 | Ilomastat | IC50 | 1.0 [1], 56.3 [2] |
 | Apratastat | IC50 | 85.0 [1] |
 | Grassystatin A | IC50 | 10000.0 [1], 46100.0 [2] |
 | (6S,7S)-N-Hydroxy-5-methyl-6-[4-[5-(trifluoromethyl)pyridin-2-yl]piperazine-1-carbonyl]-5-azaspiro[2.5]octane-7-carboxamide | IC50 | 5000.0 [1] |
 | (6S,7S)-N-Hydroxy-5-methyl-6-[4-[5-(trifluoromethyl)pyridin-2-yl]piperazine-1-carbonyl]-5-azaspiro[2.5]octane-7-carboxamide | Ki | 2200.0 [1] |
 | Pepstatin | IC50 | 56.3 [1] |
 | Unii-Q56UE7E40Y | IC50 | 5000.0 [1] |
 | (3S)-2-[Ethoxy-(4-methoxyphenyl)phosphoryl]-N-hydroxy-3,4-dihydro-1H-isoquinoline-3-carboxamide | IC50 | 10000.0 [1] |
 | Grassystatin B | IC50 | 85500.0 [1] |
 | N-Hydroxy-2-[methoxy-(4-methoxyphenyl)phosphoryl]-3,4-dihydro-1H-isoquinoline-3-carboxamide | IC50 | 70.0 [1] |
 | 2-[Ethoxy-(4-methoxyphenyl)phosphoryl]-N-hydroxy-3,4-dihydro-1H-isoquinoline-3-carboxamide | IC50 | 230.0 [1] |
 | 2-[Ethoxy-(4-methoxyphenyl)phosphoryl]-N-hydroxy-3,4-dihydro-1H-isoquinoline-3-carboxamide | IC50 | 10000.0 [1] |
 | (3S)-2-[Ethoxy-(4-methoxyphenyl)phosphoryl]-N-hydroxy-3,4-dihydro-1H-isoquinoline-3-carboxamide | IC50 | 10000.0 [1] |
 | 5-((5-Methoxy-3-oxo-1H-indazol-2(3H)-yl)methyl)-5-methylimidazolidine-2,4-dione | Ki | 10000.0 [1] |
 | 6-[Ethoxy-(4-methoxyphenyl)phosphoryl]-N-hydroxy-7,8-dihydro-5H-pyrido[3,4-b]pyrazine-7-carboxamide | IC50 | 560.0 [1] |
 | N-Hydroxy-3-[methyl-[4-[(2-methylquinolin-4-yl)methoxy]phenyl]sulfonylamino]-1-(2-methylpropanoyl)azetidine-3-carboxamide | IC50 | 90.0 [1] |
 | N-Hydroxy-1-(3-methylbutanoyl)-3-[methyl-[4-[(2-methylquinolin-4-yl)methoxy]phenyl]sulfonylamino]azetidine-3-carboxamide | IC50 | 480.0 [1] |
 | 1-(2,2-Dimethylpropanoyl)-N-hydroxy-4-[4-[(2-methyl-5,6,7,8-tetrahydroquinolin-4-yl)methoxy]phenyl]sulfonylpiperazine-2-carboxamide | IC50 | 10000.0 [1] |
 | Grassystatin C | IC50 | 100000.0 [1] |
 | 2-[2-(Diethylamino)ethoxy-(4-methoxyphenyl)phosphoryl]-N-hydroxy-3,4-dihydro-1H-isoquinoline-3-carboxamide | IC50 | 1140.0 [1] |
 | 2-[Ethoxy-(4-phenoxyphenyl)phosphoryl]-N-hydroxy-3,4-dihydro-1H-isoquinoline-3-carboxamide | IC50 | 260.0 [1] |
 | 2-[[4-(4-Aminophenoxy)phenyl]-ethoxyphosphoryl]-N-hydroxy-3,4-dihydro-1H-isoquinoline-3-carboxamide | IC50 | 1670.0 [1] |
 | N-Hydroxy-2-[(4-methoxyphenyl)-(2-phenylethoxy)phosphoryl]-3,4-dihydro-1H-isoquinoline-3-carboxamide | IC50 | 3110.0 [1] |
 | 2-[Ethoxy-(4-pyridin-4-yloxyphenyl)phosphoryl]-N-hydroxy-3,4-dihydro-1H-isoquinoline-3-carboxamide | IC50 | 660.0 [1] |
