 | 1-(5-Amino-1H-1,2,4-triazol-3-yl)-N-[2-(4-chlorophenyl)ethyl]-N-(2-methylpropyl)piperidin-4-amine | IC50 | 14.2 [1] |
 | 1-(5-Amino-1H-1,2,4-triazol-3-yl)-N-[2-(4-chlorophenyl)ethyl]-N-(2-methylpropyl)piperidin-4-amine | Ki | 13.5 [1] |
 | 5-{4-[2-(4-Bromophenoxy)ethyl]piperazin-1-Yl}-4h-1,2,4-Triazol-3-Amine | IC50 | 210.0 [1], 5450.0 [2] |
 | Acetazolamide | IC50 | 1000000.0 [1] |
 | Kinetin | IC50 | 1000000.0 [1] |
 | Allosamidin | IC50 | 40.0 [1] |
 | 8-Chlorotheophylline | IC50 | 2500000.0 [1] |
 | Argifin | IC50 | 4500.0 [1] |
 | 2-[(3-Amino-4-methyl-6-phenylfuro[2,3-b]pyridin-2-yl)carbonyl]-N-methyl-1-hydrazinecarbothioamide | IC50 | 30000.0 [1] |
 | 2-Piperazin-1-ylnicotinamide | IC50 | 101700.0 [1] |
 | 2-Methyl-3-{[4-(Pyridin-2-Yl)piperazin-1-Yl]methyl}-1h-Indole | IC50 | 700.0 [1] |
 | 1-[1-(5-Amino-1H-1,2,4-triazol-3-yl)piperidin-4-yl]-3-(4-bromophenyl)urea | IC50 | 100000.0 [1] |
 | 1-(5-Amino-1H-1,2,4-triazol-3-yl)-N-[(4-bromophenyl)methyl]piperidine-4-carboxamide | IC50 | 100000.0 [1] |
 | 1-(5-Amino-1H-1,2,4-triazol-3-yl)-N-[2-(4-bromophenyl)ethyl]-N-ethylpiperidin-4-amine | IC50 | 73.0 [1] |
 | N-[[1-(5-Amino-1H-1,2,4-triazol-3-yl)piperidin-4-yl]methyl]-4-bromobenzamide | IC50 | 100000.0 [1] |
 | N-[1-(5-Amino-1H-1,2,4-triazol-3-yl)piperidin-4-yl]-1-(4-bromophenyl)methanesulfonamide | IC50 | 3325.0 [1] |
 | 1-(5-Amino-1H-1,2,4-triazol-3-yl)-N-benzyl-N-[2-(4-chlorophenyl)ethyl]piperidin-4-amine | IC50 | 5.4 [1] |
 | 1-(5-Amino-1H-1,2,4-triazol-3-yl)-N-[2-(4-chlorophenyl)ethyl]-N-ethylpiperidin-4-amine | IC50 | 182.0 [1] |
 | 1-(5-Amino-1H-1,2,4-triazol-3-yl)-N-[2-(4-cyclopropylphenyl)ethyl]-N-methylpiperidin-4-amine | IC50 | 1545.0 [1] |
 | N-[1-(5-Amino-1H-1,2,4-triazol-3-yl)piperidin-4-yl]-2-(4-bromophenyl)acetamide | IC50 | 100000.0 [1] |
 | 1-(5-Amino-1H-1,2,4-triazol-3-yl)-N-[2-(4-bromophenyl)ethyl]-N-(2-methylpropyl)piperidin-4-amine | IC50 | 8.7 [1] |
 | 1-(5-Amino-1H-1,2,4-triazol-3-yl)-N-[2-(4-chlorophenyl)ethyl]-N-(naphthalen-1-ylmethyl)piperidin-4-amine | IC50 | 3.4 [1] |
 | 1-(5-Amino-1H-1,2,4-triazol-3-yl)-N-methyl-N-(2-phenylethyl)piperidin-4-amine | IC50 | 18450.0 [1] |
 | 1-(5-Amino-1H-1,2,4-triazol-3-yl)-N-[2-(4-bromophenyl)ethyl]-N-methylpiperidin-4-amine | IC50 | 348.0 [1] |
