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20S proteasome Inhibitors (IC50, Ki)

Structure
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Compound Name
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Standard Type
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Standard Values (in nM)
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▼
Z-Leu-leu-leu-alIC5068.0 [1], 1400.0 [2], 4500.0 [3]
Tyropeptin AIC50140.0 [1], 5000.0 [2], 68000.0 [3]
(2S)-2-[[(2S)-3-(4-Methoxyphenyl)-2-[(2-naphthalen-1-ylacetyl)amino]propanoyl]amino]-N-[1-(4-methoxyphenyl)-3-oxopropan-2-yl]-3-methylbutanamideIC5027.0 [1], 100000.0 [2]
(2S)-2-[[(2S)-3-(4-Hydroxyphenyl)-2-[(2-naphthalen-1-ylacetyl)amino]propanoyl]amino]-N-[1-(4-hydroxyphenyl)-3-oxopropan-2-yl]-3-methylbutanamideIC507.0 [1], 1200.0 [2], 4900.0 [3]
N-[(2S)-3-(4-Hydroxyphenyl)-1-[[(2S)-1-[[1-(4-hydroxyphenyl)-3-oxopropan-2-yl]amino]-3-methyl-1-oxobutan-2-yl]amino]-1-oxopropan-2-yl]hexanamideIC5037.0 [1], 2000.0 [2], 20000.0 [3]
Tyropeptin A-4IC50330.0 [1], 3000.0 [2], 17000.0 [3]
(2S)-2-[[(2S)-3-(4-Hydroxyphenyl)-2-(3-methylbutanoylamino)propanoyl]amino]-N-[1-(4-methoxyphenyl)-3-oxopropan-2-yl]-3-methylbutanamideIC50190.0 [1], 21000.0 [2]
(2S)-2-[[(2S)-3-(4-Methoxyphenyl)-2-(3-methylbutanoylamino)propanoyl]amino]-N-[1-(4-methoxyphenyl)-3-oxopropan-2-yl]-3-methylbutanamideIC50120.0 [1], 37000.0 [2], 56000.0 [3]
(2S)-2-[[(2S)-3-(4-Hydroxyphenyl)-2-[(2-naphthalen-1-ylacetyl)amino]propanoyl]amino]-N-[1-(4-methoxyphenyl)-3-oxopropan-2-yl]-3-methylbutanamideIC5018.0 [1], 6000.0 [2], 38000.0 [3]
(2S)-N-[1-(4-Hydroxyphenyl)-3-oxopropan-2-yl]-2-[[(2S)-3-(4-methoxyphenyl)-2-[(2-naphthalen-1-ylacetyl)amino]propanoyl]amino]-3-methylbutanamideIC5020.0 [1], 6000.0 [2], 31000.0 [3]
(2S)-N-[1-(4-Hydroxyphenyl)-3-oxopropan-2-yl]-2-[[(2S)-3-(4-hydroxyphenyl)-2-[(2-phenylacetyl)amino]propanoyl]amino]-3-methylbutanamideIC5027.0 [1], 2000.0 [2], 16000.0 [3]
(2S)-2-[[(2S)-3-(4-Hydroxyphenyl)-2-[(2-naphthalen-2-ylacetyl)amino]propanoyl]amino]-N-[1-(4-hydroxyphenyl)-3-oxopropan-2-yl]-3-methylbutanamideIC5014.0 [1], 700.0 [2], 4700.0 [3]
(2S)-2-[[(2S)-2-[[2-(Dimethylamino)acetyl]amino]-3-(4-methoxyphenyl)propanoyl]amino]-N-[(2S)-1-(4-methoxyphenyl)-3-oxopropan-2-yl]-3-methylbutanamideIC501200.0 [1], 7800.0 [2], 100000.0 [3]
LactacystinIC50259.0 [1]
CarfilzomibIC5010.0 [1]
Cinnabaramide AIC501.0 [1]
Cinnabaramide BIC50245.0 [1]
Cinnabaramide DIC50100.0 [1]
Cinnabaramide FIC506.0 [1]
Cinnabaramide EIC50136.0 [1]
Cinnabaramide GIC500.6 [1]
Cinnabaramide CIC5012.0 [1]
Items per page: 1 - 10 of 22
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References

This online tool may be cited as follows

MLA

"Quest Database™ 20S proteasome Inhibitors (IC50, Ki)." AAT Bioquest, Inc., 19 Feb. 2025, https://www.aatbio.com/data-sets/20s-proteasome-inhibitors-ic50-ki.

APA

AAT Bioquest, Inc. (2025, February 19). Quest Database™ 20S proteasome Inhibitors (IC50, Ki). AAT Bioquest. https://www.aatbio.com/data-sets/20s-proteasome-inhibitors-ic50-ki.
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