![](https://images.aatbio.com/dataset/ic50/activin-receptor-type-1_4744f719e061d188f64f7298e92769bc.svg) | 4-(6-(4-(Piperazin-1-yl)phenyl)pyrazolo[1,5-a]pyrimidin-3-yl)quinoline | IC50 | 3.26 [1], 17.0 [2], 40.7 [3] |
![](https://images.aatbio.com/dataset/ic50/activin-receptor-type-1_25bb7c73525ae09d6bb7f575a6958c76.svg) | 4-[6-(4-Propan-2-yloxyphenyl)pyrazolo[1,5-a]pyrimidin-3-yl]quinoline | IC50 | 100.0 [1], 107.9 [2] |
![](https://images.aatbio.com/dataset/ic50/activin-receptor-type-1_d2aaae557a3df420b61b69998679cc44.svg) | Dorsomorphin | IC50 | 67.5 [1], 148.1 [2] |
![](https://images.aatbio.com/dataset/ic50/activin-receptor-type-1_77133570e896153ed2bcf3545f22a0e5.svg) | 1-(4-(6-Methyl-5-(3,4,5-trimethoxyphenyl)pyridin-3-yl)phenyl)piperazine | IC50 | 24.0 [1], 27.0 [2] |
![](https://images.aatbio.com/dataset/ic50/activin-receptor-type-1_43448187fad0a0db3095c2031784e2a3.svg) | (4S,9S,10S)-9,10,18-Trihydroxy-16-methoxy-4-methyl-3-oxabicyclo[12.4.0]octadeca-1(14),15,17-triene-2,8-dione | IC50 | 217.0 [1], 3353.0 [2] |
![](https://images.aatbio.com/dataset/ic50/activin-receptor-type-1_1d5eba4b4bb57896dda18b1604bab021.svg) | Staurosporine | IC50 | 10005.0 [1] |
![](https://images.aatbio.com/dataset/ic50/activin-receptor-type-1_a257c791d1de1df5d4a1fa04612f9c76.svg) | Nvp-aew541 | IC50 | 2900.0 [1] |
![](https://images.aatbio.com/dataset/ic50/activin-receptor-type-1_bca7f3db243d5647ee899b9d088c6b6c.svg) | Vactosertib | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/activin-receptor-type-1_ff0d43edb17f983137c243b2b294bebc.svg) | 3-[6-Amino-5-(3,4,5-Trimethoxyphenyl)pyridin-3-Yl]phenol | IC50 | 35.0 [1] |
![](https://images.aatbio.com/dataset/ic50/activin-receptor-type-1_7c61426636de742e3bc9e56260715465.svg) | 5-[6-[4-(1-Piperazinyl)phenyl]pyrazolo[1,5-a]pyrimidin-3-yl]quinoline | IC50 | 26.2 [1] |
![](https://images.aatbio.com/dataset/ic50/activin-receptor-type-1_3940d1581c72730211474d10f75b49fe.svg) | 5-[6-(4-Methoxyphenyl)pyrazolo[1,5-a]pyrimidin-3-yl]quinoline | IC50 | 32.0 [1] |
![](https://images.aatbio.com/dataset/ic50/activin-receptor-type-1_f582e48a8747f8841ea380984678484a.svg) | 4-[4-[(Dimethylamino)methyl]-2,5-Dimethoxy-Phenyl]-2-Methyl-2,7-Naphthyridin-1-One | IC50 | 5090.0 [1] |
![](https://images.aatbio.com/dataset/ic50/activin-receptor-type-1_27155136dbc077658c8857b4cc311fec.svg) | 4-[2-[4-(3-Phenylpyrazolo[1,5-a]pyrimidin-6-yl)phenoxy]ethyl]morpholine | IC50 | 2570.0 [1] |
![](https://images.aatbio.com/dataset/ic50/activin-receptor-type-1_a1f0a177d77a1f7fc2f33030a8ca8f2f.svg) | 4-[4-[(Dimethylamino)methyl]-3,5-Dimethoxy-Phenyl]-2-Methyl-2,7-Naphthyridin-1-One | IC50 | 5130.0 [1] |