 | 1-(5-Amino-1H-1,2,4-triazol-3-yl)-N-[2-(4-chlorophenyl)ethyl]-N-methylpiperidin-4-amine | IC50 | 660.0 [1] |
 | 1-(5-Amino-1H-1,2,4-triazol-3-yl)-N-[2-(4-ethylphenyl)ethyl]-N-methylpiperidin-4-amine | IC50 | 970.0 [1] |
 | 1-(5-Amino-1H-1,2,4-triazol-3-yl)-N-[2-(4-tert-butylphenyl)ethyl]-N-methylpiperidin-4-amine | IC50 | 13200.0 [1] |
 | 1-(5-Amino-1H-1,2,4-triazol-3-yl)-N-methyl-N-[2-(4-methylphenyl)ethyl]piperidin-4-amine | IC50 | 1111.0 [1] |
 | 3-[4-[[(4-Bromophenyl)methyl-methylamino]methyl]piperidin-1-yl]-1H-1,2,4-triazol-5-amine | IC50 | 100000.0 [1] |
 | 1-(5-Amino-1H-1,2,4-triazol-3-yl)-N-[2-(4-chlorophenyl)ethyl]-N-propan-2-ylpiperidin-4-amine | IC50 | 134.0 [1] |
 | 1-(5-Amino-1H-1,2,4-triazol-3-yl)-N-methyl-N-[2-(4-propan-2-ylphenyl)ethyl]piperidin-4-amine | IC50 | 4137.0 [1] |
 | 1-(5-Amino-1H-1,2,4-triazol-3-yl)-N-[2-(4-chlorophenyl)ethyl]-N-[(2-chlorophenyl)methyl]piperidin-4-amine | IC50 | 3.5 [1] |
 | 1-(5-Amino-1H-1,2,4-triazol-3-yl)-N-[2-(2,4-dichlorophenyl)ethyl]-N-methylpiperidin-4-amine | IC50 | 2025.0 [1] |
 | N-[1-(5-Amino-1H-1,2,4-triazol-3-yl)piperidin-4-yl]-1-(4-bromophenyl)-N-methylmethanesulfonamide | IC50 | 100000.0 [1] |
 | 1-(5-Amino-1H-1,2,4-triazol-3-yl)-N-[2-(4-chlorophenyl)ethyl]-N-(cyclohexylmethyl)piperidin-4-amine | IC50 | 8.7 [1] |
 | 1-[4-(5-Amino-1H-1,2,4-triazol-3-yl)piperazin-1-yl]-2-(4-bromophenoxy)ethanone | IC50 | 12250.0 [1] |
 | 1-[(E)-(3-Ethoxy-4-hydroxy-5-nitrophenyl)methylideneamino]-3-prop-2-enylthiourea | IC50 | 100000.0 [1] |
 | 1,2-Bis[(E)-furan-2-ylmethylideneamino]guanidine | IC50 | 15000.0 [1] |
 | N-({4-[(2,6-Dimethoxypyrimidin-4-yl)sulfamoyl]phenyl}carbamothioyl)cyclopropanecarboxamide | IC50 | 100000.0 [1] |
 | 4-(4-Chlorophenyl)piperazine-1-carboximidamide | IC50 | 13000.0 [1] |
 | N-[[4-[(5-Methyl-1,2-oxazol-3-yl)sulfamoyl]phenyl]carbamothioyl]prop-2-enamide | IC50 | 80000.0 [1] |
 | N-Ethyl-2-(4-methylpiperazin-1-yl)pyridine-3-carboxamide | IC50 | 22000.0 [1] |
 | N-[(Z)-3-(2-Carbamothioylhydrazinyl)-1-[4-(dimethylamino)phenyl]-3-oxoprop-1-en-2-yl]benzamide | IC50 | 4000.0 [1] |
 | N-[(2-Phenyl-1,3-benzoxazol-5-yl)carbamothioyl]propanamide | IC50 | 40000.0 [1] |