propanoic acid | Ki | 300.0 [1] |
 | 3-[[4-[2-(4-Tert-butylphenyl)-3-(3-ethylanilino)-3-oxopropyl]benzoyl]amino]propanoic acid | Ki | 2000.0 [1] |
 | 3-[[4-[2-(4-Tert-butylphenyl)-3-(4-ethylanilino)-3-oxopropyl]benzoyl]amino]propanoic acid | Ki | 2000.0 [1] |
 | 3-[[4-[2-(4-Tert-butylphenyl)-3-oxo-3-(4-piperidin-1-ylanilino)propyl]benzoyl]amino]propanoic acid | Ki | 2000.0 [1] |
 | 3-[[4-[2-(4-Tert-butylphenyl)-3-oxo-3-(4-pyrazol-1-ylanilino)propyl]benzoyl]amino]propanoic acid | Ki | 2000.0 [1] |
 | 3-[[4-[2-(4-Tert-butylphenyl)-3-[4-(2,4-dichlorophenyl)anilino]-3-oxopropyl]benzoyl]amino]propanoic acid | Ki | 33.0 [1] |
 | 3-[[4-[2-(4-Tert-butylphenyl)-3-[4-(4-methylphenyl)piperazin-1-yl]-3-oxopropyl]benzoyl]amino]propanoic acid | Ki | 2000.0 [1] |
 | 3-[[4-[1-[4-(2,4-Dichlorophenyl)anilino]-1-oxooctan-2-yl]oxybenzoyl]amino]propanoic acid | Ki | 14.0 [1] |
 | 3-[[4-[2-(4-Tert-butylphenyl)-3-[4-(hydroxymethyl)anilino]-3-oxopropyl]benzoyl]amino]propanoic acid | Ki | 1000.0 [1] |
 | 3-[[4-[1-(4-Tert-butylphenyl)-2-oxo-2-(4-phenylanilino)ethoxy]benzoyl]amino]-2-fluoropropanoic acid | Ki | 2000.0 [1] |
 | 4-[1-(4-Tert-butylphenyl)-2-oxo-2-(4-phenylanilino)ethoxy]-N-(2H-tetrazol-5-yl)benzamide | Ki | 317.0 [1] |
 | 3-[[4-[1-(4-Tert-butylphenyl)-2-oxo-2-(4-phenylanilino)ethoxy]benzoyl]amino]propanoic acid | Ki | 144.0 [1] |
 | 3-[[4-[2-(4-Tert-butylphenyl)-3-(4-ethylpiperazin-1-yl)-3-oxopropyl]benzoyl]amino]propanoic acid | Ki | 2000.0 [1] |
 | 3-{4-[2-(4-Benzofuran-2-yl-phenylcarbamoyl)-octyl]-benzoylamino}-propionic acid | Ki | 20.0 [1] |
 | 3-[[4-[2-(4-Tert-butylphenyl)-3-oxo-3-[4-(trifluoromethoxymethyl)anilino]propyl]benzoyl]amino]propanoic acid | Ki | 2000.0 [1] |
 | 3-[[4-[2-(4-Tert-butylphenyl)-3-oxo-3-(quinolin-3-ylamino)propyl]benzoyl]amino]propanoic acid | Ki | 610.0 [1] |
 | 3-[[4-[1-(4-Tert-butylphenyl)-2-oxo-2-(4-phenylanilino)ethoxy]benzoyl]amino]-2-hydroxypropanoic acid | Ki | 2000.0 [1] |
 | 3-{4-[1-(4-Benzofuran-2-yl-phenylcarbamoyl)-heptyloxy]-benzoylamino}-propionic acid | Ki | 17.0 [1] |
 | (4R,7S,10S,13S,16R)-N-[(2S)-6-Amino-1-[[(2S)-1-amino-5-(diaminomethylideneamino)-1-oxopentan-2-yl]amino]-1-oxohexan-2-yl]-7-(2-amino-2-oxoethyl)-13-benzyl-20,20-dicyclopentyl-16-[(4-ethoxyphenyl)methyl]-6,9,12,15,18-pentaoxo-10-propan-2-yl-1,2-dithia-5,8,11,14,17-pentazacycloicosane-4-carboxamide | Ki | 4.2 [1] |