![](https://images.aatbio.com/dataset/ic50/activin-receptor-type-1_b076cdaba7bb8b7d9a4e8120c86a34a8.svg) | N-Propyl-4-({4-[(2,2,2-trifluoroethyl)amino]-1H-pyrrolo[2,3-d]pyrimidin-2-yl}amino)benzamide | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/activin-receptor-type-1_3690b6820a353232ff0cbe080abaf2b0.svg) | 4-(6-(4-Methoxyphenyl)pyrazolo[1,5-a]pyrimidin-3-yl)quinoline | IC50 | 33.3 [1] |
![](https://images.aatbio.com/dataset/ic50/activin-receptor-type-1_a7ee75d4a7ce2e8d7ffa73cb444c324f.svg) | 5-(2-Amino-[1,2,4]triazolo[1,5-a]pyridin-7-yl)-N-tert-butylpyridine-3-sulfonamide | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/activin-receptor-type-1_12ca6da21f5fd32ed946d0ce3dcbb3ef.svg) | CID 60182364 | IC50 | 5.0 [1] |
![](https://images.aatbio.com/dataset/ic50/activin-receptor-type-1_9ff18c07942722398a15ef844b620ff9.svg) | CID 60182389 | IC50 | 5.0 [1] |
![](https://images.aatbio.com/dataset/ic50/activin-receptor-type-1_412de614e4031e722d3d92aad63f1520.svg) | 4-(4-(3-(1H-Pyrazol-4-yl)pyrazolo[1,5-a]pyrimidin-6-yl)phenyl)morpholine | IC50 | 53.4 [1] |
![](https://images.aatbio.com/dataset/ic50/activin-receptor-type-1_ef431bf27ff7842bbb4caafd947b43c7.svg) | Tilfrinib | IC50 | 220.0 [1] |
![](https://images.aatbio.com/dataset/ic50/activin-receptor-type-1_4f5d2c8450283020f2d640dc5aa7efbf.svg) | 4-[6-[4-[(2S,6R)-2,6-Dimethylpiperazin-1-yl]phenyl]pyrazolo[1,5-a]pyrimidin-3-yl]quinoline | IC50 | 9.0 [1] |
![](https://images.aatbio.com/dataset/ic50/activin-receptor-type-1_6064c420308a7d1ef6bb9c4609b7804b.svg) | 5-(3-Piperazin-1-ylphenyl)-3-(3,4,5-trimethoxyphenyl)pyridin-2-amine | IC50 | 17.0 [1] |
![](https://images.aatbio.com/dataset/ic50/activin-receptor-type-1_35bd35df1541bfed036a1acfb8784db4.svg) | 5-(4-Piperazin-1-ylphenyl)-3-quinolin-4-ylpyridin-2-amine | IC50 | 120.0 [1] |
![](https://images.aatbio.com/dataset/ic50/activin-receptor-type-1_a1ab92c4a58a4f13a706d2880af25ee9.svg) | 5-(4-Piperazin-1-ylphenyl)-3-(3-propan-2-yloxyphenyl)pyridin-2-amine | IC50 | 790.0 [1] |
![](https://images.aatbio.com/dataset/ic50/activin-receptor-type-1_ee9bea86fa6dd7d5ba39b740cee25ccf.svg) | 3-(4-Chloro-3-methoxyphenyl)-5-(4-piperazin-1-ylphenyl)pyridin-2-amine | IC50 | 63.0 [1] |
![](https://images.aatbio.com/dataset/ic50/activin-receptor-type-1_1efebba178ba1b19b74bcb7d3c1111f2.svg) | 3-(3,4-Dimethoxyphenyl)-5-(4-piperazin-1-ylphenyl)pyridin-2-amine | IC50 | 23.0 [1] |
![](https://images.aatbio.com/dataset/ic50/activin-receptor-type-1_5693da5e8b82fdcbcecff172c35b8f06.svg) | 3-(3-Methoxy-4-methylphenyl)-5-(4-piperazin-1-ylphenyl)pyridin-2-amine | IC50 | 110.0 [1] |