 | N-Hydroxy-2-[(4-methoxyphenyl)-[2-(4-phenylphenyl)ethoxy]phosphoryl]-3,4-dihydro-1H-isoquinoline-3-carboxamide | IC50 | 3560.0 [1] |
 | 2-[Cyclohexylmethoxy-(4-methoxyphenyl)phosphoryl]-N-hydroxy-3,4-dihydro-1H-isoquinoline-3-carboxamide | IC50 | 1340.0 [1] |
 | 2-[Ethoxy(thiophen-2-yl)phosphoryl]-N-hydroxy-3,4-dihydro-1H-isoquinoline-3-carboxamide | IC50 | 890.0 [1] |
 | 2-[(4-Aminophenyl)-ethoxyphosphoryl]-N-hydroxy-3,4-dihydro-1H-isoquinoline-3-carboxamide | IC50 | 660.0 [1] |
 | 2-[Ethoxy(pyridin-4-yl)phosphoryl]-N-hydroxy-3,4-dihydro-1H-isoquinoline-3-carboxamide | IC50 | 2600.0 [1] |
 | 2-[Ethoxy-(2-fluorophenyl)phosphoryl]-N-hydroxy-3,4-dihydro-1H-isoquinoline-3-carboxamide | IC50 | 1060.0 [1] |
 | 7-Amino-2-[ethoxy-(4-methoxyphenyl)phosphoryl]-N-hydroxy-3,4-dihydro-1H-isoquinoline-3-carboxamide | IC50 | 190.0 [1] |
 | 2-[Ethoxy-(3-fluorophenyl)phosphoryl]-N-hydroxy-3,4-dihydro-1H-isoquinoline-3-carboxamide | IC50 | 830.0 [1] |
 | 2-[Ethoxy-(4-methoxyphenyl)phosphoryl]-N-hydroxy-1,3,4,9-tetrahydropyrido[3,4-b]indole-3-carboxamide | IC50 | 800.0 [1] |
 | (2-Hydroxycarbamoyl-pyrrolidin-1-yl)-(4-methoxy-phenyl)-phosphinic acid ethyl ester | IC50 | 10000.0 [1] |
 | N-Hydroxy-2-[(4-methoxyphenyl)-(2-pyridin-2-ylethoxy)phosphoryl]-3,4-dihydro-1H-isoquinoline-3-carboxamide | IC50 | 180.0 [1] |
 | 2-[Ethoxy-(4-fluorophenyl)phosphoryl]-N-hydroxy-3,4-dihydro-1H-isoquinoline-3-carboxamide | IC50 | 300.0 [1] |
 | 2-[Ethoxy-(4-methylphenyl)phosphoryl]-N-hydroxy-3,4-dihydro-1H-isoquinoline-3-carboxamide | IC50 | 1890.0 [1] |
 | (3-Hydroxycarbamoyl-3,4-dihydro-1H-isoquinolin-2-yl)-styryl-phosphinic acid ethyl ester | IC50 | 910.0 [1] |
 | (3-Hydroxycarbamoyl-3,4-dihydro-1H-isoquinolin-2-yl)-phenyl-phosphinic acid ethyl ester | IC50 | 370.0 [1] |
 | 2-[2-Ethoxyethoxy-(4-methoxyphenyl)phosphoryl]-N-hydroxy-3,4-dihydro-1H-isoquinoline-3-carboxamide | IC50 | 510.0 [1] |
 | Benzyl 4-[ethoxy-(4-methoxyphenyl)phosphoryl]-3-(hydroxycarbamoyl)piperazine-1-carboxylate | IC50 | 430.0 [1] |
 | 5-[Ethoxy-(4-methoxyphenyl)phosphoryl]-N-hydroxy-6,7-dihydro-4H-thieno[3,2-c]pyridine-6-carboxamide | IC50 | 520.0 [1] |
 | 2-[Ethoxy-(4-phenylphenyl)phosphoryl]-N-hydroxy-3,4-dihydro-1H-isoquinoline-3-carboxamide | IC50 | 1960.0 [1] |
 | 2-[Ethoxy-[4-(2-ethoxyethoxy)phenyl]phosphoryl]-N-hydroxy-3,4-dihydro-1H-isoquinoline-3-carboxamide | IC50 | 70.0 [1] |
 | N-Hydroxy-2-[(4-methoxyphenyl)-propan-2-yloxyphosphoryl]-3,4-dihydro-1H-isoquinoline-3-carboxamide | IC50 | 2240.0 [1] |
 | 2-[Hexoxy-(4-methoxyphenyl)phosphoryl]-N-hydroxy-3,4-dihydro-1H-isoquinoline-3-carboxamide | IC50 | 1600.0 [1] |