 | (4R,7S,10S,13S,16R)-7-(2-Amino-2-oxoethyl)-13-benzyl-20,20-dicyclopentyl-N-[(2S)-5-(diaminomethylideneamino)-1-[[(2S)-1,6-diamino-1-oxohexan-2-yl]amino]-1-oxopentan-2-yl]-16-[(4-ethoxyphenyl)methyl]-6,9,12,15,18-pentaoxo-10-propan-2-yl-1,2-dithia-5,8,11,14,17-pentazacycloicosane-4-carboxamide | Ki | 2.6 [1] |
 | (4R,7S,10S,13S,16S)-N-[(2R)-1-[[(2R)-1-Amino-5-(diaminomethylideneamino)-1-oxopentan-2-yl]amino]-5-(diaminomethylideneamino)-1-oxopentan-2-yl]-7-(2-amino-2-oxoethyl)-13-benzyl-20,20-dicyclopentyl-16-[(4-ethoxyphenyl)methyl]-6,9,12,15,18-pentaoxo-10-propan-2-yl-1,2-dithia-5,8,11,14,17-pentazacycloicosane-4-carboxamide | Ki | 0.88 [1] |
 | (2S)-2-[[(2S)-2-[[(4R,7S,10S,13S,16S)-7-(2-Amino-2-oxoethyl)-13-benzyl-20,20-dicyclopentyl-16-[(4-ethoxyphenyl)methyl]-6,9,12,15,18-pentaoxo-10-propan-2-yl-1,2-dithia-5,8,11,14,17-pentazacycloicosane-4-carbonyl]amino]-5-(diaminomethylideneamino)pentanoyl]amino]-5-(diaminomethylideneamino)pentanoic acid | Ki | 7.8 [1] |
 | (4R,7S,10S,13S,16S)-N-[(2S)-1-[[(2S)-1-Amino-5-(diaminomethylideneamino)-1-oxopentan-2-yl]amino]-5-(diaminomethylideneamino)-1-oxopentan-2-yl]-7-(2-amino-2-oxoethyl)-13-benzyl-20,20-dicyclopentyl-16-[(4-ethoxyphenyl)methyl]-6,9,12,15,18-pentaoxo-10-propan-2-yl-1,2-dithia-5,8,11,14,17-pentazacycloicosane-4-carboxamide | Ki | 1.7 [1] |
 | (4R,7S,10S,13S,16S)-N-[(2R)-1-[[(2S)-1-Amino-5-(diaminomethylideneamino)-1-oxopentan-2-yl]amino]-5-(diaminomethylideneamino)-1-oxopentan-2-yl]-7-(2-amino-2-oxoethyl)-13-benzyl-20,20-dicyclopentyl-16-[(4-ethoxyphenyl)methyl]-6,9,12,15,18-pentaoxo-10-propan-2-yl-1,2-dithia-5,8,11,14,17-pentazacycloicosane-4-carboxamide | Ki | 1.9 [1] |
 | (4R,7S,10S,13S,16S)-N-[(2S)-1-Amino-5-(diaminomethylideneamino)-1-oxopentan-2-yl]-7-(2-amino-2-oxoethyl)-13-benzyl-20,20-dicyclopentyl-16-[(4-ethoxyphenyl)methyl]-6,9,12,15,18-pentaoxo-10-propan-2-yl-1,2-dithia-5,8,11,14,17-pentazacycloicosane-4-carboxamide | Ki | 2.5 [1] |
 | (4R,7S,10S,13S,16S)-N-[(2S)-1-[[(2R)-1-Amino-5-(diaminomethylideneamino)-1-oxopentan-2-yl]amino]-5-(diaminomethylideneamino)-1-oxopentan-2-yl]-7-(2-amino-2-oxoethyl)-13-benzyl-20,20-dicyclopentyl-16-[(4-ethoxyphenyl)methyl]-6,9,12,15,18-pentaoxo-10-propan-2-yl-1,2-dithia-5,8,11,14,17-pentazacycloicosane-4-carboxamide | Ki | 1.7 [1] |
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