![](https://images.aatbio.com/dataset/ic50/activin-receptor-type-1_ff0c7cea372fbb405fc2c071ffdbae9b.svg) | 3-(3-Methoxyphenyl)-5-(4-piperazin-1-ylphenyl)pyridin-2-amine | IC50 | 86.0 [1] |
![](https://images.aatbio.com/dataset/ic50/activin-receptor-type-1_9884b2945a4321a86a4f31d51bc4fd77.svg) | 6-(4-Piperazin-1-ylphenyl)-3-(3,4,5-trimethoxyphenyl)pyrazolo[1,5-a]pyrimidine | IC50 | 10.0 [1] |
![](https://images.aatbio.com/dataset/ic50/activin-receptor-type-1_aa654ff86c0dc0ea1cde8a8dec943955.svg) | 3-[6-[4-[(2S,6R)-2,6-Dimethylpiperazin-1-yl]phenyl]pyrazolo[1,5-a]pyrimidin-3-yl]benzenesulfonamide | IC50 | 109.0 [1] |
![](https://images.aatbio.com/dataset/ic50/activin-receptor-type-1_ff28abd4c50694e887b226b1fab683cb.svg) | 4-[6-[4-[(2S,6R)-2,6-Dimethylpiperazin-1-yl]phenyl]pyrazolo[1,5-a]pyrimidin-3-yl]-2-methylbenzenesulfonamide | IC50 | 246.0 [1] |
![](https://images.aatbio.com/dataset/ic50/activin-receptor-type-1_856fa2124b27d61b83553dc565511d49.svg) | 2-Amino-4-[6-[4-[(2R,6S)-2,6-dimethylpiperazin-1-yl]phenyl]pyrazolo[1,5-a]pyrimidin-3-yl]benzenesulfonamide | IC50 | 291.0 [1] |
![](https://images.aatbio.com/dataset/ic50/activin-receptor-type-1_73839304920c5549caa183bb78ae2408.svg) | 4-[6-[4-[(2S,6R)-2,6-Dimethylpiperazin-1-yl]phenyl]pyrazolo[1,5-a]pyrimidin-3-yl]naphthalene-1-sulfonamide | IC50 | 19.0 [1] |
![](https://images.aatbio.com/dataset/ic50/activin-receptor-type-1_2ce2b33dd8dafe53639097680d3912ca.svg) | 4-[6-[4-(2-Piperidin-1-ylethoxy)phenyl]pyrazolo[1,5-a]pyrimidin-3-yl]naphthalene-1-sulfonamide | IC50 | 63.0 [1] |
![](https://images.aatbio.com/dataset/ic50/activin-receptor-type-1_b2efc5e6798c70a05b82b8ef48666778.svg) | 4-[6-[4-[(2S,6R)-2,6-Dimethylpiperazin-1-yl]phenyl]pyrazolo[1,5-a]pyrimidin-3-yl]-N,N-dimethylnaphthalene-1-sulfonamide | IC50 | 5990.0 [1] |
![](https://images.aatbio.com/dataset/ic50/activin-receptor-type-1_d3c6b447894acbff39fee64210f97a26.svg) | 4-[6-[4-[(2S,6R)-2,6-Dimethylpiperazin-1-yl]phenyl]pyrazolo[1,5-a]pyrimidin-3-yl]-N-methylnaphthalene-1-sulfonamide | IC50 | 326.0 [1] |
![](https://images.aatbio.com/dataset/ic50/activin-receptor-type-1_a6ebbb44f1217a3af89eb8f0430e2fd9.svg) | 4-[6-[4-(2-Methyl-1-piperidin-1-ylpropan-2-yl)oxyphenyl]pyrazolo[1,5-a]pyrimidin-3-yl]naphthalene-1-sulfonamide | IC50 | 47.0 [1] |
![](https://images.aatbio.com/dataset/ic50/activin-receptor-type-1_8e4d3ef32e6f44246e96e3b0e88b1a94.svg) | 6-[4-[(2S,6R)-2,6-Dimethylpiperazin-1-yl]phenyl]-3-(4-methylsulfonylphenyl)pyrazolo[1,5-a]pyrimidine | IC50 | 1971.0 [1] |
![](https://images.aatbio.com/dataset/ic50/activin-receptor-type-1_f9cf80575e6b8831015a4b299421c268.svg) | 4-[6-(6-Piperazin-1-ylpyridin-3-yl)pyrazolo[1,5-a]pyrimidin-3-yl]naphthalene-1-sulfonamide | IC50 | 422.0 [1] |