 | 2-[Ethoxy(2-phenylethyl)phosphoryl]-N-hydroxy-3,4-dihydro-1H-isoquinoline-3-carboxamide | IC50 | 700.0 [1] |
 | 2-[Butoxy-(4-methoxyphenyl)phosphoryl]-N-hydroxy-3,4-dihydro-1H-isoquinoline-3-carboxamide | IC50 | 810.0 [1] |
 | (2S)-N-Hydroxy-3-[[4-[(2-methylquinolin-4-yl)methoxy]phenyl]sulfonylamino]-2-(4-propan-2-ylsulfonylpiperazin-1-yl)propanamide | IC50 | 10000.0 [1] |
 | (2S)-2-[4-[(4-Fluorophenyl)methyl]piperazin-1-yl]-N-hydroxy-3-[[4-[(2-methylquinolin-4-yl)methoxy]phenyl]sulfonylamino]propanamide | IC50 | 9254.0 [1] |
 | (2S)-2-(4-Ethylpiperazin-1-yl)-N-hydroxy-3-[[4-[(2-methylquinolin-4-yl)methoxy]phenyl]sulfonylamino]propanamide | IC50 | 3054.0 [1] |
 | (2S)-N-Hydroxy-3-[[4-[(2-methylquinolin-4-yl)methoxy]phenyl]sulfonylamino]-2-[4-[[4-(trifluoromethyl)phenyl]methyl]piperazin-1-yl]propanamide | IC50 | 10000.0 [1] |
 | (2S)-N-Hydroxy-2-[4-[(4-methylphenyl)methyl]piperazin-1-yl]-3-[[4-[(2-methylquinolin-4-yl)methoxy]phenyl]sulfonylamino]propanamide | IC50 | 10000.0 [1] |
 | (2S)-N-Hydroxy-2-[4-(2-methylpropanoyl)piperazin-1-yl]-3-[[4-[(2-methylquinolin-4-yl)methoxy]phenyl]sulfonylamino]propanamide | IC50 | 10000.0 [1] |
 | (2S)-N-Hydroxy-2-[4-(2-methylpropylsulfonyl)piperazin-1-yl]-3-[[4-[(2-methylquinolin-4-yl)methoxy]phenyl]sulfonylamino]propanamide | IC50 | 10000.0 [1] |
 | (2S)-N-Hydroxy-3-[[4-[(2-methylquinolin-4-yl)methoxy]phenyl]sulfonylamino]-2-(4-methylsulfonylpiperazin-1-yl)propanamide | IC50 | 10000.0 [1] |
 | 4-But-2-ynoxy-N-[(2S)-3-(hydroxyamino)-2-(4-methylsulfonylpiperazin-1-yl)-3-oxopropyl]benzamide | IC50 | 3251.0 [1] |
 | N-[(2S)-3-(Hydroxyamino)-2-(4-methylsulfonylpiperazin-1-yl)-3-oxopropyl]-4-[(2-methylquinolin-4-yl)methoxy]benzamide | IC50 | 10000.0 [1] |
 | N-[(2S)-3-(Hydroxyamino)-3-oxo-2-piperidin-1-ylpropyl]-4-[(2-methylquinolin-4-yl)methoxy]benzamide | IC50 | 10000.0 [1] |
 | N-[(2S)-3-(Hydroxyamino)-3-oxo-2-piperidin-1-ylpropyl]-4-[(2-phenylpyridin-4-yl)methoxy]benzamide | IC50 | 10000.0 [1] |
 | N-[(2S)-3-(Hydroxyamino)-3-oxo-2-piperidin-1-ylpropyl]-4-(pyridin-4-ylmethoxy)benzamide | IC50 | 10000.0 [1] |
 | N-[(2S)-2-(Diethylamino)-3-(hydroxyamino)-3-oxopropyl]-4-[(2-methylquinolin-4-yl)methoxy]benzamide | IC50 | 10000.0 [1] |
 | N-[2-(4-Benzylpiperazin-1-yl)-3-(hydroxyamino)-3-oxopropyl]-4-[[2-(trifluoromethyl)pyrazolo[1,5-a]pyridin-3-yl]methoxy]benzamide | IC50 | 10000.0 [1] |
 | N-Hydroxy-4-[4-(4-hydroxybut-2-ynoxy)phenyl]sulfonyl-2,2-dimethylthiomorpholine-3-carboxamide | IC50 | 85.0 [1] |