| 4-(6-(4-(Piperazin-1-yl)phenyl)pyrazolo[1,5-a]pyrimidin-3-yl)quinoline | IC50 | 43.29 [1], 1825.0 [2] |
| Staurosporine | IC50 | 9118.0 [1] |
| Dorsomorphin | IC50 | 25740.0 [1] |
| Doramapimod | IC50 | 44000.0 [1] |
| Galunisertib | IC50 | 199.0 [1] |
| 2-(4-(Benzo[d][1,3]dioxol-5-yl)-2-tert-butyl-1H-imidazol-5-yl)-6-methylpyridine | IC50 | 70.0 [1] |
| 4-(4-(3-(Pyridin-2-yl)-1H-pyrazol-4-yl)pyridin-2-yl)-N-(tetrahydro-2H-pyran-4-yl)benzamide | IC50 | 1000.0 [1] |
| Benzamide, 3-((4-(6-methyl-2-pyridinyl)-5-(6-quinoxalinyl)-1H-imidazol-2-yl)methyl)- | IC50 | 23.0 [1] |
| Vactosertib | IC50 | 13.0 [1] |
| 5-[6-[4-(1-Piperazinyl)phenyl]pyrazolo[1,5-a]pyrimidin-3-yl]quinoline | IC50 | 4090.0 [1] |
| 4-[6-(4-Propan-2-yloxyphenyl)pyrazolo[1,5-a]pyrimidin-3-yl]quinoline | IC50 | 9622.0 [1] |
| Khk-IN-1 | IC50 | 40000.0 [1] |
| Dimethyl-{2-[(4-{4-[3-(pyridin-2-yl)-1H-pyrazol-4-yl]-2-pyridinyl}phenyl)oxy]ethyl}amine | IC50 | 46.0 [1] |
| 4-(6-(4-Methoxyphenyl)pyrazolo[1,5-a]pyrimidin-3-yl)quinoline | IC50 | 1840.0 [1] |
| 5-(2-Amino-[1,2,4]triazolo[1,5-a]pyridin-7-yl)-N-tert-butylpyridine-3-sulfonamide | IC50 | 10000.0 [1] |
| 1-[5-Tert-butyl-3-[4-[2-(dimethylamino)ethyl]-5-oxo-1,4-diazepane-1-carbonyl]thiophen-2-yl]-3-(2,3-dichlorophenyl)urea | IC50 | 35000.0 [1] |
| CID 60182364 | IC50 | 183.0 [1] |
| CID 60182389 | IC50 | 326.0 [1] |
| 4-(4-(3-(1H-Pyrazol-4-yl)pyrazolo[1,5-a]pyrimidin-6-yl)phenyl)morpholine | IC50 | 5930.0 [1] |
| 2-Anilino-7-[(1S)-4-hydroxy-2,3-dihydro-1H-inden-1-yl]-5,5-dimethylpyrrolo[2,3-d]pyrimidin-6-one | IC50 | 10000.0 [1] |
| N-[4-[3-[5-(Trideuteriomethoxy)pyridin-2-yl]-1H-pyrrolo[3,2-b]pyridin-2-yl]pyridin-2-yl]acetamide | IC50 | 100.0 [1] |
| N-[4-[3-[6-(Difluoromethyl)pyridin-2-yl]-1H-pyrrolo[3,2-b]pyridin-2-yl]pyridin-2-yl]acetamide | IC50 | 100.0 [1] |
| (4S,9S,10S)-9,10,18-Trihydroxy-16-methoxy-4-methyl-3-oxabicyclo[12.4.0]octadeca-1(14),15,17-triene-2,8-dione | IC50 | 2761.0 [1] |
| Alk2-IN-2 | IC50 | 18330.0 [1] |
| 2-Pyrazol-1-yl-4-(5-pyridin-2-yl-1H-pyrazol-4-yl)pyridine | IC50 | 882.0 [1] |
| 2-(1-Methylpyrazol-4-yl)-4-(5-pyridin-2-yl-1H-pyrazol-4-yl)pyridine | IC50 | 224.0 [1] |
| 1-Methyl-4-[5-[4-(5-pyridin-2-yl-1H-pyrazol-4-yl)pyridin-2-yl]pyridin-2-yl]piperazine | IC50 | 108.0 [1] |
| N,N-Dimethyl-3-[5-[4-(5-pyridin-2-yl-1H-pyrazol-4-yl)pyridin-2-yl]pyridin-2-yl]oxypropan-1-amine | IC50 | 18.0 [1] |
| 2-Imidazol-1-yl-4-(5-pyridin-2-yl-1H-pyrazol-4-yl)pyridine | IC50 | 956.0 [1] |
| 6-(4-Piperazin-1-ylphenyl)-3-(1H-pyrazol-4-yl)pyrazolo[1,5-a]pyrimidine | IC50 | 3420.0 [1] |
| 8-N-(Cyclopropylmethyl)-4-N-(2-methylsulfanylphenyl)-2-(4-piperidin-4-ylpiperazin-1-yl)pyrimido[5,4-d]pyrimidine-4,8-diamine | IC50 | 10000.0 [1] |
| 3-Methyl-6-[2-(6-methylpyridin-2-yl)pyrazol-3-yl]quinazolin-4-one | IC50 | 59.0 [1] |
| N-[4-[(6-Chloro-[1,3]dioxolo[4,5-B]pyridin-7-Yl)amino]-2-Pyridyl]cyclopropanecarboxamide | IC50 | 31.0 [1] |