![](https://images.aatbio.com/dataset/ic50/activin-receptor-type-1_5b48c3cd6f71ee6ba6a2d7c2415bfe9b.svg) | 4-[6-[4-(2-Aminopropan-2-yl)phenyl]pyrazolo[1,5-a]pyrimidin-3-yl]naphthalene-1-sulfonamide | IC50 | 29.0 [1] |
![](https://images.aatbio.com/dataset/ic50/activin-receptor-type-1_8ed849936b3ae6f8799edf9ac45a18f2.svg) | 4-[6-[6-(2-Piperidin-1-ylethoxy)pyridin-3-yl]pyrazolo[1,5-a]pyrimidin-3-yl]naphthalene-1-sulfonamide | IC50 | 738.0 [1] |
![](https://images.aatbio.com/dataset/ic50/activin-receptor-type-1_66e08e2cbc7ecec55cab43c93814d7f0.svg) | N-[4-[6-[4-[(2S,6R)-2,6-Dimethylpiperazin-1-yl]phenyl]pyrazolo[1,5-a]pyrimidin-3-yl]naphthalen-1-yl]methanesulfonamide | IC50 | 796.0 [1] |
![](https://images.aatbio.com/dataset/ic50/activin-receptor-type-1_a12c79ee3319806748c6a323d9a4a799.svg) | 4-[6-[4-(Pyrrolidin-1-ylmethyl)phenyl]pyrazolo[1,5-a]pyrimidin-3-yl]naphthalene-1-sulfonamide | IC50 | 27.0 [1] |
![](https://images.aatbio.com/dataset/ic50/activin-receptor-type-1_5192474bf6e20f4b859d2a34a9e32e88.svg) | 4-[6-[4-(2-Pyrrolidin-1-ylethoxy)phenyl]pyrazolo[1,5-a]pyrimidin-3-yl]naphthalene-1-sulfonamide | IC50 | 48.0 [1] |
![](https://images.aatbio.com/dataset/ic50/activin-receptor-type-1_4ac996a07f36ebc8e9283c918225a9a2.svg) | 4-[6-[4-(1-Aminocyclobutyl)phenyl]pyrazolo[1,5-a]pyrimidin-3-yl]naphthalene-1-sulfonamide | IC50 | 16.0 [1] |
![](https://images.aatbio.com/dataset/ic50/activin-receptor-type-1_4c18cfbdd0c7c8e982f2803a2d994d54.svg) | 4-[6-[6-[2-(Dimethylamino)ethoxy]pyridin-3-yl]pyrazolo[1,5-a]pyrimidin-3-yl]naphthalene-1-sulfonamide | IC50 | 1026.0 [1] |
![](https://images.aatbio.com/dataset/ic50/activin-receptor-type-1_3208b75cd4f171826a14348e40e2f80c.svg) | 4-[6-[4-[(2S,6R)-2,6-Dimethylpiperazin-1-yl]phenyl]pyrazolo[1,5-a]pyrimidin-3-yl]benzenesulfonamide | IC50 | 526.0 [1] |
![](https://images.aatbio.com/dataset/ic50/activin-receptor-type-1_ea16c1cbbcf11e2b86b7e425bca206cc.svg) | 5-[6-[4-[(2S,6R)-2,6-Dimethylpiperazin-1-yl]phenyl]pyrazolo[1,5-a]pyrimidin-3-yl]naphthalene-1-sulfonamide | IC50 | 54.0 [1] |
![](https://images.aatbio.com/dataset/ic50/activin-receptor-type-1_280a27c441ee007477aeb0213b644bb8.svg) | 4-[6-(4-Piperidin-4-ylphenyl)pyrazolo[1,5-a]pyrimidin-3-yl]naphthalene-1-sulfonamide | IC50 | 93.0 [1] |
![](https://images.aatbio.com/dataset/ic50/activin-receptor-type-1_f603c5babb7df63df8611b461be84c89.svg) | 4-[6-[4-(1-Aminoethyl)phenyl]pyrazolo[1,5-a]pyrimidin-3-yl]naphthalene-1-sulfonamide | IC50 | 25.0 [1] |
![](https://images.aatbio.com/dataset/ic50/activin-receptor-type-1_100925b45550d059944fa6c1998a3b53.svg) | 5-(3-Piperazin-1-ylphenyl)-3-quinolin-4-ylpyridin-2-amine | IC50 | 110.0 [1] |
![](https://images.aatbio.com/dataset/ic50/activin-receptor-type-1_66f36880dc0ccb51d905052f031a5586.svg) | 5-(4-Piperazin-1-ylphenyl)-3-quinolin-5-ylpyridin-2-amine | IC50 | 270.0 [1] |
![](https://images.aatbio.com/dataset/ic50/activin-receptor-type-1_ffcf0060d8899c5d4484924cc80cde8c.svg) | N-[3-[6-Amino-5-(3,4,5-trimethoxyphenyl)pyridin-3-yl]phenyl]methanesulfonamide | IC50 | 6.0 [1] |
![](https://images.aatbio.com/dataset/ic50/activin-receptor-type-1_52a1b06b1aaba6c3dd167b666f0e070d.svg) | 3-(3,5-Dimethoxyphenyl)-5-(4-piperazin-1-ylphenyl)pyridin-2-amine | IC50 | 14.0 [1] |
![](https://images.aatbio.com/dataset/ic50/activin-receptor-type-1_cca55ad4698efd809983ab6d0351ef63.svg) | 3-(2,3-Dihydro-1,4-benzodioxin-6-yl)-5-(4-piperazin-1-ylphenyl)pyridin-2-amine | IC50 | 1870.0 [1] |
![](https://images.aatbio.com/dataset/ic50/activin-receptor-type-1_12c4445cd51f07c97cd04134baa1a329.svg) | 3-(4-Morpholin-4-ylphenyl)-6-quinolin-4-yl-quinazolin-4-one | IC50 | 32.0 [1] |
![](https://images.aatbio.com/dataset/ic50/activin-receptor-type-1_19ee7159e838908f6fd4e209b712057e.svg) | 5-Methyl-6-quinolin-5-yl-3~{H}-quinazolin-4-one | IC50 | 194.0 [1] |
![](https://images.aatbio.com/dataset/ic50/activin-receptor-type-1_d7d52a48817f8cf3a5aea1d3f3bb27d6.svg) | 2,5-Dimethyl-6-quinolin-4-yl-3~{H}-quinazolin-4-one | IC50 | 42.0 [1] |
![](https://images.aatbio.com/dataset/ic50/activin-receptor-type-1_ef3f8c616472a5f444d78be7d9da05f7.svg) | 6-Quinolin-5-yl-3H-quinazolin-4-one | IC50 | 344.0 [1] |
![](https://images.aatbio.com/dataset/ic50/activin-receptor-type-1_9afc6ca4ab83a6ecd16ee93068cb0812.svg) | 6-(1-Methylpyrazol-4-yl)-3H-quinazolin-4-one | IC50 | 18200.0 [1] |
![](https://images.aatbio.com/dataset/ic50/activin-receptor-type-1_c8fe38d2a428fc01911544f6acc1619a.svg) | 6-(1H-Pyrazol-4-yl)-3H-quinazolin-4-one | IC50 | 8200.0 [1] |
![](https://images.aatbio.com/dataset/ic50/activin-receptor-type-1_0b43927816ebbc9be13e6e44e4f9f2e1.svg) | 5,5-Dimethyl-8-[[4-(2,2,2-trifluoroethylamino)furo[3,2-d]pyrimidin-2-yl]amino]-1H-4,1-benzoxazepin-2-one | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/activin-receptor-type-1_7465485b49f08e4cd9a2cea57d31727d.svg) | Alk2-IN-2 | IC50 | 9.0 [1] |
![](https://images.aatbio.com/dataset/ic50/activin-receptor-type-1_10c5a7bbb3ea1bd88a9172e3c330c25b.svg) | 3-[4-(Dimethylamino)phenyl]-6-quinolin-4-ylquinazolin-4-one | IC50 | 68.0 [1] |
![](https://images.aatbio.com/dataset/ic50/activin-receptor-type-1_95da2b984c277fba4018df037a578962.svg) | 6-(3,5-Dimethyl-1H-pyrazol-4-yl)-3H-quinazolin-4-one | IC50 | 293.0 [1] |
![](https://images.aatbio.com/dataset/ic50/activin-receptor-type-1_8208e022a5ff936b1926ce4351029263.svg) | 2-Benzyl-5-methyl-6-quinolin-4-yl-3H-quinazolin-4-one | IC50 | 439.0 [1] |
![](https://images.aatbio.com/dataset/ic50/activin-receptor-type-1_28d11dc5e99a15354396efb00dacd9b2.svg) | 6-(5-Methyl-1H-pyrazol-4-yl)-3H-quinazolin-4-one | IC50 | 2300.0 [1] |
![](https://images.aatbio.com/dataset/ic50/activin-receptor-type-1_4983b1ae34644dd47b593e03ace92308.svg) | 5-Methyl-6-quinolin-4-yl-3H-quinazolin-4-one | IC50 | 220.0 [1] |
![](https://images.aatbio.com/dataset/ic50/activin-receptor-type-1_d8143569b9307ecaccd92dd9bebdbca3.svg) | 3-Cyclohexyl-6-quinolin-4-ylquinazolin-4-one | IC50 | 1525.0 [1] |
![](https://images.aatbio.com/dataset/ic50/activin-receptor-type-1_cb19377c3b27e3864e8a256748138924.svg) | 3-(3-Morpholin-4-ylpropyl)-6-quinolin-4-ylquinazolin-4-one | IC50 | 165.0 [1] |
![](https://images.aatbio.com/dataset/ic50/activin-receptor-type-1_1d07028eecafb4e191013a1c25b6a6f9.svg) | 6-(5-Ethyl-1H-pyrazol-4-yl)-3H-quinazolin-4-one | IC50 | 1000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/activin-receptor-type-1_74582637f2a3c792b2b009ace658a1ee.svg) | 2-Methyl-6-quinolin-5-yl-3H-quinazolin-4-one | IC50 | 138.0 [1] |
![](https://images.aatbio.com/dataset/ic50/activin-receptor-type-1_e546b3d8bccd00afc956c87f043a1868.svg) | 3-Methyl-6-quinolin-4-ylquinazolin-4-one | IC50 | 186.0 [1] |
![](https://images.aatbio.com/dataset/ic50/activin-receptor-type-1_0d3c7c8be88718c3dc9bebcea2d60ca5.svg) | 6-Pyrazolo[1,5-a]pyridin-3-yl-3H-quinazolin-4-one | IC50 | 653.0 [1] |
![](https://images.aatbio.com/dataset/ic50/activin-receptor-type-1_16f8d38d044982cca8679f54a403383f.svg) | 6-Quinolin-4-yl-3H-quinazolin-4-one | IC50 | 167.0 [1] |
![](https://images.aatbio.com/dataset/ic50/activin-receptor-type-1_b09975fc05fd0f6f88376af3b795bf22.svg) | 3-Phenyl-6-quinolin-4-ylquinazolin-4-one | IC50 | 431.0 [1] |
![](https://images.aatbio.com/dataset/ic50/activin-receptor-type-1_683934066721698a529e4ed2e890721c.svg) | 3,8-Dimethyl-7-quinolin-4-yl-2H-isoquinolin-1-one | IC50 | 10.0 [1] |
![](https://images.aatbio.com/dataset/ic50/activin-receptor-type-1_36ef5f1208ba6ac09f10e34c68ed37ce.svg) | 2-Methyl-6-quinolin-4-yl-3H-quinazolin-4-one | IC50 | 248.0 [1] |
![](https://images.aatbio.com/dataset/ic50/activin-receptor-type-1_eb151864cf94da7e0d6b04019baebc12.svg) | 2-Ethyl-5-methyl-6-quinolin-4-yl-3H-quinazolin-4-one | IC50 | 91.0 [1] |
![](https://images.aatbio.com/dataset/ic50/activin-receptor-type-1_6f22aa38d9835cd86ef0d49546abfbdd.svg) | 3-Methyl-6-quinolin-5-ylquinazolin-4-one | IC50 | 383.0 [1] |
![](https://images.aatbio.com/dataset/ic50/activin-receptor-type-1_5b5854f345ba460c5969ca46210d9a7b.svg) | 6-(5-Cyclopropyl-1H-pyrazol-4-yl)-3H-quinazolin-4-one | IC50 | 386.0 [1] |
![](https://images.aatbio.com/dataset/ic50/activin-receptor-type-1_7730a10f6996edf8e7943a45ce136ecf.svg) | 4-[2-[4-(3-Quinolin-4-ylpyrazolo[1,5-a]pyrimidin-6-yl)phenoxy]ethyl]morpholine | IC50 | 42.77 [1] |
![](https://images.aatbio.com/dataset/ic50/activin-receptor-type-1_eaa73d75510a6c5cdc1b0a54850d8724.svg) | 6-(4-Methoxyphenyl)-3-(1H-pyrazol-4-yl)pyrazolo[1,5-a]pyrimidine | IC50 | 110.0 [1] |
![](https://images.aatbio.com/dataset/ic50/activin-receptor-type-1_2abc1ac9e2da534b713054f6bbfee584.svg) | 6-(4-Piperazin-1-ylphenyl)-3-(1H-pyrazol-4-yl)pyrazolo[1,5-a]pyrimidine | IC50 | 43.0 [1] |
![](https://images.aatbio.com/dataset/ic50/activin-receptor-type-1_607d44385547ac9557ccd2144772c3c8.svg) | 3-Phenyl-6-(4-piperazin-1-ylphenyl)pyrazolo[1,5-a]pyrimidine | IC50 | 40.72 [1] |
![](https://images.aatbio.com/dataset/ic50/activin-receptor-type-1_f980e35cc5a89e33324ed62d29bf7e45.svg) | 2-N-(1H-Indazol-6-yl)-4-N-(2,2,2-trifluoroethyl)furo[3,2-d]pyrimidine-2,4-diamine | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/activin-receptor-type-1_ea7d68d5631badf4d76195468cfe148a.svg) | N~4~-Cyclopropyl-N~2~-(3-Methyl-1h-Indazol-6-Yl)furo[3,2-D]pyrimidine-2,4-Diamine | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/activin-receptor-type-1_4c1c8e479c2e24660577929dfcea7599.svg) | 1-[4-[3-[4-Amino-5-[2-fluoro-5-[[(2S)-oxolan-2-yl]methoxy]phenyl]pyrrolo[2,3-d]pyrimidin-7-yl]cyclobutyl]piperazin-1-yl]ethanone | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/activin-receptor-type-1_f8ee55f6cac6bc1babf9b394bab747fe.svg) | 2-N-(3-Chloro-4-morpholin-4-ylphenyl)-4-N-(2,2,2-trifluoroethyl)furo[3,2-d]pyrimidine-2,4-diamine | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/activin-receptor-type-1_335e463d5d679d47b0cd52f71ccae0e6.svg) | 1-{4-[5-(3,4,5-Trimethoxyphenyl)pyridin-3-Yl]phenyl}piperazine | IC50 | 15.0 [1] |
![](https://images.aatbio.com/dataset/ic50/activin-receptor-type-1_5711133ca718b66fa0cee0f039b3b462.svg) | 4-Amino-8-(5-Methyl-1h-Indazol-6-Yl)cinnoline-3-Carboxamide | IC50 | 7.0 [1] |
![](https://images.aatbio.com/dataset/ic50/activin-receptor-type-1_ca2a95447671d6df953b2d5e22064d52.svg) | 5-(4-Piperazin-1-ylphenyl)-3-(3,4,5-trimethoxyphenyl)pyridin-2-amine | IC50 | 10.0 [1] |
![](https://images.aatbio.com/dataset/ic50/activin-receptor-type-1_5f828372bf2a58f07ed46e53b21ac79d.svg) | N-[4-[(6-Chloro-[1,3]dioxolo[4,5-B]pyridin-7-Yl)amino]-2-Pyridyl]cyclopropanecarboxamide | IC50 | 1.2 [1] |
![](https://images.aatbio.com/dataset/ic50/activin-receptor-type-1_d9834fa2bdb30c87803e1700bd33f500.svg) | N,N-Dimethyl-3-[4-(3-quinolin-4-ylpyrazolo[1,5-a]pyrimidin-6-yl)phenoxy]propan-1-amine | IC50 | 26.68 [1] |